|
Asymmetric Synthesis of Quinoline-Naphthalene Atropisomers by Central-to-Axial Chirality Conversion 2020-10-30 |
|
1 |
|
Palladium-Catalyzed Chemoselective Aminomethylative Cyclization and Aromatizing Allylic Amination: Access to Functionalized Naphthalenes 2020-10-30 |
|
1 |
|
Chiral Electron-Rich PNP Ligand with a Phospholane Motif: Structural Features and Application in Asymmetric Hydrogenation 2020-10-29 |
|
0.95 |
|
Nickel-Catalyzed Three-Component Reductive Alkylacylation of Electron-Deficient Activated Alkenes 2020-10-29 |
|
1 |
|
Total Synthesis and Immunological Evaluation of the Tri-d-glycero-d-manno-heptose Antigen of the Lipopolysaccharide as a Vaccine Candidate against Helicobacter pylori 2020-10-29 |
|
1 |
|
A CTV Analogue: Arene-Persubstituted Cyclotrixylohydroquinoylene and Its Derivatives 2020-10-28 |
|
1 |
|
Aaptodines A–D, Spiro Naphthyridine–Furooxazoloquinoline Hybrid Alkaloids from the Sponge Aaptos suberitoides 2020-10-28 |
|
0.71 |
|
Visible-Light-Promoted Regioselective 1,3-Fluoroallylation of gem-Difluorocyclopropanes 2020-10-28 |
|
1 |
|
Chemoselective Perfluoromethylation of Thio- and Selenoamides 2020-10-27 |
|
1 |
|
Cu(II)/Iodine(III) Oxide Dimerization of Heterocyclic Ketene Aminals: Tandem TEMPO Oxidation for the Highly Selective Synthesis of Functionalized 2H-Pyrrolo[1,2-a]imidazol-7(3H)-ones 2020-10-27 |
|
1 |
|
Dual Nickel- and Photoredox-Catalyzed Reductive Cross-Coupling of Aryl Halides with Dichloromethane via a Radical Process 2020-10-27 |
|
1 |
|
Modular Synthesis of Drimane Meroterpenoids Leveraging Decarboxylative Borylation and Suzuki Coupling 2020-10-27 |
|
1 |
|
Asymmetric Total Synthesis and Assignment of Absolute Configuration of Arbornamine 2020-10-26 |
|
1 |
|
Deciphering the Biosynthetic Mechanism of Pelletierine in Lycopodium Alkaloid Biosynthesis 2020-10-26 |
|
0.77 |
|
Synthesis and Biological Evaluation of N-Aminoimidazolidin-2-one-Containing Angiotensin-(1–7) Peptidomimetics 2020-10-26 |
|
1 |
|
Generation of Carbocations under Photoredox Catalysis: Electrophilic Aromatic Substitution with 1-Fluoroalkylbenzyl Bromides 2020-10-23 |
|
0.83 |
|
Nickel-Catalyzed Highly Selective Hydroalkenylation of Alkenyl Boronic Esters to Access Allyl Boron 2020-10-22 |
|
1 |
|
Triphenylphosphine-Catalyzed Alkylative Iododecarboxylation with Lithium Iodide under Visible Light 2020-10-22 |
|
0.83 |
|
Biomimetic Total Synthesis of (±)-Carbocyclinone-534 Reveals Its Biosynthetic Pathway 2020-10-21 |
|
1 |
|
Cyanide-Free Synthesis of Glycosyl Carboxylic Acids and Application for the Synthesis of Scleropentaside A 2020-10-21 |
|
1 |
|
Enantioselective Synthesis of 4-Cyanotetrahydroquinolines via Ni-Catalyzed Hydrocyanation of 1,2-Dihydroquinolines 2020-10-21 |
|
1 |
|
Palladium-Catalyzed Hydroxylation of Aryl Halides with Boric Acid 2020-10-21 |
|
1 |
|
Diastereodivergent Synthesis of α-Chiral Tertiary Azides through Catalytic Asymmetric Michael Addition 2020-10-20 |
|
1 |
|
A Bispidine-Based Chiral Amine Catalyst for Asymmetric Mannich Reaction of Ketones with Isatin Ketimines 2020-10-19 |
|
1 |
|
Cu-Catalyzed Regioselective C–H Alkylation of Benzimidazoles with Aromatic Alkenes 2020-10-19 |
|
1 |
|
Peptide Modification via N-Terminal-Residue-Directed γ-C(sp3)–H Arylation 2020-10-19 |
|
1 |
|
Relay Palladium/Copper Catalysis Enabled Silylative [5 + 1] Benzannulation Using Terminal Alkynes as One-Carbon Units 2020-10-19 |
|
1 |
|
Synthetic Investigation toward QS-21 Analogues 2020-10-19 |
|
1 |
|
Switching of C–C and C–N Coupling/Cleavage for Hypersensitive Detection of Cu2+ by a Catalytically Mediated 2-Aminoimidazolyl-Tailored Six-Membered Rhodamine Probe 2020-10-16 |
|
1 |
|
Dichloroacetophenone Derivatives: A Class of Bioconjugation Reagents for Disulfide Bridging 2020-10-14 |
|
0.75 |
|
Nickel(II)-Catalyzed Oxygen Transfer Reaction of N-Vinyl Nitrones to Prepare 2-(Pyridin-2-yl)ethanols 2020-10-14 |
|
1 |
|
Pd-Catalyzed Domino Imidoylation/Heck/C(sp2)–H Cyclization: Isocyanide Relay Strategy toward Tricyclic-Fused Heterocycles Containing an All-Carbon Quaternary Center 2020-10-14 |
|
1 |
|
Rh-Catalyzed Annulation of Benzoic Acids, Formaldehyde, and Malonates via ortho-Hydroarylation to Indanones 2020-10-14 |
|
1 |
|
A Series of Deoxyfluorination Reagents Featuring OCF2 Functional Groups 2020-10-13 |
|
1 |
|
Construction of β-Quaternary α,α-Difluoroketones via Catalytic Nucleophilic Substitution of Tertiary Alcohols with Difluoroenoxysilanes 2020-10-13 |
|
1 |
|
Iodine-Promoted Multicomponent Synthesis of 2,4-Diamino-1,3,5-triazines 2020-10-13 |
|
1 |
|
Light-Mediated Difluoromethylthiolation of Aldehydes with a Hydrogen Atom Transfer Photocatalyst 2020-10-13 |
|
1 |
|
NHC/Copper-Cocatalyzed [4 + 3] Annulations of Salicylaldehydes with Aziridines for the Synthesis of 1,4-Benzoxazepinones 2020-10-13 |
|
1 |
|
Synthesis of C4-Substituted Indoles via a Catellani and C–N Bond Activation Strategy 2020-10-13 |
|
1 |
|
Visible-Light-Mediated Hydroacylation of Azobenzenes with α-Keto Acids 2020-10-13 |
|
1 |
|
A Construction of α-Alkenyl Lactones via Reduction Radical Cascade Reaction of Allyl Alcohols and Acetylenic Acids 2020-10-12 |
|
1 |
|
Asymmetric Transfer Hydrogenation of Densely Functionalized Diheteroaryl and Diaryl Ketones by a Ru-Catalyst of Minimal Stereogenicity 2020-10-12 |
|
1 |
|
Chemical Synthesis of Homogeneous Human E-Cadherin N-Linked Glycopeptides: Stereoselective Convergent Glycosylation and Chemoselective Solid-Phase Aspartylation 2020-10-12 |
|
0.21 |
|
Direct Electrochemical Defluorinative Carboxylation of gem-Difluoroalkenes with Carbon Dioxide 2020-10-12 |
|
1 |
|
Highly Enantioselective Synthesis of Monofluoroalkenes by Rhodium-Catalyzed Asymmetric Arylation/Defluorination of Allyl Difluorides 2020-10-12 |
|
0.80 |
|
Nickel-Catalyzed Asymmetric Transfer Hydrogenation and α-Selective Deuteration of N-Sulfonyl Imines with Alcohols: Access to α-Deuterated Chiral Amines 2020-10-12 |
|
1 |
|
P(NMe2)3-Mediated Umpolung Spirocyclopropanation Reaction of p-Quinone Methides: Diastereoselective Synthesis of Spirocyclopropane-Cyclohexadienones 2020-10-12 |
|
1 |
|
Radical Tandem Bicyclization Triggered by the α-Position of α,β-Unsaturated Ketones Bearing Nonterminal 1,6-Enynes: Synthesis of the 5H-Benzo[a]fluoren-5-one Skeleton 2020-10-12 |
|
1 |
|
Reductive CO2 Fixation via the Selective Formation of C–C Bonds: Bridging Enaminones and Synthesis of 1,4-Dihydropyridines 2020-10-12 |
|
1 |
|
Unconventional Transformation of the Two Carbonyl Groups in 4,4′,5,5′-Tetrachloro-10H,10′H-[9,9′-bianthracenylidene]-10,10′-dione into Diallenes 2020-10-12 |
|
1 |
|
Vinylogous Elimination/C–H Functionalization/Allylation Cascade Reaction of Allenoate Adducts: Synthesis of Ring-Fused Dihydropyridinones 2020-10-12 |
|
1 |
|
General Synthesis of α-Alkyl Ynones from Morpholine Amides and 1-Copper(I) Alkynes Promoted by Triflic Anhydride 2020-10-09 |
|
1 |
|
In(OTf)3-Catalyzed Synthesis of 2,3-Dihydro-1H-benzo[e]indoles and 2,3-Dihydrobenzofurans via [3 + 2] Annulation 2020-10-09 |
|
1 |
|
Combined KOH/BEt3 Catalyst for Selective Deaminative Hydroboration of Aromatic Carboxamides for Construction of Luminophores 2020-10-07 |
|
1 |
|
Copper-Catalyzed Oxidative Fragmentation of Alkynes with NFSI Provides Aryl Ketones 2020-10-07 |
|
1 |
|
Stereodivergent Synthesis of Alkenylpyridines via Pd/Cu Catalyzed C–H Alkenylation of Pyridinium Salts with Alkynes 2020-10-07 |
|
1 |
|
Transition-Metal Free Chemoselective Hydroxylation and Hydroxylation–Deuteration of Heterobenzylic Methylenes 2020-10-07 |
|
1 |
|
6,12-Dihydro-6,12-diboradibenzo[def,mno]chrysene: A Doubly Boron-Doped Polycyclic Aromatic Hydrocarbon for Organic Light Emitting Diodes by a One-Pot Synthesis 2020-10-06 |
|
1 |
|
Aminothiolation of α-Bromocinnamaldehydes to Access Imidazo[2,1-b]thiazoles by Incorporation of Two Distinct Photoinduced Processes 2020-10-06 |
|
1 |
|
Copper-Catalyzed Aerobic Cyclization of β,γ-Unsaturated Hydrazones with Concomitant C═C Bond Cleavage 2020-10-06 |
|
1 |
|
Scocycamides, a Pair of Macrocyclic Dicaffeoylspermidines with Butyrylcholinesterase Inhibition and Antioxidation Activity from the Roots of Scopolia tangutica 2020-10-06 |
|
1 |
|
Synthesis of Heterobiaryl 4-Aryl Furans through a Base-Promoted Decarboxylative Propargylation/Cycloisomerization Annulation 2020-10-06 |
|
1 |
|
γ-Difluoroalkylation: Synthesis of γ-Difluoroalkyl-α,β-Unsaturated Esters via Photoredox NHC-Catalyzed Radical Reaction 2020-10-06 |
|
1 |
|
The Biomimetic Total Syntheses of the Antiplasmodial Tomentosones A and B 2020-10-05 |
|
1 |
|
Annulation of Diaryl(aryl)phosphenes and Cyclic Imines to Access Benzo-δ-phospholactams 2020-10-02 |
|
1 |
|
Nickel-Catalyzed Cyanation of Unactivated Alkyl Sulfonates with Zn(CN)2 2020-10-02 |
|
1 |
|
Ustethylin Biosynthesis Implies Phenethyl Derivative Formation in Aspergillus ustus 2020-10-02 |
|
0.33 |
|
Access to Dibenzofurans through Dimerization/Trimerization of Cyclohexanones Followed by Dehydroaromatization 2020-10-01 |
|
1 |
|
Bisaspochalasins A–C: Three Cytochalasan Homodimers with Highly Fused Ring System from an Endophytic Aspergillus flavipes 2020-10-01 |
|
1 |
|
Longisglucinols A–C, Structurally Intriguing Polycyclic Polyprenylated Acylphloroglucinols with Anti-inflammatory Activity from Hypericum longistylum 2020-10-01 |
|
1 |
|
Photochemical Decarboxylative C(sp3)–X Coupling Facilitated by Weak Interaction of N-Heterocyclic Carbene 2020-10-01 |
|
1 |
|
Polysulfuration via a Bilateral Thiamine Disulfurating Reagent 2020-10-01 |
|
1 |
|
Cleavage of Aromatic C–O Bonds via Intramolecular SNAr Reaction and Preparation of P,C,Axial-Stereogenic Menthyl Phosphine Derivatives 2020-09-30 |
|
1 |
|
Copper-Catalyzed Selective 1,2-Difunctionalization of N-Heteroaromatics through Cascade C–N/C═C/C═O Bond Formation 2020-09-30 |
|
1 |
|
Palladium-Catalyzed Addition/Cyclization of (2-Hydroxyaryl)boronic Acids with Alkynylphosphonates: Access to Phosphacoumarins 2020-09-30 |
|
1 |
|
Access to Cycloalkeno[c]-Fused Pyridines via Pd-Catalyzed C(sp2)–H Activation and Cyclization of N-Acetyl Hydrazones of Acylcycloalkenes with Vinyl Azides 2020-09-29 |
|
1 |
|
B(C6F5)3-Catalyzed β-Functionalization of Pyrrolidines Using Isatins via Borrowing Hydrogen: Divergent Access to Substituted Pyrrolidines and Pyrroles 2020-09-29 |
|
1 |
|
Carboxyl-Assisted meta-Selective C–H Functionalizations of Benzylsulfonamides 2020-09-29 |
|
1 |
|
Chiral Hydroxytetraphenylene–Boron Complex Catalyzed Asymmetric Diels–Alder Cycloaddition of 2′-Hydroxychalcones 2020-09-29 |
|
1 |
|
Cu-Catalyzed o-Amino Benzofuranthioether Formation from N-Tosylhydrazone-Bearing Thiocarbamates and Arylative Electrophiles 2020-09-29 |
|
1 |
|
Difluoroisoxazolacetophenone: A Difluoroalkylation Reagent for Organocatalytic Vinylogous Nitroaldol Reactions of 1,2-Diketones 2020-09-29 |
|
1 |
|
Euphopias A–C: Three Rearranged Jatrophane Diterpenoids with Tricyclo[8.3.0.02,7]tridecane and Tetracyclo[11.3.0.02,10.03,7]hexadecane Cores from Euphorbia helioscopia 2020-09-29 |
|
1 |
|
Organocatalytic Regio- and Enantioselective 1,8-Additions of Nitrogen and Sulfur Nucleophiles to 6-Methylene-6H-indoles 2020-09-29 |
|
1 |
|
Silver-Catalyzed para-Selective Amination and Aminative Dearomatization of Phenols with Azodicarboxylates in Water 2020-09-29 |
|
1 |
|
Synthesis of l-glycero- and d-glycero-d-manno-Heptose Building Blocks for Stereoselective Assembly of the Lipopolysaccharide Core Trisaccharide of Vibrio parahemolyticus O2 2020-09-29 |
|
1 |
|
Unconventional [2 + 3] Cyclization Involving [1,4]-Sulfonyl Transfer to Construct Polysubstituted Fluorazones as Inhibitors of Indoleamine 2,3-Dioxygenase 1 2020-09-29 |
|
1 |
|
Synthesis of Substituted Naphtho[1,8-bc]thiopyrans by Sulfhydryl-Directed Rhodium-Catalyzed peri-Selective C–H Bond Activation and Cyclization of Naphthalene-1-thiols 2020-09-28 |
|
1 |
|
Chiral Calcium Phosphate Catalyzed Enantioselective Amination of 3-Aryl-2-benzofuranones 2020-09-24 |
|
1 |
|
Metal-Free Radical-Mediated C(sp3)–H Heteroarylation of Alkanes 2020-09-24 |
|
1 |
|
Strategic Construction of Ethene-Bridged BODIPY Arrays with Absorption Bands Reaching the Near-Infrared II Region 2020-09-24 |
|
1 |
|
Thianthrenation-Enabled α-Arylation of Carbonyl Compounds with Arenes 2020-09-24 |
|
1 |
|
Catalytic Asymmetric Synthesis of Atropisomeric Nitrones: Versatile Intermediate for Axially Chiral Biaryls 2020-09-23 |
|
1 |
|
Catalytic Direct Construction of Cyano-tetrazoles 2020-09-23 |
|
1 |
|
Chalcogenide-Catalyzed Intermolecular Electrophilic Thio- and Halofunctionalization of gem-Difluoroalkenes: Construction of Diverse Difluoroalkyl Sulfides and Halides 2020-09-23 |
|
1 |
|
Copper-Catalyzed Anti-Markovnikov Hydrosilylation of Terminal Alkynes 2020-09-23 |
|
1 |
|
NHC-Catalyzed Enantioselective [3 + 3] Annulation to Construct 5,6-Dihydropyrimidin-4-ones 2020-09-23 |
|
1 |
|
Organocatalytic Enantioselective Conjugate Alkynylation of β-Aminoenones: Access to Chiral β-Alkynyl-β-Amino Carbonyl Derivatives 2020-09-23 |
|
1 |
|
Rh(III)-Catalyzed [3 + 2] Spirocyclization of 2H-Imidazoles with 1,3-Diynes for the Synthesis of Spiro-[imidazole-indene] Derivatives 2020-09-23 |
|
1 |
|
Synergistic N-Heterocyclic Carbene/Palladium-Catalyzed [3 + 2] Annulation of Vinyl Enolates with 1-Tosyl-2-vinylaziridine 2020-09-23 |
|
1 |
|
Vinyl Sulfonium Salts as the Radical Acceptor for Metal-Free Decarboxylative Alkenylation 2020-09-23 |
|
1 |
|
Divergent Synthesis of Trifluoromethyl Sulfoxides and β-SCF3 Carbonyl Compounds by Tandem Trifluoromethylthiolation/Rearrangement of Allylic and Propargylic Alcohols 2020-09-22 |
|
1 |
|
Oligo(5-amino-N-acylanthranilic acids): Amide Bond Formation without Coupling Reagent and Folding upon Binding Anions 2020-09-22 |
|
0.25 |
|
Cage-Monoterpenoid Quinoline Alkaloids with Neurite Growth Promoting Effects from the Fruits of Melodinus yunnanensis 2020-09-21 |
|
0.83 |
|
A Photochemical Dehydrogenative Strategy for Direct and Regioselective Dimerization of BODIPY Dyes 2020-09-18 |
|
1 |
|
Decarboxylative and Deaminative Alkylation of Difluoroenoxysilanes via Photoredox Catalysis: A General Method for Site-Selective Synthesis of Difluoroalkylated Alkanes 2020-09-18 |
|
1 |
|
Pd-Catalyzed C(sp3)–H Biarylation via Transient Directing Group Strategy 2020-09-18 |
|
1 |
|
Ruthenium-Catalyzed Enantioselective Hydrogenation of Hydrazones 2020-09-18 |
|
0.20 |
|
Synthesis of Enantioenriched α,α-Difluoro-β-arylbutanoic Esters by Pd-Catalyzed Asymmetric Hydrogenation 2020-09-18 |
|
1 |
|
Tandem [5 + 2]/[4 + 2] Cycloadditions To Construct the [6–7–6] Tricyclic Skeleton of Icetexane Diterpenes: Total Synthesis of Euolutchuol E, Przewalskine E and Brussonol 2020-09-18 |
|
1 |
|
Asymmetric Dearomative Cascade Multiple Functionalizations of Activated N-Alkylpyridinium and N-Alkylquinolinium Salts 2020-09-17 |
|
1 |
|
Cross-Dehydrogenative Coupling of Strong C(sp3)–H with N-Heteroarenes through Visible-Light-Induced Energy Transfer 2020-09-17 |
|
1 |
|
Photoredox-Catalyzed α-C(sp3)–H Activation of Unprotected Secondary Amines: Facile Access to 1,4-Dicarbonyl Compounds 2020-09-17 |
|
1 |
|
Enantioselective Total Syntheses of Pentacyclic Homoproaporphine Alkaloids 2020-09-16 |
|
1 |
|
Palladium-Catalyzed Oxidative Annulation of Sulfoximines and Arynes by C–H Functionalization as an Approach to Dibenzothiazines 2020-09-16 |
|
1 |
|
Pegaharmols A–B, Axially Chiral β-Carboline-quinazoline Dimers from the Roots of Peganum harmala 2020-09-16 |
|
0.89 |
|
Visible-Light-Mediated Trifluoromethylation/Benzylation of Styrenes Catalyzed by 4-CzIPN 2020-09-16 |
|
1 |
|
Silver-Catalyzed Cascade Cyclization Reaction of Isocyanides with Sulfoxonium Ylides: Synthesis of 3-Aminofurans and 4-Aminoquinolines 2020-09-15 |
|
1 |
|
Mono/Dual Amination of Phenols with Amines in Water 2020-09-11 |
|
1 |
|
Synthesis of Polysubstituted Pyrroles via Silver-Catalyzed Oxidative Radical Addition of Cyclopropanols to Imines 2020-09-11 |
|
1 |
|
CuI/2-Aminopyridine 1-Oxide Catalyzed Amination of Aryl Chlorides with Aliphatic Amines 2020-09-10 |
|
1 |
|
Divergent Synthesis of Bicyclo[3.2.1]octenes and Cyclohexenes via Catalytic Annulations of Nazarov Reagent and Vinyl 1,2-Diketones 2020-09-10 |
|
1 |
|
Nickel-Catalyzed Mizoroki–Heck/Amination Cascade Reactions of o-Dihaloarenes with Allylamines: Synthesis of Indoles 2020-09-10 |
|
1 |
|
Asymmetric Construction of Cyclobutanes via Direct Vinylogous Michael Addition/Cyclization of β,γ-Unsaturated Amides 2020-09-09 |
|
1 |
|
Copper(I)/DDQ-Mediated Double-Dehydrogenative Diels–Alder Reaction of Aryl Butenes with 1,4-Diketones and Indolones 2020-09-09 |
|
1 |
|
Iodonium Ylides as Carbene Precursors in Rh(III)-Catalyzed C–H Activation 2020-09-09 |
|
1 |
|
Silver-Catalyzed Activation of Pyridotriazoles for Formal Intramolecular Carbene Insertion into Vinylic C(sp2)–H Bonds 2020-09-09 |
|
1 |
|
Synthesis and Catalytic Properties of Metal–N-Heterocyclic-Carbene-Decorated Covalent Organic Framework 2020-09-09 |
|
1 |
|
Tuning the Properties of Corannulene-Based Polycyclic Aromatic Hydrocarbons by Varying the Fusing Positions of Corannulene 2020-09-09 |
|
1 |
|
Visible Light-Driven α-Alkylation of N-Aryl tetrahydroisoquinolines Initiated by Electron Donor–Acceptor Complexes 2020-09-09 |
|
1 |
|
Visible-Light-Promoted Site-Selective N1-Alkylation of Benzotriazoles with α-Diazoacetates 2020-09-09 |
|
0.86 |
|
Asymmetric Synthesis of γ-Secondary Amino Alcohols via a Borrowing-Hydrogen Cascade 2020-09-08 |
|
1 |
|
Chlorotrifluoromethylthiolation of Sulfur Ylides for the Formation of Tetrasubstituted Trifluoromethylthiolated Alkenes 2020-09-08 |
|
1 |
|
Controlling Keto–Enol Tautomerism of Ureidopyrimidinone to Generate a Single-Quadruple AADD-DDAA Dimeric Array 2020-09-08 |
|
1 |
|
Iron-Catalyzed Redox-Neutral Radical Cascade Reaction of [60]Fullerene with γ,δ-Unsaturated Oxime Esters: Preparation of Free (N–H) Pyrrolidino[2′,3′:1,2]fullerenes 2020-09-08 |
|
1 |
|
β-Carboline Alkaloids from the Seeds of Peganum harmala and Their Anti-HSV-2 Virus Activities 2020-09-08 |
|
1 |
|
Au(I)-Catalyzed Cyclization/Semipinacol Rearrangement Reaction of Allenes to Construct Quaternary Carbon-Containing Scaffolds 2020-09-04 |
|
1 |
|
Baicalensines A and B, Two Isoquinoline Alkaloids from the Roots of Thalictrum baicalense 2020-09-04 |
|
1 |
|
Visible-Light-Promoted Intramolecular α-Allylation of Aldehydes in the Absence of Sacrificial Hydrogen Acceptors 2020-09-04 |
|
1 |
|
Palladium-Catalyzed [5 + 2] Annulation of Vinylethylene Carbonates with Barbiturate-Derived Alkenes 2020-09-03 |
|
1 |
|
A Role for Isatin Azomethine Imines as a Dipolarophile in Cycloaddition Reactions 2020-09-02 |
|
1 |
|
A Strategy for Amide to β-Oxo Ester Transformation via N-Alkenoxypyridinium Salts as the Activator and H2O as the Nucleophile 2020-09-02 |
|
1 |
|
Splitting Methyl Ketones into Two Parts: Synthesis of 4(3H)-Quinazolinones via Consecutive Cyclization/Ring-Opening Reaction 2020-09-02 |
|
1 |
|
Synthesis of γ-Lactams via Pd(II)-Catalyzed C(sp3)–H Olefination Using a Self-Cleaving Polyfluoroethylsulfinyl Directing Group 2020-09-02 |
|
1 |
|
Solvation-Free Li+ Lewis Acid Enhancing Reaction: Kinetic Study of [5,6]-Li+@PCBM to [6,6]-Li+@PCBM 2020-09-01 |
|
0.33 |
|
Visible-Light-Promoted Photoredox Dehydrogenative Coupling of Phosphines and Thiophenols 2020-09-01 |
|
1 |
|
Zwitterion-Catalyzed Deacylative Dihalogenation of β-Oxo Amides 2020-09-01 |
|
1 |
|
Access to Cyanoimines Enabled by Dual Photoredox/Copper-Catalyzed Cyanation of O-Acyl Oximes 2020-08-31 |
|
1 |
|
Iridium-Catalyzed Asymmetric Hydrogenation of α-Fluoro Ketones via a Dynamic Kinetic Resolution Strategy 2020-08-31 |
|
1 |
|
Visible-Light-Triggered Iodinations Facilitated by Weak Electrostatic Interaction of N-Heterocyclic Carbenes 2020-08-31 |
|
1 |
|
Catalytic Enantioselective Dearomatization/Rearomatization of 2-Nitroindoles to Access 3-Indolyl-3′-Aryl-/Alkyloxindoles: Application in the Formal Synthesis of Cyclotryptamine Alkaloids 2020-08-28 |
|
1 |
|
Directing-Group-Assisted C(sp2)–H Arylsulfonylation from Sulfur Dioxide 2020-08-28 |
|
1 |
|
Palladium-Catalyzed Decarbonylative Heck Coupling of Aromatic Carboxylic Acids with Terminal Alkenes 2020-08-28 |
|
1 |
|
Rapid Access of Alkynyl and Alkenyl Coumarins via a Dipyridinium Methylide and Propargylamine Cascade Reaction 2020-08-28 |
|
1 |
|
Regioselective Direct C–H Trifluoromethylation of Pyridine 2020-08-28 |
|
1 |
|
Synthesis of Indenopyrazole Frameworks via Cascade C–H Functionalization/[3 + 2] Dipolar Cycloaddition/Aromatization Rearrangement Reactions 2020-08-28 |
|
1 |
|
Copper-Mediated Decarboxylative Sulfonylation of Arylacetic Acids with Sodium Sulfinates 2020-08-27 |
|
1 |
|
Electrochemical Alkoxyhalogenation of Alkenes with Organohalides as the Halide Sources via Dehalogenation 2020-08-27 |
|
1 |
|
1,1-Addition of α-C2-Bridged Biphospholes with Alkynes 2020-08-26 |
|
1 |
|
Arylaminomethyl Radical-Initiated Cascade Annulation Reaction of Quinoxalin-2(1H)-ones Catalyzed by Recyclable Photocatalyst Perovskite 2020-08-26 |
|
1 |
|
Chiral Naphthyl-C2-Indole as Scaffold for Phosphine Organocatalysis: Application in Asymmetric Formal [4 + 2] Cycloaddition Reactions 2020-08-26 |
|
1 |
|
Cu(I)-Catalyzed Oxidative Cyclization of Enynamides: Regioselective Access to Cyclopentadiene Frameworks and 2-Aminofurans 2020-08-26 |
|
1 |
|
Ni-Catalyzed Reductive Antiarylative Cyclization of Alkynones 2020-08-26 |
|
1 |
|
Lewis-Acid-Mediated Intramolecular Trifluoromethylthiolation of Alkenes with Phenols: Access to SCF3-Containing Chromane and Dihydrobenzofuran Compounds 2020-08-25 |
|
1 |
|
Terreuspyridine: An Unexpected Pyridine-Fused Meroterpenoid Alkaloid with a Tetracyclic 6/6/6/6 Skeleton from Aspergillus terreus 2020-08-25 |
|
1 |
|
Hemin-Catalyzed Oxidative Phenol-Hydrazone [3+3] Cycloaddition Enables Rapid Construction of 1,3,4-Oxadiazines 2020-08-24 |
|
1 |
|
Total Synthesis of Gastrodinol via Photocatalytic 6π Electrocyclization 2020-08-24 |
|
1 |
|
2-(Dimesitylboryl)phenyl-Substituted [2.2]Paracyclophanes Featuring Intense and Sign-Invertible Circularly Polarized Luminescence 2020-08-21 |
|
1 |
|
C–H Borylation of Diphenylamines through Adamantane-1-carbonyl Auxiliary by BBr3 2020-08-21 |
|
1 |
|
Elucidation of the Tailoring Steps in Julichrome Biosynthesis by Marine Gastropod Mollusk-Associated Streptomyces sampsonii SCSIO 054 2020-08-21 |
|
1 |
|
Hyperfols A and B: Two Highly Modified Polycyclic Polyprenylated Acylphloroglucinols from Hypericum perforatum 2020-08-21 |
|
1 |
|
Lewis-Acid-Catalyzed Asymmetric Alkynylation of Alkynyl 1,2-Diketones: Controllable Formation of 3(2H)-Furanones and α-Hydroxy Ketones 2020-08-21 |
|
1 |
|
Palladium-Catalyzed Tandem C–C Activation/Cyclization Induced by Carbopalladation of Functionalized Nitriles: Synthesis of Benzo Dipyrromethenes 2020-08-21 |
|
1 |
|
Radical-Dual-Difunctionalization and Trifluoromethylative Decarboxylation of Two Different Alkenes 2020-08-21 |
|
1 |
|
Remote C–H Activation Strategy Enables Total Syntheses of Nortriterpenoids (±)-Walsucochin B and (±)-Walsucochinoids M and N 2020-08-21 |
|
1 |
|
Asymmetric Catalytic Synthesis of Epoxides via Three-Component Reaction of Diazoacetates, 2-Oxo-3-ynoates, and Nitrosoarenes 2020-08-20 |
|
1 |
|
Difluorocarbene-Triggered Cyclization: Synthesis of (Hetero)arene-Fused 2,2-Difluoro-2,3-dihydrothiophenes 2020-08-20 |
|
1 |
|
Ligand-Controlled Palladium-Catalyzed Chemoselective Multicomponent Reaction of Olefin-Tethered Aryl Halides, Isocyanides, and Carboxylic Acids: Diversified Synthesis of Imides 2020-08-20 |
|
1 |
|
Phosphine-Catalyzed Stereoselective Tandem Annulation Reaction for the Synthesis of Chromeno[4,3-b]pyrroles 2020-08-20 |
|
1 |
|
Construction of Cyclophane-Braced Peptide Macrocycles via Palladium-Catalyzed Picolinamide-Directed Intramolecular C(sp2)–H Arylation 2020-08-19 |
|
1 |
|
Electrochemically Enabled Sulfonylation of Alkynes with Sodium Sulfinates 2020-08-19 |
|
1 |
|
Ni-Catalyzed Direct Carboxylation of an Unactivated C–H Bond with CO2 2020-08-19 |
|
1 |
|
Acyl Radicals from α-Keto Acids Using a Carbonyl Photocatalyst: Photoredox-Catalyzed Synthesis of Ketones 2020-08-18 |
|
0.83 |
|
Catalytic Asymmetric Three-Component Reaction of 2-Alkynylbenzaldehydes, Amines, and Dimethylphosphonate 2020-08-18 |
|
1 |
|
Chemo- and Diastereoselective Synthesis of Pyrrolidines from Aroylformates and δ-Tosylamino Enones via P(NMe2)3-Mediated Reductive Amination/Base-Catalyzed Michael Addition Cascade 2020-08-18 |
|
1 |
|
Enantioselective Dehydrative γ-Arylation of α-Indolyl Propargylic Alcohols with Phenols: Access to Chiral Tetrasubstituted Allenes and Naphthopyrans 2020-08-18 |
|
1 |
|
Palladium-Catalyzed Secondary Benzylic Imidoylative Reactions 2020-08-18 |
|
1 |
|
Photoinduced Copper-Catalyzed Site-Selective C(sp2)–C(sp) Cross-Coupling via Aryl Sulfonium Salts 2020-08-18 |
|
1 |
|
Ruthenium(II)-Catalyzed C–H Arylation of N,N-Dialkyl Thiobenzamides with Boronic Acids by Sulfur Coordination in 2-MeTHF 2020-08-18 |
|
0.92 |
|
Synthesis of Spiroisoxazolines via TEMPO/NaNO2-Catalyzed Aerobic Oxidative Dearomatization 2020-08-18 |
|
1 |
|
Catalytic Claisen Rearrangement by Intercepting Ketenimines with Propargylic Alcohols: A Strategy to Generate and Transform Ketenimines from Radicals 2020-08-14 |
|
1 |
|
Construction of CF3-Containing Tetrahydropyrano[3,2-b]indoles through DMAP-Catalyzed [4+1]/[3+3] Domino Sequential Annulation 2020-08-14 |
|
1 |
|
Multiturn Hollow Helices: Synthesis and Folding of Long Aromatic Oligoamides 2020-08-14 |
|
0.22 |
|
Selective Synthesis of 2-Indolyl-3-oxoindolines or 2-(2-Aminophenyl)quinolines through Cu(II)- or Bi(III)-Catalyzed Tunable Dimerizations of 2-Alkynylanilines 2020-08-14 |
|
1 |
|
Cu/Ag-Catalyzed Reaction of Azirines with Anthranils: Synthesis of (Quinazolin-2-yl)methanone Derivatives 2020-08-13 |
|
1 |
|
NHC-Catalyzed Asymmetric α-Regioselective [4 + 2] Annulation to Construct α-Alkylidene-δ-lactones 2020-08-13 |
|
1 |
|
Nickel-Catalyzed Reductive Aryl Thiocarbonylation of Alkene via Thioester Group Transfer Strategy 2020-08-13 |
|
1 |
|
Cobalt-Catalyzed Radical Hydrotrifluoroethylation of Styrenes with Trifluoroethyl Iodide 2020-08-12 |
|
1 |
|
Dehydroxylative Fluorination of Tertiary Alcohols 2020-08-12 |
|
0.75 |
|
Phthalaldehyde-Amine Capture Reactions for Bioconjugation and Immobilization of Phthalocyanines 2020-08-12 |
|
1 |
|
Rh(III)-Catalyzed [4 + 2] Annulation of 3-Aryl-5-isoxazolone with Maleimides or Maleic Ester 2020-08-12 |
|
1 |
|
Ruthenium(II)-Catalyzed Regioselective [3 + 2] Spiroannulation of 2H-Imidazoles with 2-Alkynoates 2020-08-12 |
|
1 |
|
Asymmetric Reductive Amination/Ring-Closing Cascade: Direct Synthesis of Enantioenriched Biaryl-Bridged NH Lactams 2020-08-11 |
|
1 |
|
Cu-Catalyzed Direct Amination of Cyclic Amides via C–OH Bond Activation Using DMF 2020-08-11 |
|
1 |
|
Isothiourea-Catalyzed Atroposelective N-Acylation of Sulfonamides 2020-08-11 |
|
0.21 |
|
Ynamide-Mediated Thionoester and Dithioester Syntheses 2020-08-11 |
|
1 |
|
Decarbonylative Suzuki–Miyaura Cross-Coupling of Aroyl Chlorides 2020-08-10 |
|
0.60 |
|
Engineered Biosynthesis of Fungal 4-Quinolone Natural Products 2020-08-10 |
|
0.11 |
|
Metal-Free Chemoselective Reaction of Sulfoxonium Ylides and Thiosulfonates: Diverse Synthesis of 1,4-Diketones, Aryl Sulfursulfoxonium Ylides, and β-Keto Thiosulfones Derivatives 2020-08-10 |
|
1 |
|
Site-Selective Silylation of Arenes Mediated by Thianthrene S-Oxide 2020-08-10 |
|
1 |
|
Synthesis of Bridged Bicyclic Amines by Intramolecular Amination of Remote C–H Bonds: Synergistic Activation by Light and Heat 2020-08-10 |
|
0.09 |
|
Cu-Catalyzed Site-Selective and Enantioselective Ring Opening of Cyclic Diaryliodoniums with 1,2,3-Triazoles 2020-08-07 |
|
1 |
|
Dual Nickel-/Palladium-Catalyzed Reductive Cross-Coupling Reactions between Two Phenol Derivatives 2020-08-07 |
|
0.80 |
|
Nickel-Catalyzed Thiocarbonylation of Arylboronic Acids with Sulfonyl Chlorides for the Synthesis of Thioesters 2020-08-07 |
|
0.88 |
|
Synthesis of Aza-Eight-Membered Ring-Fused Indolines Initiated by Zn-Catalyzed C2 Alkylation of Indoles and Subsequent Base-Promoted Ring Expansion 2020-08-06 |
|
1 |
|
Synthesis of O-Sulfated Human Syndecan-1-like Glyco-polypeptides by Incorporating Peptide Ligation and O-Sulfated Glycopeptide Cassette Strategies 2020-08-06 |
|
0.08 |
|
Bio- and Medicinally Compatible α-Amino-Acid Modification via Merging Photoredox and N-Heterocyclic Carbene Catalysis 2020-08-05 |
|
1 |
|
Organocatalytic Atroposelective Construction of Axially Chiral N-Aryl Benzimidazoles Involving Carbon–Carbon Bond Cleavage 2020-08-05 |
|
1 |
|
Pd/Cu-Catalyzed Domino Cyclization/Deborylation of Alkene-Tethered Carbamoyl Chloride and 1,1-Diborylmethane 2020-08-05 |
|
1 |
|
Asymmetric Transfer Hydrogenation of Unhindered and Non-Electron-Rich 1-Aryl Dihydroisoquinolines with High Enantioselectivity 2020-08-04 |
|
0.33 |
|
Novel Meroterpenoids from Hypericum patulum: Highly Potent Late Nav1.5 Sodium Current Inhibitors 2020-08-04 |
|
0.96 |
|
PIDA-Mediated Rearrangement for the Synthesis of Enantiopure Triazolopyridinones 2020-08-04 |
|
1 |
|
Penicimeroterpenoids A–C, Meroterpenoids with Rearrangement Skeletons from the Marine-Derived Fungus Penicillium sp. SCSIO 41512 2020-08-04 |
|
1 |
|
Rapid Access to Tetracyclic Core of Wortmannin via an Intramolecular Reductive Olefin Coupling Strategy 2020-08-04 |
|
1 |
|
Rationally Designed Self-Immolative Rotaxane Sensor Based on Pillar[5]arene for Fluoride Sensing 2020-08-04 |
|
1 |
|
Silver-Promoted Direct Phosphorylation of Bulky C(sp2)–H Bond to Build Fully Substituted β-Phosphonodehydroamino Acids 2020-08-04 |
|
1 |
|
Tris(4-bromophenyl)aminium Hexachloroantimonate-Initiated Oxidative Povarov-Type Reaction between Glycine Esters and (Cyclopropylidenemethyl)benzenes Using the Counterion as a Chlorine Donor 2020-08-04 |
|
1 |
|
Visible-Light-Induced Pd-Catalyzed Radical Strategy for Constructing C-Vinyl Glycosides 2020-08-04 |
|
1 |
|
Asymmetric Ruthenium-Catalyzed Hydrogenation of Terpyridine-Type N-Heteroarenes: Direct Access to Chiral Tridentate Nitrogen Ligands 2020-08-03 |
|
1 |
|
Selective C-5 Oxidative Radical Silylation of Imidazopyridines Promoted by Lewis Acid 2020-08-03 |
|
1 |
|
Synthesis of Vitamin B12-Antibiotic Conjugates with Greatly Improved Activity against Gram-Negative Bacteria 2020-08-03 |
|
1 |
|
A B2(OH)4-Mediated Synthesis of 2-Substituted Indazolone and Its Application in a DNA-Encoded Library 2020-08-01 |
|
1 |
|
Slicing and Splicing of Bromodifluoro-N-arylacetamides: Dearomatization and Difunctionalization of Pyridines 2020-08-01 |
|
1 |
|
Copper-Catalyzed Asymmetric Cyanation of Alkenes via Carbonyl-Assisted Coupling of Alkyl-Substituted Carbon-Centered Radicals 2020-07-31 |
|
1 |
|
Ligand-Accelerated Palladium(II)-Catalyzed Enantioselective Amination of C(sp2)–H Bonds 2020-07-31 |
|
1 |
|
Nickel(II)-Catalyzed Borylation of Alkenyl Methyl Ethers via C–O Bond Cleavage 2020-07-31 |
|
1 |
|
Asymmetric Synthesis of 3,3′-Tetrahydrofuryl Spirooxindoles via Palladium-Catalyzed [3+2] Cycloadditions of Methyleneindolinones with Vinylethylene Carbonates 2020-07-29 |
|
1 |
|
Brønsted Acid Catalyzed Cyclization of Aminodiazoesters with Aldehydes to 3-Carboxylate-N-Heterocycles 2020-07-29 |
|
1 |
|
Divergent Domino Reactions of Prop-2-ynylsulfonium Salts: Access to Sulfur-Containing Benzo-Fused Dioxabicyclo[3.3.1]nonanes and Dihydrofuro[2,3-c]chromenes 2020-07-29 |
|
1 |
|
Indoline Catalyzed Acylhydrazone/Oxime Condensation under Neutral Aqueous Conditions 2020-07-29 |
|
0.38 |
|
Synthesis of N–H-Free 1,4-Dihydroisoquinoline-3(2H)-ones via Pd-Catalyzed C–H Olefination Using Polyfluorosulfinyl as the Auxiliary Group 2020-07-29 |
|
1 |
|
Visible-Light-Induced Beckmann Rearrangement by Organic Photoredox Catalysis 2020-07-29 |
|
1 |
|
Construction of a Highly Diastereoselective Aldol Reaction System with l-Threonine Aldolase by Computer-Assisted Rational Molecular Modification and Medium Engineering 2020-07-27 |
|
1 |
|
Rhodium-Catalyzed Carbonylative Synthesis of Aryl Salicylates from Unactivated Phenols 2020-07-27 |
|
0.13 |
|
BI-OAc-Accelerated C3–H Alkylation of Quinoxalin-2(1H)-ones under Visible-Light Irradiation 2020-07-24 |
|
1 |
|
Synthesis of Cyclophane-Braced Peptide Macrocycles via Palladium-Catalyzed Intramolecular C(sp3)–H Arylation of N-Methyl Alanine at C-Termini 2020-07-24 |
|
1 |
|
Phakefustatins A–C: Kynurenine-Bearing Cycloheptapeptides as RXRα Modulators from the Marine Sponge Phakellia fusca 2020-07-23 |
|
1 |
|
Radical-Mediated Distal Ipso-Migration of O/S-Containing Heteroaryls and DFT Studies for Migratory Aptitude 2020-07-23 |
|
1 |
|
Cobalt-Catalyzed Reductive C–O Bond Cleavage of Lignin β-O-4 Ketone Models via In Situ Generation of the Cobalt–Boryl Species 2020-07-22 |
|
1 |
|
Enantioselective Remote C(sp3)–H Cyanation via Dual Photoredox and Copper Catalysis 2020-07-22 |
|
1 |
|
Regio- and Stereoselective Photoredox-Catalyzed Atom Transfer Radical Addition of Thiosulfonates to Aryl Alkynes 2020-07-22 |
|
0.75 |
|
Catalytic Asymmetric Transfer Hydrogenation of trans-Chalcone Derivatives Using BINOL-derived Boro-phosphates 2020-07-21 |
|
0.50 |
|
Direct Synthesis of Mono-α-arylated Ketones from Alcohols and Olefins via Ni-Catalyzed Oxidative Cross-Coupling 2020-07-21 |
|
1 |
|
Simultaneous Implementation of N-Heterocycle-Fused Bridge and Modified Pyrrole Unit on Ni(II) Porphyrin Dimers 2020-07-21 |
|
1 |
|
Copper(0)/PPh3-Mediated Bisheteroannulations of o-Nitroalkynes with Methylketoximes Accessing Pyrazo-Fused Pseudoindoxyls 2020-07-20 |
|
1 |
|
Tetrahydroxydiboron-Promoted Radical Addition of Alkynols 2020-07-19 |
|
1 |
|
Co(III)-Catalyzed Annulative Vinylene Transfer via C–H Activation: Three-Step Total Synthesis of 8-Oxopseudopalmatine and Oxopalmatine 2020-07-17 |
|
1 |
|
Copper-Catalyzed Selective Arylation of Nitriles with Cyclic Diaryl Iodonium Salts: Direct Access to Structurally Diversified Diarylmethane Amides with Potential Neuroprotective and Anticancer Activities 2020-07-17 |
|
1 |
|
Gold-Catalyzed Intermolecular Formal [4 + 2 + 2]-Cycloaddition of Anthranils with Allenamides 2020-07-17 |
|
1 |
|
Synthesis of 2-Formylpyrroles from Pyridinium Iodide Salts 2020-07-17 |
|
1 |
|
[4 + 2]-Annulation of Prop-2-ynylsulfonium Salts and Isatoic Anhydrides: Access to 3-Methylthio-4-quinolones 2020-07-17 |
|
1 |
|
A One-Step Approach to N-(Hetero)aryl-3,5-dinitropyrazoles from (Hetero)aryl Amines 2020-07-16 |
|
1 |
|
Silver(I)-Mediated Cascade Reaction of 2-(1-Alkynyl)-2-alken-1-ones with 2-Naphthols 2020-07-16 |
|
1 |
|
Stereoselective Synthesis of Vinylcyclopropa[b]indolines via a Rh-Migration Strategy 2020-07-16 |
|
0.67 |
|
Ag(I)-Catalyzed Addition of Cyclopropenones and Nitrones to Access Imides 2020-07-14 |
|
1 |
|
Asymmetric Transfer Hydrogenation of N-Unprotected Indoles with Ammonia Borane 2020-07-14 |
|
1 |
|
Copper-Catalyzed Direct C(sp3)–H Alkoxylation to Access Quaternary α-Alkoxylated Amino Acid Derivatives 2020-07-14 |
|
1 |
|
Enantioselective [4 + 2] Cycloaddition Reaction of Vinylquinolines with Dienals Enabled by Synergistic Organocatalysis 2020-07-14 |
|
0.93 |
|
Imine Amidation Catalyzed by a Chiral VAPOL Calcium Phosphate 2020-07-14 |
|
1 |
|
Iodine-Mediated Electrochemical C(sp2)–H Amination: Switchable Synthesis of Indolines and Indoles 2020-07-14 |
|
1 |
|
Palladium-Catalyzed Imidoylation-Triggered [2 + 2 + 1] Cyclization of Internal Alkyne with Isocyanides 2020-07-14 |
|
1 |
|
Perfluoroalkylation of Thiosulfonates: Synthesis of Perfluoroalkyl Sulfides 2020-07-10 |
|
1 |
|
Redox-Neutral P(O)–N Coupling between P(O)–H Compounds and Azides via Dual Copper and Photoredox Catalysis 2020-07-10 |
|
0.95 |
|
Two Reaction Modes of Pyridinium 1,4-Zwitterionic Thiolates with Sulfenes: Synthesis of 3H-1,2-Dithiole 2,2-Dioxides, 1,9a-Dihydropyrido[2,1-c][1,4]thiazines, and Indolizines 2020-07-10 |
|
1 |
|
A Bifunctional Ligand Enables Gold-Catalyzed Hydroarylation of Terminal Alkynes under Soft Reaction Conditions 2020-07-09 |
|
0.72 |
|
CaCl2-Promoted Dehydroxytrifluoromethylselenolation of Alcohols with [Me4N][SeCF3] 2020-07-09 |
|
1 |
|
Construction of Spironaphthalenones via Gold-Catalyzed Intramolecular Dearomatization Reaction of β-Naphthol Derivatives 2020-07-09 |
|
0.75 |
|
On-DNA Cross-Dehydrogenative Coupling Reaction toward the Synthesis of Focused DNA-Encoded Tetrahydroisoquinoline Libraries 2020-07-09 |
|
1 |
|
Selective [3 + 2] Cycloaddition of Cyclopropenone Derivatives and Elemental Chalcogens 2020-07-09 |
|
1 |
|
Silver-Catalyzed C–H Aryloxydifluoromethylation and Arylthiodifluoromethylation of Heteroarenes 2020-07-09 |
|
1 |
|
Substituent Effect Induces Emission Modulation of Stilbene Photoswitches by Spatial Tuning of the N/B Electronic Constraints 2020-07-09 |
|
1 |
|
Twisted Bodipy Derivative as a Heavy-Atom-Free Triplet Photosensitizer Showing Strong Absorption of Yellow Light, Intersystem Crossing, and a High-Energy Long-Lived Triplet State 2020-07-09 |
|
0.67 |
|
Zwitterion-Catalyzed Intermolecular Bromoesterifications 2020-07-08 |
|
1 |
|
Double Enzyme-Catalyzed One-Pot Synthesis of Enantiocomplementary Vicinal Fluoro Alcohols 2020-07-07 |
|
1 |
|
I2-Catalyzed Aerobic α,β-Dehydrogenation and Deamination of Tertiary Alkylamines: Highly Selective Synthesis of Polysubstituted Pyrimidines via Hidden Acyclic Enamines 2020-07-07 |
|
1 |
|
Ruthenium-Catalyzed Brook Rearrangement Involved Domino Sequence Enabled by Acylsilane–Aldehyde Corporation 2020-07-07 |
|
1 |
|
Site-Selective Pyridyl Alkyl Ketone Synthesis from N-Alkenoxypyridiniums through Boekelheide-Type Rearrangements 2020-07-07 |
|
0.67 |
|
Regioselective Hydroboration and Hydrosilylation of N-Heteroarenes Catalyzed by a Zinc Alkyl Complex 2020-07-06 |
|
1 |
|
Rh(III)-Catalyzed C(sp3)–H Acetoxylation of 8-Methylquinolines 2020-07-06 |
|
1 |
|
Rhodium-Catalyzed Sequential Cycloisomerization/Aldol Addition of Cyclopropene Carboxylic Acids with Isatins 2020-07-06 |
|
1 |
|
Visible-Light-Mediated Intermolecular Radical Conjugate Addition for the Construction of Vicinal Quaternary Carbon Centers 2020-07-06 |
|
1 |
|
Oxidant-Induced Azolation of Electron-Rich Phenol Derivatives 2020-07-02 |
|
1 |
|
Sulfoxide Reduction/C(sp3)–S Metathesis Cascade in Ionic Liquid 2020-07-02 |
|
1 |
|
Experimental and Computational Studies on Cp*CyRh(III)/KOPiv-Catalyzed Intramolecular Dehydrogenative Cross-Couplings for Building Eight-Membered Sultam/Lactam Frameworks 2020-07-01 |
|
1 |
|
FeCl3-Mediated Synthesis of 2-(Trifluoromethyl)quinazolin-4(3H)-ones from Isatins and Trifluoroacetimidoyl Chlorides 2020-07-01 |
|
0.88 |
|
Asymmetric Aza-Diels–Alder Reactions of in Situ Generated β,β-Disubstituted α,β-Unsaturated N–H Ketimines Catalyzed by Chiral Phosphoric Acids 2020-06-30 |
|
1 |
|
Asymmetric Synthesis of Axially Chiral Anilides via Organocatalytic Atroposelective N-Acylation 2020-06-30 |
|
1 |
|
Convergent Synthesis of Dihydropyrans from Catalytic Three-Component Reactions of Vinylcyclopropanes, Diazoesters, and Diphenyl Sulfoxide 2020-06-30 |
|
1 |
|
Copper(II)-Mediated Ring Opening/Alkynylation of Tertiary Cyclopropanols by Using Nonmodified Terminal Alkynes 2020-06-30 |
|
1 |
|
Palladium-Catalyzed N-Acylation of Tertiary Amines by Carboxylic Acids: A Method for the Synthesis of Amides 2020-06-30 |
|
1 |
|
Regio- and Enantioselective Palladium-Catalyzed Asymmetric Allylation of N-Fluorenyl Trifluoromethyl Imine 2020-06-30 |
|
1 |
|
Rh(III)-Catalyzed Oxidative C–H Activation/Domino Annulation of Anilines with 1,3-Diynes: A Rapid Access to Blue-Emitting Tricyclic N,O-Heteroaromatics 2020-06-30 |
|
1 |
|
Synthesis of Thiazoles and Isothiazoles via Three-Component Reaction of Enaminoesters, Sulfur, and Bromodifluoroacetamides/Esters 2020-06-30 |
|
1 |
|
Organocatalytic Formal (3 + 2) Cycloaddition toward Chiral Pyrrolo[1,2-a]indoles via Dynamic Kinetic Resolution of Allene Intermediates 2020-06-29 |
|
0.71 |
|
Ring-Strain-Enabled Catalytic Asymmetric Umpolung C–O Bond-Forming Reactions of 1,2-Oxazetidines for the Synthesis of Functionalized Chiral Ethers 2020-06-28 |
|
1 |
|
Copper-Catalyzed Intramolecular C–H Alkoxylation of Diaryltriazoles: Synthesis of Tricyclic Triazole Benzoxazines 2020-06-26 |
|
0.79 |
|
Copper-Catalyzed N,N-Diarylation of Amides for the Construction of 9,10-Dihydroacridine Structure and Applications in the Synthesis of Diverse Nitrogen-Embedded Polyacenes 2020-06-26 |
|
1 |
|
Hexafluoroisopropanol-Promoted Disulfidation and Diselenation of Alkyne, Alkene, and Allene 2020-06-26 |
|
0.17 |
|
Merger of C–F and C–N Bond Cleavage in Cross-Electrophile Coupling for the Synthesis of gem-Difluoroalkenes 2020-06-26 |
|
1 |
|
Palladium(II)-Catalyzed Oxidative Decarboxylative [2 + 2 + 1] Annulation of Cinnamic Acids with Alkynes: Access to Polysubstituted Pentafulvenes 2020-06-26 |
|
1 |
|
Palladium-Catalyzed Asymmetric Decarboxylative [4+2] Dipolar Cycloaddition of 4-Vinyl-1,3-dioxan-2-ones with α,β-Disubstituted Nitroalkenes Enabled by a Benzylic Substituted P,N-Ligand 2020-06-26 |
|
1 |
|
Transition-Metal-Free Site-Selective γ-C(sp2)–H Monoiodination of Arenes Directed by an Aliphatic Keto Group 2020-06-26 |
|
1 |
|
Cobaloxime Catalysis for Enamine Phosphorylation with Hydrogen Evolution 2020-06-25 |
|
1 |
|
Cu(II)-Catalyzed 6π-Photocyclization of Non-6π Substrates 2020-06-25 |
|
1 |
|
Development and Mechanistic Studies of Iron-Catalyzed Construction of Csp2–B Bonds via C–O Bond Activation 2020-06-25 |
|
1 |
|
Divergent Construction of Fully Substituted Pyrroles and Cyclopentadiene Derivatives by Ynamide Annulations: 1,2-Cyclopropyl Migration versus Proton Transfer 2020-06-25 |
|
1 |
|
Nickel-Catalyzed Asymmetric Addition of Aromatic Halides to Ketones: Highly Enantioselective Synthesis of Chiral 2,3-Dihydrobenzofurans Containing a Tertiary Alcohol 2020-06-23 |
|
1 |
|
Regio- and Diastereoselective Spirocyclopropanation of Benzofuran-Derived Azadienes through 1,4-Addition-Induced Dearomatization Reaction under Mild Conditions 2020-06-23 |
|
1 |
|
Ytterbium-Catalyzed Intramolecular [3 + 2] Cycloaddition based on Furan Dearomatization to Construct Fused Triazoles 2020-06-23 |
|
1 |
|
Catalytic Asymmetric Synthesis of Vicinal Tetrasubstituted Diamines via Umpolung Cross-Mannich Reaction of Cyclic Ketimines 2020-06-22 |
|
1 |
|
Characterization of SepE and SepF for the N6-Glycosylated Adenine Structure Formation in Septacidin Biosynthesis 2020-06-21 |
|
1 |
|
Allylboronates from Vinyl Triflates and α-Chloroboronates by Reductive Nickel Catalysis 2020-06-19 |
|
1 |
|
Direct Intramolecular Aminoboration of Allenes 2020-06-19 |
|
1 |
|
Palladium-Catalyzed Fluoroarylation of gem-Difluoroenynes to Access Trisubstituted Trifluoromethyl Allenes 2020-06-19 |
|
1 |
|
Photoinduced, Copper-Catalyzed Three-Component Annulation of gem-Dialkylthio Enynes 2020-06-19 |
|
1 |
|
Ruthenium(II)-Catalyzed Ortho-C–H Alkylation of Naphthylamines with Diazo Compounds for Synthesis of 2,2-Disubstituted π-Extended 3-Oxindoles in Water 2020-06-19 |
|
0.94 |
|
An Indirect Strategy for Trifluoromethylation via an Iridium Catalyst: Approach to Generate Isocoumarin Skeletons in Bioactive Molecules 2020-06-18 |
|
1 |
|
Cobalt-Catalyzed Cycloamination: Synthesis and Photophysical Properties of Polycyclic N-Heterocycles 2020-06-18 |
|
1 |
|
Synthesis of Cyclopropanes via 1,3-Migration of Acyloxy Groups Triggered by Formation of α-Imino Rhodium Carbenes 2020-06-18 |
|
1 |
|
Tandem Oxidative Ring Expansion for Synthesis of Dibenzocyclooctaphenanthrenes 2020-06-18 |
|
0.10 |
|
1,4-Fluoroamination of 1,3-Enynes en Route to Fluorinated Allenes 2020-06-17 |
|
1 |
|
Atroposelective Synthesis of Axially Chiral 3-Arylindoles by Copper-Catalyzed Asymmetric Cross-Coupling of Indoles with Quinones and Naphthoquinones 2020-06-17 |
|
1 |
|
Catalytic Asymmetric Acyloin Rearrangements of α-Ketols, α-Hydroxy Aldehydes, and α-Iminols by N,N′-Dioxide–Metal Complexes 2020-06-17 |
|
1 |
|
Direct Synthesis of Propen-2-yl Sulfones through Cascade Reactions Using Calcium Carbide as an Alkyne Source 2020-06-17 |
|
1 |
|
General Synthesis of Chiral α,α-Diaryl Carboxamides by Enantioselective Palladium-Catalyzed Cross-Coupling 2020-06-17 |
|
1 |
|
One-Pot Synthesis of Furo[3,4-c]indolo[2,1-a]isoquinolines through Rh(III)-Catalyzed Cascade Reactions of 2-Phenylindoles with 4-Hydroxy-2-alkynoates 2020-06-17 |
|
0.97 |
|
Palladium-Catalyzed Stereoselective Hydrodefluorination of Tetrasubstituted gem-Difluoroalkenes 2020-06-17 |
|
1 |
|
Rhodium-Catalyzed Ring-Opening Hydroacylation of Alkylidenecyclopropanes with Chelating Aldehydes for the Synthesis of γ,δ-Unsaturated Ketones 2020-06-17 |
|
1 |
|
Silver-Catalyzed Trifluoromethoxylation of Alkyl Trifluoroborates 2020-06-17 |
|
1 |
|
Synthesis of 3,4-Fused Tricyclic Indoles through Cascade Carbopalladation and C–H Amination: Development and Total Synthesis of Rucaparib 2020-06-17 |
|
1 |
|
Tuning Vinylethylene Carbonates into [4 + 2] Cycloaddition via Silylation and Vinylogous Peterson Elimination 2020-06-17 |
|
1 |
|
Unnatural α-Amino Acid Synthesized through α-Alkylation of Glycine Derivatives by Diacyl Peroxides 2020-06-17 |
|
1 |
|
Visible-Light-Mediated Decarboxylative Tandem Carbocyclization of Acrylamide-Attached Alkylidenecyclopropanes: Access to Polycyclic Benzazepine Derivatives 2020-06-17 |
|
1 |
|
Asymmetric Total Syntheses of (+)-Penostatins A and C 2020-06-16 |
|
1 |
|
Copper-Catalyzed Oxalamide-Directed ortho-C–H Amination of Anilines with Alkylamines 2020-06-16 |
|
1 |
|
Acid-Promoted [3 + 1 + 1] Cyclization of N-Tosylhydrazones and Isocyanides: A Method for the Preparation of 4,5-Diaminopyrazoles 2020-06-15 |
|
1 |
|
Palladium-Catalyzed Intermolecular Heck-Type Dearomative [4 + 2] Annulation of 2H-Isoindole Derivatives with Internal Alkynes 2020-06-15 |
|
1 |
|
1,2-Hydroboration of Pyridines by Organomagnesium 2020-06-11 |
|
1 |
|
Catalytic Asymmetric Addition Reactions of Formaldehyde N,N-Dialkylhydrazone to Synthesize Chiral Nitrile Derivatives 2020-06-11 |
|
1 |
|
Isolation, Total Synthesis, and Absolute Configuration Determination of Renoprotective Dimeric N-Acetyldopamine–Adenine Hybrids from the Insect Aspongopus chinensis 2020-06-11 |
|
0.75 |
|
Ni-Catalyzed Denitrogenative Cross-Coupling of Benzotriazinones and Cyclopropanols: An Easy Access to Functionalized β-Aryl Ketones 2020-06-11 |
|
1 |
|
Highly Chemo- and Enantioselective Hydrogenation of 2-Substituted-4-oxo-2-alkenoic Acids 2020-06-10 |
|
1 |
|
Palladium-Catalyzed Site-Selective Benzocylization of Aromatic Acids with o-Fluoro-Substituted Diaryliodonium Salts toward 3,4-Benzocoumarins 2020-06-10 |
|
1 |
|
Visible-Light-Promoted Cross-Coupling Reactions of 4-Alkyl-1,4-dihydropyridines with Thiosulfonate or Selenium Sulfonate: A Unified Approach to Sulfides, Selenides, and Sulfoxides 2020-06-10 |
|
1 |
|
Palladium-Catalyzed Regioselective Coupling Cyclohexenone into Indoles: Atom-Economic Synthesis of β-Indolyl Cyclohexenones and Derivatization Applications 2020-06-09 |
|
1 |
|
gem-Dinitromethyl-Functionalized 5-Amino-1,3,4-oxadiazolate Derivatives: Alternate Route, Characterization, and Property Analysis 2020-06-09 |
|
0.30 |
|
Characterization of Tailoring Methyltransferases Involved in K-41A Biosynthesis: Modulating Methylation to Improve K-41A Anti-infective Activity 2020-06-08 |
|
0.89 |
|
Cu-Catalyzed C–H Alkenylation of Benzoic Acid and Acrylic Acid Derivatives with Vinyl Boronates 2020-06-08 |
|
0.80 |
|
Stereodivergent Synthesis of α-Quaternary Serine and Cysteine Derivatives Containing Two Contiguous Stereogenic Centers via Synergistic Cu/Ir Catalysis 2020-06-06 |
|
1 |
|
Free-Radical-Promoted Dehydrogenative Coupling of Polyfluorinated Alcohol with Quinone, Chromone, and Coumarin 2020-06-05 |
|
1 |
|
Cu(I)-Catalyzed Asymmetric α-Allenylation of Activated Ketimines with 3-Butynoates 2020-06-04 |
|
1 |
|
Fe-Catalyzed Sequential C(sp3)–H/N–H Annulation of 2-Methylindoles with Ethyl Trifluoropyruvate at Room Temperature: Construction of Pyrrolo[1,2-α]indoles 2020-06-04 |
|
1 |
|
Rapid Synthesis of Alkenylated BINOL Derivatives via Rh(III)-Catalyzed C–H Bond Activation 2020-06-04 |
|
1 |
|
Reciprocal-Activation Strategy for Allylic Sulfination with Unactivated Allylic Alcohols 2020-06-04 |
|
0.97 |
|
Selective Recognition of Chloride Anion in Water 2020-06-04 |
|
1 |
|
Remarkable Ligand Effect on Rh-Catalyzed C–H-Active [3 + 2] Annulation of Ketimines and Alkynes 2020-06-03 |
|
1 |
|
Ruthenium-Catalyzed Hydrogen Evolution o-Aminoalkylation of Phenols with Cyclic Amines 2020-06-03 |
|
1 |
|
Stereoselective Construction of the Highly Congested Tricyclic Core Structure in Leucosceptroid H 2020-06-03 |
|
1 |
|
Convergent Synthesis of Calcium-Dependent Antibiotic CDA3a and Analogues with Improved Antibacterial Activity via Late-Stage Serine Ligation 2020-06-02 |
|
1 |
|
Curved Carbon Skeleton in Oriented External Electric Fields: Modulated Curvature, Directional Bowl Inversion, and Face-Selective Cycloadditions of Corannulene 2020-06-02 |
|
1 |
|
Discovery, Biosynthesis, and Heterologous Production of Loonamycin, a Potent Anticancer Indolocarbazole Alkaloid 2020-06-02 |
|
1 |
|
Enantioselective Construction of Spiro Quaternary Carbon Stereocenters via Pd-Catalyzed Intramolecular α-Arylation 2020-06-02 |
|
1 |
|
O-Phosphination of Aldehydes/Ketones toward Phosphoric Esters: Experimental and Mechanistic Studies 2020-06-02 |
|
1 |
|
Pd-Catalyzed Asymmetric Allylic Substitution Cascade of But-2-ene-1,4-diyl Dimethyl Dicarbonate for the Synthesis of Chiral 2,3-Dihydrofurans 2020-06-02 |
|
1 |
|
Geometrically Selective Denitrative Trifluoromethylthiolation of β-Nitrostyrenes with AgSCF3 for (E)-Vinyl Trifluoromethyl Thioethers 2020-06-01 |
|
1 |
|
Activation and Characterization of Bohemamine Biosynthetic Gene Cluster from Streptomyces sp. CB02009 2020-05-28 |
|
1 |
|
Azetidine-Containing Heterospirocycles Enhance the Performance of Fluorophores 2020-05-28 |
|
1 |
|
Cobalt/Bisoxazolinephosphine-Catalyzed Asymmetric Alkynylation of Isatins 2020-05-28 |
|
1 |
|
Diazo Activation with Diazonium Salts: Synthesis of Indazole and 1,2,4-Triazole 2020-05-28 |
|
0.14 |
|
Peptide-Catalyzed Highly Asymmetric Cross-Aldol Reaction of Aldehydes to Biomimetically Synthesize 1,4-Dicarbonyls 2020-05-28 |
|
1 |
|
Radical Pentafluoroethylation of Unactivated Alkenes Using CuCF2CF3 2020-05-28 |
|
1 |
|
Selective Synthesis of Pyrazolo[1,2-a]pyrazolones and 2-Acylindoles via Rh(III)-Catalyzed Tunable Redox-Neutral Coupling of 1-Phenylpyrazolidinones with Alkynyl Cyclobutanols 2020-05-28 |
|
1 |
|
Biosynthesis and Chemical Diversification of Verucopeptin Leads to Structural and Functional Versatility 2020-05-27 |
|
1 |
|
Cobalt-Catalyzed Switchable Intramolecular Thioenolization/C–H Thiolation and C(sp2)–H/C(sp3)–H Dehydrogenative Coupling 2020-05-27 |
|
1 |
|
Palladium-Catalyzed C-2 and C-3 Dual C–H Functionalization of Indoles: Synthesis of Fluorinated Isocryptolepine Analogues 2020-05-27 |
|
1 |
|
Regioselective and Diastereoselective Dearomative Multifunctionalization of In-Situ-Activated Azaarenes: An Access to Bridged Azaheterocycles 2020-05-27 |
|
1 |
|
Remote and Selective C(sp2)–H Olefination for Sequential Regioselective Linkage of Phenanthrenes 2020-05-27 |
|
0.90 |
|
A Versatile Synthesis of Vinyl-Substituted Heterocycles via Regio- and Enantioselective Pd-Catalyzed Tandem Allylic Substitution 2020-05-26 |
|
1 |
|
Catalytic Asymmetric [3 + 2] Annulation via Indolyl Copper–Allenylidene Intermediates: Diastereo- and Enantioselective Assembly of Pyrrolo[1,2-a]indoles 2020-05-26 |
|
1 |
|
Crotonpenoids A and B, Two Highly Modified Clerodane Diterpenoids with a Tricyclo[7.2.1.02,7]dodecane Core from Croton yanhuii: Isolation, Structural Elucidation, and Biomimetic Semisynthesis 2020-05-26 |
|
1 |
|
One-Pot Preparation of 9,10-Dihydrophenanthrenes Initiated by Rhodium(III)-Catalyzed C–H Activation and Relay Diels–Alder Reaction 2020-05-26 |
|
1 |
|
Organocatalytic Approach for Assembling Flavanones via a Cascade 1,4-Conjugate Addition/oxa-Michael Addition between Propargylamines with Water 2020-05-22 |
|
1 |
|
Asymmetric Total Syntheses of (−)-Fennebricin A, (−)-Renieramycin J, (−)-Renieramycin G, (−)-Renieramycin M, and (−)- Jorunnamycin A via C–H Activation 2020-05-21 |
|
1 |
|
Thermo/Anion Dual-Responsive Supramolecular Organoplatinum–Crown Ether Complex 2020-05-21 |
|
0.83 |
|
tBuOK-Promoted Cyclization of Imines with Aryl Halides 2020-05-21 |
|
1 |
|
Cobalt-Bisoxazoline-Catalyzed Enantioselective Cross-Coupling of α-Bromo Esters with Alkenyl Grignard Reagents 2020-05-20 |
|
1 |
|
Cobalt-Catalyzed Asymmetric Cross-Coupling Reaction of Fluorinated Secondary Benzyl Bromides with Lithium Aryl Boronates/ZnBr2 2020-05-20 |
|
1 |
|
Palladium-Catalyzed Asymmetric (2+3) Annulation of p-Quinone Methides with Trimethylenemethanes: Enantioselective Synthesis of Functionalized Chiral Spirocyclopentyl p-Dienones 2020-05-20 |
|
1 |
|
Visible-Light-Induced Dehydrohalogenative Coupling for Intramolecular α-Alkenylation: A Way to Build Seven- and Eight-Membered Rings 2020-05-20 |
|
0.31 |
|
Waikikiamides A–C: Complex Diketopiperazine Dimer and Diketopiperazine–Polyketide Hybrids from a Hawaiian Marine Fungal Strain Aspergillus sp. FM242 2020-05-20 |
|
0.06 |
|
[2 + 2 + 1] Heteroannulation of Alkenes with Enynyl Benziodoxolones and Silver Nitrite Involving C≡C bond Oxidative Cleavage: Entry to 3-Aryl-Δ2-isoxazolines 2020-05-20 |
|
1 |
|
AIBN-Induced Remote Trifluoromethyl-Alkynylation of Thioalkynes 2020-05-19 |
|
1 |
|
Nickel-Catalyzed Homo- and Cross-Coupling of Allyl Alcohols via Allyl Boronates 2020-05-19 |
|
1 |
|
The C–H Activation/Bidirecting Group Strategy for Selective Direct Synthesis of Diverse 1,1′-Biisoquinolines 2020-05-19 |
|
1 |
|
pH-Controlled Chirality Inversion in Enantiodifferentiating Photocyclodimerization of 2-Antharacenecarboxylic Acid Mediated by γ-Cyclodextrin Derivatives 2020-05-17 |
|
1 |
|
Asymmetric (4 + 3) and (4 + 1) Annulations of Isatin-derived Morita–Baylis–Hillman Carbonates to Construct Diverse Chiral Heterocyclic Frameworks 2020-05-15 |
|
1 |
|
A Simple Protocol for the Stereoselective Construction of Enaminyl Sulfonyl Fluorides 2020-05-14 |
|
1 |
|
Blue Light Promoted Difluoroalkylation of Aryl Ketones: Synthesis of Quaternary Alkyl Difluorides and Tetrasubstituted Monofluoroalkenes 2020-05-14 |
|
1 |
|
Copper-Catalyzed Chemodivergent Cyclization of N-(ortho-alkynyl)aryl-Pyrrole and Indoles 2020-05-14 |
|
1 |
|
Ruthenium-Catalyzed Highly Enantioselective Synthesis of cis-3-Quinuclidinols via DKR Asymmetric Transfer Hydrogenation 2020-05-14 |
|
1 |
|
Selective Inclusion of Fluoride within the Cavity of a Two-Wall Bis-calix[4]pyrrole 2020-05-14 |
|
0.64 |
|
Base-Promoted Radical Azofluoromethylation of Unactivated Alkenes 2020-05-13 |
|
0.20 |
|
Directed Cobalt-Catalyzed anti-Markovnikov Hydroalkylation of Unactivated Alkenes Enabled by “Co–H” Catalysis 2020-05-13 |
|
1 |
|
Electrochemical Annulation–Iodosulfonylation of 1,5-Enyne-containing para-Quinone Methides (p-QMs) to Access (E)-Spiroindenes 2020-05-13 |
|
1 |
|
Rhodium(III)-Catalyzed [4+3] Annulation of N-Aryl-pyrazolidinones and Propargylic Acetates: Access to Benzo[c][1,2]diazepines 2020-05-13 |
|
0.96 |
|
Structural Diversification of Andiconin-Derived Natural Products by α-Ketoglutarate-Dependent Dioxygenases 2020-05-13 |
|
0.33 |
|
Asymmetric Linear-Selective Hydroformylation of 1,1-Dialkyl Olefins Assisted by a Steric-Auxiliary Strategy 2020-05-12 |
|
1 |
|
Quantum Mechanical–NMR-Aided Configuration and Conformation of Two Unreported Macrocycles Isolated from the Soft Coral Lobophytum sp.: Energy Calculations versus Coupling Constants 2020-05-12 |
|
0.60 |
|
When Anthracene and Quinone Avoid Cycloaddition: Acid-Catalyzed Redox Neutral Functionalization of Anthracene to Aryl Ethers 2020-05-12 |
|
1 |
|
N-Iodosuccinimide-Mediated Dimerization of 2-Alkynylnaphthols: A Highly Diastereoselective Construction of Bridged Polycyclic Compounds via Vinylidene ortho-Quinone Methide Intermediate 2020-05-11 |
|
1 |
|
Synthesis of 2-Imino-1,3,4-thiadiazoles from Hydrazides and Isothiocyanates via Sequential Oxidation and P(NMe2)3-Mediated Annulation Reactions 2020-05-10 |
|
1 |
|
A General One-Pot Protocol for Hindered N-Alkyl Azaheterocycles from Tertiary Carboxylic Acids 2020-05-08 |
|
0.57 |
|
Copper-Mediated DNA-Compatible One-Pot Click Reactions of Alkynes with Aryl Borates and TMS-N3 2020-05-08 |
|
1 |
|
Nickel-Catalyzed Formal Aminocarbonylation of Secondary Benzyl Chlorides with Isocyanides 2020-05-08 |
|
1 |
|
Palladium-Catalyzed Regio- and Stereoselective Cross-Coupling of Vinylethylene Carbonates with Ketimine Esters to Generate (Z)-Tri- and Tetra-substituted Allylic Amino Acid Derivatives 2020-05-08 |
|
1 |
|
Rh(I)-Catalyzed C6-Selective Decarbonylative Alkylation of 2-Pyridones with Alkyl Carboxylic Acids and Anhydrides 2020-05-08 |
|
0.83 |
|
Synthesis of Spiroisoxazolines via an Oximation/Dearomatization Cascade under Air 2020-05-08 |
|
1 |
|
Iron-Catalyzed Oxidative Coupling of Indoline-2-ones with Aminobenzamides via Dual C–H Functionalization 2020-05-07 |
|
1 |
|
Nickel(II)-Catalyzed Addition of Aryl-, Alkenyl-, and Alkylboronic Acids to Alkenylazaarenes 2020-05-07 |
|
1 |
|
Sequential Visible-Light and N-Heterocyclic Carbene Catalysis: Stereoselective Synthesis of Tetrahydropyrano[2,3-b]indoles 2020-05-07 |
|
1 |
|
Enantioselective Copper-Catalyzed Remote C(sp3)–H Alkynylation of Linear Primary Sulfonamides 2020-05-05 |
|
1 |
|
DNA Compatible Intermolecular Wittig Olefination for the Construction of α, β-Unsaturated Carbonyl Compounds 2020-05-04 |
|
1 |
|
Organocatalytic Regiodivergent Ring Expansion of Cyclobutanones for the Enantioselective Synthesis of Azepino[1,2-a]indoles and Cyclohepta[b]indoles 2020-05-04 |
|
1 |
|
Palladium-Catalyzed Cascade Decarboxylative Amination/6-endo-dig Benzannulation of o-Alkynylarylketones with N-Hydroxyamides To Access Diverse 1-Naphthylamine Derivatives 2020-05-04 |
|
1 |
|
K2S as Sulfur Source and DMSO as Carbon Source for the Synthesis of 2-Unsubstituted Benzothiazoles 2020-05-03 |
|
1 |
|
Acylation of Aryl Halides and α-Bromo Acetates with Aldehydes Enabled by Nickel/TBADT Cocatalysis 2020-05-01 |
|
1 |
|
Carbocation versus Carbene Controlled Chemoselectivity: DFT Study on Gold- and Silver-Catalyzed Alkylation/Cyclopropanation of Indoles with Vinyl Diazoesters 2020-05-01 |
|
0.80 |
|
Chiral Binaphthyl Box-Copper-Catalyzed Enantioselective Tandem Michael–Ketalization Annulations for Optically Active Aryl and Heteroaryl Fused Bicyclicnonanes 2020-05-01 |
|
1 |
|
Pd-Catalyzed Regiodivergent Synthesis of Diverse Oxindoles Enabled by the Versatile Heck Reaction of Carbamoyl Chlorides 2020-05-01 |
|
1 |
|
Visible-Light-Induced Palladium-Catalyzed Intermolecular Narasaka–Heck Reaction at Room Temperature 2020-05-01 |
|
1 |
|
Catalytic C–C Cleavage/Alkyne–Carbonyl Metathesis Sequence of Cyclobutanones 2020-04-30 |
|
1 |
|
Pd-Catalyzed Cross-Coupling of Highly Sterically Congested Enol Carbamates with Grignard Reagents via C–O Bond Activation 2020-04-30 |
|
1 |
|
Electrochemical Oxidative Phosphorylation of Aldehyde Hydrazones 2020-04-28 |
|
1 |
|
Thiol Activation toward Selective Thiolation of Aromatic C–H Bond 2020-04-28 |
|
1 |
|
A Dual-Protein Cascade Reaction for the Regioselective Synthesis of Quinoxalines 2020-04-27 |
|
1 |
|
Synthesis of ortho-Phenolic Sulfilimines via an Intermolecular Sulfur Atom Transfer Cascade Reaction 2020-04-27 |
|
1 |
|
Postulated Biogenesis-Guided Total Synthesis and Structural Revision of 2,18-seco-Lankacidinol A 2020-04-24 |
|
1 |
|
Total Synthesis of Fawcettimine-Type Alkaloid, Lycojaponicumin A 2020-04-24 |
|
1 |
|
Visible-Light-Induced Regioselective Dicarbonylation of Indolizines with Oxoaldehydes via Direct C–H Functionalization 2020-04-23 |
|
1 |
|
Absolute Configurations and Stereochemical Inversion Mechanism of Epimeric Securinega Alkaloids from Flueggea suffruticosa 2020-04-22 |
|
1 |
|
Structure-Guided Directed Evolution of a Carbonyl Reductase Enables the Stereoselective Synthesis of (2S,3S)-2,2-Disubstituted-3-hydroxycyclopentanones via Desymmetric Reduction 2020-04-22 |
|
1 |
|
Copper-Catalyzed Radical N-Demethylation of Amides Using N-Fluorobenzenesulfonimide as an Oxidant 2020-04-21 |
|
0.83 |
|
Redox Neutral Radical-Relay Cobalt Catalysis toward C–H Fluorination and Amination 2020-04-20 |
|
1 |
|
Cobalt-Catalyzed Regio- and Enantioselective Allylic Alkylation of Malononitriles 2020-04-17 |
|
1 |
|
Directing-Group-Controlled Ring-Opening Addition and Hydroarylation of Oxa/azabenzonorbornadienes with Arenes via C–H Activation 2020-04-17 |
|
1 |
|
Terpenoids from Resina Commiphora Regulating Lipid Metabolism via Activating PPARα and CPT1 Expression 2020-04-17 |
|
1 |
|
Transamidation for the Synthesis of Primary Amides at Room Temperature 2020-04-16 |
|
0.50 |
|
Directing-Group-Based Strategy Enabling Intermolecular Heck-Type Reaction of Cycloketone Oxime Esters and Unactivated Alkenes 2020-04-15 |
|
1 |
|
Eleucanainones A and B: Two Dimeric Structures from the Bulbs of Eleutherine americana with Anti-MRSA Activity 2020-04-15 |
|
1 |
|
Access to Optically Enriched α-Aryloxycarboxylic Esters via Carbene-Catalyzed Dynamic Kinetic Resolution and Transesterification 2020-04-14 |
|
0.48 |
|
Bimetallic Catalytic Tandem Reaction of Acyclic Enynones: Enantioselective Access to Tetrahydrobenzofuran Derivatives 2020-04-14 |
|
1 |
|
Spiroinonotsuoxotriols A and B, Two Highly Rearranged Triterpenoids from Inonotus obliquus 2020-04-14 |
|
1 |
|
Switchable Copper-Catalyzed Approach to Benzodithiole, Benzothiaselenole, and Dibenzodithiocine Skeletons 2020-04-14 |
|
0.58 |
|
A Family of BODIPY-like Highly Fluorescent and Unsymmetrical Bis(BF2) Pyrrolyl–Acylhydrazone Chromophores: BOAPY 2020-04-13 |
|
1 |
|
Copper-Catalyzed Annulation of Oxime Acetates with α-Amino Acid Ester Derivatives: Synthesis of 3-Sulfonamido/Imino 4-Pyrrolin-2-ones 2020-04-13 |
|
1 |
|
Organocatalytic Aza-Michael/Michael Cyclization Cascade Reaction: Enantioselective Synthesis of Spiro-oxindole Piperidin-2-one Derivatives 2020-04-13 |
|
1 |
|
Photo-on-Demand Synthesis of Chloroformates with a Chloroform Solution Containing an Alcohol and Its One-Pot Conversion to Carbonates and Carbamates 2020-04-13 |
|
0.25 |
|
Stereocomplementary Synthesis of Pharmaceutically Relevant Chiral 2-Aryl-Substituted Pyrrolidines Using Imine Reductases 2020-04-13 |
|
1 |
|
Decarboxylative Thiolation of Redox-Active Esters to Thioesters by Merging Photoredox and Copper Catalysis 2020-04-12 |
|
1 |
|
Cobalt-Catalyzed Regioselective Carboamidation of Alkynes with Imides Enabled by Cleavage of C–N and C–C Bonds 2020-04-10 |
|
1 |
|
Cyanide Boosting Copper Catalysis: A Mild Approach to Fluorescent Benzazole Derivatives from Nonemissive Schiff Bases in Biological Media 2020-04-10 |
|
1 |
|
Liquid-Phase Total Synthesis of Plecanatide Aided by Diphenylphosphinyloxyl Diphenyl Ketone (DDK) Derivatives 2020-04-10 |
|
1 |
|
Photocatalytic Remote Oxyfluoroalkylation of Heteroalkynes: Regio-, Stereo-, and Site-Selective Access to Complex Fluoroalkylated (Z)-Alkenes 2020-04-10 |
|
1 |
|
Rhodium(III)-Catalyzed Asymmetric Addition of Inert Arene C–H Bond to Aldehydes To Afford Enantioenriched Phthalides 2020-04-10 |
|
1 |
|
Rhodium(III)-Catalyzed Kinetic Resolution of Racemic 1,6-Dienes via Asymmetric Borylative Cyclization 2020-04-10 |
|
1 |
|
Titanocene-Catalyzed Reductive Domino Epoxide Ring Opening/Defluorinative Cross-Coupling Reaction 2020-04-10 |
|
1 |
|
Deacetylative Aryl Migration of Diaryliodonium Salts with C(sp2)–N Bond Formation toward ortho-Iodo N-Aryl Sulfonamides 2020-04-09 |
|
1 |
|
Copper-Catalyzed Functionalization of Aza-Aromatic Rings with Fluoroalcohols via Direct C(sp2)–H/C(sp3)–H Coupling Reactions 2020-04-08 |
|
1 |
|
Pd-Catalyzed Oxidative Annulation of Aryl Ethers with Alkynes: Synthesis of Functionalized Spirocycles and Naphthalenes 2020-04-08 |
|
1 |
|
Computation-Guided Development of the “Click” ortho-Quinone Methide Cycloaddition with Improved Kinetics 2020-04-07 |
|
1 |
|
Diastereoselective Construction of Cyclopropane-Fused Tetrahydroquinolines via a Sequential [4 + 2]/[2 + 1] Annulation Reaction 2020-04-07 |
|
1 |
|
Electrochemical Oxidative Dehydrogenative Phosphorylation of N-Heterocycles with P(O)–H Compounds in Imidazolium-Based Ionic Liquid 2020-04-07 |
|
1 |
|
Electroreductive 4-Pyridylation of Electron-deficient Alkenes with Assistance of Ni(acac)2 2020-04-07 |
|
0.71 |
|
Time-Economical Radical Cascade Cyclization/Haloazidation of 1,6-Enynes: Construction of Highly Functional Succinimide Derivatives 2020-04-07 |
|
1 |
|
A Hg(OTf)2-Catalyzed Enolate Umpolung Reaction Enables the Synthesis of Coumaran-3-ones and Indolin-3-ones 2020-04-06 |
|
1 |
|
Multistep Photoisomerization of Dimesitylboron-Functionalized Stilbene Analogues 2020-04-06 |
|
0.13 |
|
Three-Component Borylallenylation of Alkynes: Access to Densely Boryl-Substituted Ene-allenes 2020-04-06 |
|
1 |
|
Cascade Claisen and Meinwald Rearrangement for One-Pot Divergent Synthesis of Benzofurans and 2H-Chromenes 2020-04-03 |
|
1 |
|
Construction of Thiazole-Fused Dihydropyrans via Formal [4 + 2] Cycloaddition Reaction on DNA 2020-04-03 |
|
1 |
|
Gold-Catalyzed Oxidative Cascade Cyclization of 1,3-Diynamides: Polycyclic N-Heterocycle Synthesis via Construction of a Furopyridinyl Core 2020-04-03 |
|
1 |
|
Ni-Catalyzed Allylic Dearomatization Reaction of β-Naphthols with Allylic Alcohols 2020-04-03 |
|
1 |
|
Nickel-Catalyzed Formal Aminocarbonylation of Unactivated Alkyl Iodides with Isocyanides 2020-04-03 |
|
1 |
|
Alternarin A, a Drimane Meroterpenoid, Suppresses Neuronal Excitability from the Coral-Associated Fungi Alternaria sp. ZH-15 2020-04-02 |
|
0.78 |
|
Photocatalytic [2 + 2] Cycloaddition in DNA-Encoded Chemistry 2020-04-02 |
|
0.50 |
|
Rhodium(III)-Catalyzed Asymmetric C–H Activation of N-Methoxybenzamide with Quinone and Its Application in the Asymmetric Synthesis of a Dihydrolycoricidine Analogue 2020-04-02 |
|
1 |
|
Brønsted Acid Catalyzed Enantioselective Assembly of Spirochroman-3,3-oxindoles 2020-04-01 |
|
1 |
|
Copper(I)-Catalyzed Ketenimine Formation/Aza-Claisen Rearrangement Cascade for Stereoselective Synthesis of α-Allylic Amidines 2020-04-01 |
|
1 |
|
Iron-Catalyzed Borylation of Aryl Ethers via Cleavage of C–O Bonds 2020-04-01 |
|
1 |
|
Ruthenium-Catalyzed Diastereoselective Synthesis of Fully Substituted Pyrrolidines from Anilines and Diazo Pyruvates 2020-04-01 |
|
1 |
|
Copper-Catalyzed Trifluoromethylation of Ynones Coupled with Dearomatizing Spirocyclization of Indoles: Access to CF3-Containing Spiro[cyclopentane-1,3′-indole] 2020-03-31 |
|
1 |
|
Copper-free Sandmeyer-type Reaction for the Synthesis of Sulfonyl Fluorides 2020-03-31 |
|
1 |
|
CuBr-Catalyzed α-Arylation and Aerobic Oxidative Dehydrogenative C–N Coupling for the Synthesis of Spiro[cyclohexane-1,12′-isoindolo[1,2-b]quinazolin]-10′-one Derivatives 2020-03-31 |
|
1 |
|
Iron-Catalyzed Alkylazidation of 1,1-Disubstituted Alkenes with Diacylperoxides and TMSN3 2020-03-31 |
|
1 |
|
Synthesis of Tetramic Acid Derivatives via a Tandem Umpolung Alkylation/Reduction/Cyclization Reaction of γ-Hydrazono β-Ketoester 2020-03-31 |
|
0.13 |
|
Understanding the Chemoselectivity in Palladium-Catalyzed Three-Component Reaction of o-Bromobenzaldehyde, N-Tosylhydrazone, and Methanol 2020-03-31 |
|
1 |
|
Visible-Light-Induced, Base-Promoted Transition-Metal-Free Dehalogenation of Aryl Fluorides, Chlorides, Bromides, and Iodides 2020-03-31 |
|
1 |
|
Gold(I)-Catalyzed [8+4] Cycloaddition of 1,4-All-Carbon Dipoles with Tropone 2020-03-30 |
|
1 |
|
Hydrogen-Bond-Mediated Aglycone Delivery: Synthesis of β-d-Fructofuranosides 2020-03-30 |
|
1 |
|
3,3′-Disubstituted Oxindoles Formation via Copper-Catalyzed Arylboration and Arylsilylation of Alkenes 2020-03-27 |
|
1 |
|
Development of a C2-Symmetric Chiral aza Spirocyclic Diol 2020-03-27 |
|
1 |
|
Highly Regio- and Enantioselective Hydrogenation of Conjugated α-Substituted Dienoic Acids 2020-03-27 |
|
1 |
|
Palladium-Catalyzed Tandem Dehydrogenative [4 + 2] Annulation of Terminal Olefins with N-Sulfonyl Amides via C–H Activations 2020-03-27 |
|
1 |
|
Stereoselective Phenylselenoglycosylation of Glycals Bearing a Fused Carbonate Moiety toward the Synthesis of 2-Deoxy-β-galactosides and β-Mannosides 2020-03-27 |
|
1 |
|
Gold and Brønsted Acid Catalyzed Spirocyclization of 2- and 3-Indolyl-Tethered 1,4-Enyne Acetates to Spiro[4,n]alkyl[b]indoles 2020-03-26 |
|
0.20 |
|
Asymmetric Catalytic Diverse Ring Opening/Cycloadditions of Cyclobutenones with (E)-Alkenyloxindoles and (E)-Dioxopyrrolidines 2020-03-25 |
|
1 |
|
Rh-Catalyzed C–H Amination/Annulation of Acrylic Acids and Anthranils by Using −COOH as a Deciduous Directing Group: An Access to Diverse Quinolines 2020-03-25 |
|
1 |
|
Copper-Catalyzed Remote C(sp3)–H Amination of Carboxamides 2020-03-24 |
|
1 |
|
Selective Oxidative Cleavage of 3-Methylindoles with Primary Amines Affording Quinazolinones 2020-03-24 |
|
1 |
|
Brønsted Base and Lewis Acid Cooperatively Catalyzed Asymmetric exo′-Selective [3 + 2] Cycloaddition of Trifluoromethylated Azomethine Ylides and Methyleneindolinones 2020-03-23 |
|
1 |
|
Highly Enantioselective Cobalt-Catalyzed Hydroboration of Diaryl Ketones 2020-03-23 |
|
1 |
|
Iridium-Catalyzed γ-Selective Hydroboration of γ-Substituted Allylic Amides 2020-03-23 |
|
1 |
|
Nickel-Catalyzed Asymmetric Reductive Arylbenzylation of Unactivated Alkenes 2020-03-23 |
|
1 |
|
Stereoselective Synthesis of (−)-Verazine and Congeners via a Cascade Ring-Switching Process of Furostan-26-acid 2020-03-23 |
|
1 |
|
Rhodium-Catalyzed Enantioselective Hydroselenation of Heterobicyclic Alkenes 2020-03-20 |
|
1 |
|
Carbene-Catalyzed Reaction of Indolyl Methylenemalononitriles and Enals for Access to Complex Tetrahydrocarbazoles 2020-03-19 |
|
0.33 |
|
Direct Synthesis of Chiral NH Lactams via Ru-Catalyzed Asymmetric Reductive Amination/Cyclization Cascade of Keto Acids/Esters 2020-03-19 |
|
1 |
|
NHC-Catalyzed Cascade Reaction between β-Methyl Enals and Dienones for Quick Construction of Complex Multicyclic Lactones 2020-03-19 |
|
0.77 |
|
Total Synthesis of (±)-11-O-Debenzoyltashironin via Palladium-Catalyzed 5-endo Ene-yne Cyclization Enabled trans-5–6 Ring Fusion 2020-03-19 |
|
1 |
|
Bismuth(III)-Catalyzed Sequential Enamine–Imine Tautomerism/2-Aza-Cope Rearrangement of Stable β-Enaminophosphonates: One-Pot Synthesis of β-Aminophosphonates 2020-03-18 |
|
1 |
|
Chartspiroton, a Tetracyclic Spiro-naphthoquinone Derivative from a Medicinal Plant Endophytic Streptomyces 2020-03-18 |
|
1 |
|
Hydride Transfer Initiated Redox-Neutral Cascade Cyclizations of Aurones: Facile Access to [6,5] Spirocycles 2020-03-18 |
|
1 |
|
Hyperprins A and B, Two Complex Meroterpenoids from Hypericum przewalskii 2020-03-18 |
|
1 |
|
Iron-Catalyzed Silylation of (Hetero)aryl Chlorides with Et3SiBpin 2020-03-18 |
|
1 |
|
Phosphine-Catalyzed Cascade Michael Addition/[4+2] Cycloaddition Reaction of Allenoates and 2-Arylidene-1,3-indanediones 2020-03-18 |
|
1 |
|
Rhodium(III)-Catalyzed Oxidative Annulation of 4-Aminoquinolines and Acrylate through Two Consecutive C(sp2)–H Activations 2020-03-18 |
|
0.92 |
|
Visible-Light-Driven Radical Multicomponent Reaction of 2-Vinylanilines, Sulfonyl Chlorides, and Sulfur Ylides for Synthesis of Indolines 2020-03-18 |
|
1 |
|
Direct Hiyama Cross-Coupling of (Hetero)arylsilanes with C(sp2)–H Bonds Enabled by Cobalt Catalysis 2020-03-17 |
|
0.89 |
|
Fast and Low-Cost Purification Strategy for Oligosaccharide Synthesis Based on a Hop-On/Off Carrier 2020-03-17 |
|
1 |
|
Stereospecific Electrophilic Fluorocyclization of α,β-Unsaturated Amides with Selectfluor 2020-03-16 |
|
0.75 |
|
C–O Bond Silylation Catalyzed by Iron: A General Method for the Construction of Csp2–Si Bonds 2020-03-13 |
|
1 |
|
Ganoderma cochlear Metabolites as Probes to Identify a COX-2 Active Site and as in Vitro and in Vivo Anti-Inflammatory Agents 2020-03-13 |
|
1 |
|
Kinetic Resolution of Propargylic Ethers via [2,3]-Wittig Rearrangement to Synthesize Chiral α-Hydroxyallenes 2020-03-13 |
|
1 |
|
Tuning Biradical Character to Enable High and Balanced Ambipolar Charge Transport in a Quinoidal π-System 2020-03-13 |
|
1 |
|
Highly Chemoselective and Enantioselective Synthesis of 3,4-2H-Pyrindin-2-ones by an NHC-Catalyzed [3 + 3] Cyclization 2020-03-11 |
|
1 |
|
Visible-Light-Driven Copper-Catalyzed C(sp3)–O Cross-Coupling of Benzylic Radicals with Phenols 2020-03-11 |
|
1 |
|
Highly Enantioselective [3 + 2] Annulation of 3-Butynoates with β-Trifluoromethyl Enones Promoted by an Amine−Phosphine Binary Catalytic System 2020-03-10 |
|
0.44 |
|
Three-Component Minisci Reaction with 1,3-Dicarbonyl Compounds Induced by Visible Light 2020-03-10 |
|
1 |
|
Visible Light Induced Cyclization to Spirobi[indene] Skeletons from Functionalized Alkylidienecyclopropanes 2020-03-10 |
|
1 |
|
Density Functional Theory Mechanistic Study of Ni-Catalyzed Reductive Alkyne–Alkyne Cyclodimerization: Oxidative Cyclization versus Outer-Sphere Proton Transfer 2020-03-09 |
|
1 |
|
Intermolecular Vicinal Diaminative Assembly of Tetrahydroquinoxalines via Metal-free Oxidative [4 + 2] Cycloaddition Strategy 2020-03-09 |
|
1 |
|
Yb(OTf)3-Catalyzed Alkyne–Carbonyl Metathesis–Oxa-Michael Addition Relay for Diastereoselective Synthesis of Functionalized Naphtho[2,1-b]furans 2020-03-09 |
|
1 |
|
Highly Chemo-, Site-, and Enantioseletive para C–H Aminoalkylation of N-Monosubstituted Aniline Derivatives Affording 3-Amino-2-oxindoles 2020-03-06 |
|
1 |
|
Ligand-Enabled Ni–Al Bimetallic Catalysis for Nonchelated Dual C–H Annulation of Arylformamides and Alkynes 2020-03-06 |
|
1 |
|
Organocatalytic Enantioselective Construction of Heterocycle-Substituted Styrenes with Chiral Atropisomerism 2020-03-06 |
|
1 |
|
Biosynthesis of the Prenylated Salicylaldehyde Flavoglaucin Requires Temporary Reduction to Salicyl Alcohol for Decoration before Reoxidation to the Final Product 2020-03-05 |
|
0.20 |
|
Directing-Group-Enabled Cycloaddition of Azides and Alkynes toward Functionalized Triazoles 2020-03-05 |
|
1 |
|
Visible-Light-Mediated β-C–H gem-Difluoroallylation of Aldehydes and Cyclic Ketones through C–F Bond Cleavage of 1-Trifluoromethyl Alkenes 2020-03-05 |
|
1 |
|
Catalytic Annulation of Alkynyl 1,2-Diketone Leading to Hydroxy Spirocyclopenteneindenedione: An Organic Dye with Strong Crystallization-Induced Emission and Data Storage Application 2020-03-04 |
|
1 |
|
Dimericchalasine A and Amichalasines D and E: Unexpected Cytochalasan Homodimer and Heterotrimers from Aspergillus micronesiensis PG-1 2020-03-04 |
|
1 |
|
Kinetically Controlled Radical Addition/Elimination Cascade: From Alkynyl Aziridine to Fluorinated Allenes 2020-03-04 |
|
1 |
|
Nickel-Catalyzed Claisen Condensation Reaction between Two Different Amides 2020-03-04 |
|
0.50 |
|
Electrochemical Synthesis of α-Ketoamides under Catalyst-, Oxidant-, and Electrolyte-Free Conditions 2020-03-03 |
|
1 |
|
Mesoionic Carbene–Iridium Complex Catalyzed Ortho-Selective Hydrogen Isotope Exchange of Anilines with High Functional Group Tolerance 2020-03-03 |
|
1 |
|
Selective Cross-Dehydrogenative C(sp3)–H Arylation with Arenes 2020-03-03 |
|
1 |
|
Visible-Light-Driven Nitrogen Radical-Catalyzed [3 + 2] Cyclization of Vinylcyclopropanes and N-Tosyl Vinylaziridines with Alkenes 2020-03-03 |
|
1 |
|
Arenesulfonyl Fluoride Synthesis via Copper-Catalyzed Fluorosulfonylation of Arenediazonium Salts 2020-03-02 |
|
1 |
|
Isothiourea and Brønsted Acid Cooperative Catalysis: Enantioselective Construction of Dihydropyridinones 2020-03-02 |
|
1 |
|
Competitive Selection of Conformation Chirality of Water-Soluble Pillar[5]arene Induced by Amino Acid Derivatives 2020-02-28 |
|
1 |
|
Highly Enantioselective Ruthenium-Catalyzed Cascade Double Reduction Strategy: Construction of Structurally Diverse Julolidines and Their Analogues 2020-02-28 |
|
1 |
|
Iridium/Acid Cocatalyzed Direct Access to Fused Indoles via Transfer Hydrogenative Annulation of Quinolines and 1,2-Diketones 2020-02-28 |
|
1 |
|
2H-Azirines as Potential Bifunctional Chemical Linkers of Cysteine Residues in Bioconjugate Technology 2020-02-27 |
|
0.94 |
|
Activation of Chiral (Salen)TiCl2 Complex by Phosphorane for the Highly Enantioselective Cyanation of Nitroolefins 2020-02-27 |
|
1 |
|
Electrophilic Hypervalent Trifluoromethylthio-Iodine(III) Reagent 2020-02-27 |
|
1 |
|
Iron–Phosphine Complex-Catalyzed Intramolecular C(sp3)–H Amination of Azides 2020-02-27 |
|
1 |
|
Unraveling the Fungal Strategy for Tetrahydroxanthone Biosynthesis and Diversification 2020-02-27 |
|
1 |
|
Copper-Catalyzed Disulfonation of Terminal Alkynes with Sodium Arylsulfinates 2020-02-26 |
|
1 |
|
Iridium(III)-Catalyzed C–H Amidation/Cyclization of NH-Sulfoximines with N-Alkoxyamides: Formation of Thiadiazine 1-Oxides 2020-02-26 |
|
1 |
|
Construction of Polyfunctionalized 6–5–5 Fused Tricyclic Carbocycles via One-Pot Sequential Semipinacol Rearrangement/Michael Addition/Henry Reaction 2020-02-25 |
|
1 |
|
Iron-Catalyzed Reductive Vinylation of Tertiary Alkyl Oxalates with Activated Vinyl Halides 2020-02-25 |
|
1 |
|
Protecting-Group-Free Total Syntheses of (±)-Norascyronones A and B 2020-02-25 |
|
1 |
|
Total Synthesis of (−)-Gardmultimine A 2020-02-25 |
|
1 |
|
HNTf2-Catalyzed Synthesis of Hydrodibenzofurans by an Epoxidation/Semipinacol Rearrangement Cascade 2020-02-24 |
|
1 |
|
Leptosperols A and B, Two Cinnamoylphloroglucinol–Sesquiterpenoid Hybrids from Leptospermum scoparium: Structural Elucidation and Biomimetic Synthesis 2020-02-24 |
|
1 |
|
Organocatalytic Asymmetric Three-Component Povarov Reactions of Anilines and Aldehydes 2020-02-21 |
|
1 |
|
Rh(III)-Catalyzed Relay Double Carbenoid Insertion and Diannulation of Sulfoximine Benzamides with α-Diazo Carbonyl Compounds: Access to Furo[2,3-c]isochromenes 2020-02-21 |
|
1 |
|
Water Compatible Hypophosphites-d2 Reagents: Deuteration Reaction via Deutero-deiodination in Aqueous Solution 2020-02-21 |
|
1 |
|
Palladium-Catalyzed Three-Component Coupling Reaction of o-Bromobenzaldehyde, N-Tosylhydrazone, and Methanol 2020-02-20 |
|
1 |
|
Redox Cyclization of Amides and Sulfonamides with Nitrous Oxide for Direct Synthesis of Heterocycles 2020-02-20 |
|
1 |
|
Visible-Light Mediated Hydrosilylative and Hydrophosphorylative Cyclizations of Enynes and Dienes 2020-02-20 |
|
1 |
|
C(sp2)–H Bond Multiple Functionalization in Air for Construction of Tetrahydrocarbazoles with Continuous Quaternary Carbons and Polycyclic Diversification 2020-02-19 |
|
1 |
|
Cobalt-Catalyzed C–H Acetoxylation of Phenols with Removable Monodentate Directing Groups: Access to Pyrocatechol Derivatives 2020-02-19 |
|
0.89 |
|
Cycloaddition of Trifluoroacetaldehyde N-Triftosylhydrazone (TFHZ-Tfs) with Alkynes for Synthesizing 3-Trifluoromethylpyrazoles 2020-02-19 |
|
1 |
|
Direct Alkoxycarbonylation of Heteroarenes via Cu-Mediated Trichloromethylation and In Situ Alcoholysis 2020-02-19 |
|
1 |
|
Direct Synthesis of Sulfonylated Spiro[indole-3,3′-pyrrolidines] by Silver-Mediated Sulfonylation of Acrylamides Coupled with Indole Dearomatization 2020-02-19 |
|
1 |
|
Enantioselective Synthesis of Axially Chiral Biaryls via Copper-Catalyzed Thiolation of Cyclic Diaryliodonium Salts 2020-02-19 |
|
1 |
|
On-PKS Baeyer–Villiger-Type O-Atom Insertion Catalyzed by Luciferase-Like Monooxygenase OvmO during Olimycin Biosynthesis 2020-02-19 |
|
1 |
|
Sequential C–S and S–N Coupling Approach to Sulfonamides 2020-02-19 |
|
1 |
|
Copper Catalyzed Diastereo- and Enantioselective 1,4-Addition Michael Reaction of 2,3-Dioxopyrrolidines with Nitroalkanes in Aqueous Media 2020-02-18 |
|
1 |
|
Palladium-Catalyzed Four-Component Carbonylative Cyclization Reaction of Trifluoroacetimidoyl Chlorides, Propargyl Amines, and Diaryliodonium Salts: Access to Trifluoromethyl-Containing Trisubstituted Imidazoles 2020-02-18 |
|
0.88 |
|
Diastereoselective Synthesis of Cycloheptannelated Indoles via Lewis-Acid-Catalyzed (4 + 3)-Cyclization of Donor–Acceptor Cyclopropanes 2020-02-17 |
|
1 |
|
Rhodium-Catalyzed Branched and Enantioselective Direct α-Allylic Alkylation of Simple Ketones with Alkynes 2020-02-17 |
|
1 |
|
Flavipesides A–C, PKS-NRPS Hybrids as Pancreatic Lipase Inhibitors from a Marine Sponge Symbiotic Fungus Aspergillus flavipes 164013 2020-02-14 |
|
1 |
|
Intermolecular Trifluoromethyl-Hydrazination of Alkenes Enabled by Organic Photoredox Catalysis 2020-02-14 |
|
1 |
|
Organocatalytic Enantioselective γ-Elimination: Applications in the Preparation of Chiral Peroxides and Epoxides 2020-02-14 |
|
1 |
|
Copper-Catalyzed Remote C(sp3)–H Phosphorothiolation of Sulfonamides and Carboxamides in a Multicomponent Reaction 2020-02-13 |
|
1 |
|
Engineered Biosynthesis of 5/5/6 Type Polycyclic Tetramate Macrolactams in an Ikarugamycin (5/6/5 Type)-Producing Chassis 2020-02-13 |
|
1 |
|
Photocatalytic C–F Bond Borylation of Polyfluoroarenes with NHC-boranes 2020-02-13 |
|
1 |
|
Syntheses of Epoxyguaiane Sesquiterpenes (−)-Englerin A, (−)-Oxyphyllol, (+)-Orientalol E, and (+)-Orientalol F: A Synthetic Biology Approach 2020-02-13 |
|
1 |
|
Enhanced DNA Sensing and Chiroptical Performance by Restriction of Double-Bond Rotation of AIE cis-Tetraphenylethylene Macrocycle Diammoniums 2020-02-12 |
|
1 |
|
Total Synthesis of Dysoxylactam A 2020-02-12 |
|
1 |
|
A Pd-Catalyzed Site-Controlled Isomerization of Terminal Olefins 2020-02-11 |
|
0.88 |
|
Copper-Catalyzed Annulation or Homocoupling of Sulfoxonium Ylides: Synthesis of 2,3-Diaroylquinolines or α,α,β-Tricarbonyl Sulfoxonium Ylides 2020-02-11 |
|
1 |
|
Aspermeroterpenes A–C: Three Meroterpenoids from the Marine-Derived Fungus Aspergillus terreus GZU-31-1 2020-02-10 |
|
1 |
|
Asymmetric Synthesis of Rugulotrosin A 2020-02-10 |
|
1 |
|
Asymmetric Total Synthesis of (−)-Guignardones A and B 2020-02-10 |
|
1 |
|
Synthesis of 17-Deacetoxyl Chromodorolide B Based on a Gold-Catalyzed Alkoxycyclization Reaction 2020-02-10 |
|
1 |
|
Synthesis, Properties, and Reactivity of Bis-BN Phenanthrenes: Stepwise Bromination of the Main Scaffold 2020-02-10 |
|
1 |
|
Visible-Light-Induced Charge Transfer Enables Csp3–H Functionalization of Glycine Derivatives: Access to 1,3-Oxazolidines 2020-02-10 |
|
1 |
|
Copper-Catalyzed Oxidative Thioamination of Maleimides with Amines and Bunte Salts 2020-02-07 |
|
1 |
|
Efficient Strategy for α-Selective Glycosidation of d-Glucosamine and Its Application to the Synthesis of a Bacterial Capsular Polysaccharide Repeating Unit Containing Multiple α-Linked GlcNAc Residues 2020-02-07 |
|
0.80 |
|
Copper-Catalyzed Photoinduced Enantioselective Dual Carbofunctionalization of Alkenes 2020-02-06 |
|
1 |
|
Origins of Unconventional γ Site Selectivity in Palladium-Catalyzed C(sp3)–H Activation and Arylation of Aliphatic Alcohols 2020-02-06 |
|
1 |
|
Rhodium-Catalyzed Remote Isomerization of Alkenyl Alcohols to Ketones 2020-02-06 |
|
1 |
|
Catalytic Asymmetric Conjugate Protosilylation and Protoborylation of 2-Trifluoromethyl Enynes for Synthesis of Functionalized Allenes 2020-02-04 |
|
1 |
|
Cu-Mediated Expeditious Annulation of Alkyl 3-Aminoacrylates with Aryldiazonium Salts: Access to Alkyl N2-Aryl 1,2,3-Triazole-carboxylates for Druglike Molecular Synthesis 2020-02-04 |
|
1 |
|
Homoleptic Bis(trimethylsilyl)amides of Yttrium Complexes Catalyzed Hydroboration Reduction of Amides to Amines 2020-02-04 |
|
1 |
|
Synergistic Dual Directing Groups-Enabled Diastereoselective C–H Cyclopropylation via Rh(III)-Catalyzed Couplings with Cyclopropenyl Alcohols 2020-02-04 |
|
1 |
|
Access to Divergent Fluorinated Enynes and Arenes via Palladium-Catalyzed Ring-Opening Alkynylation of gem-Difluorinated Cyclopropanes 2020-02-03 |
|
1 |
|
Aldehyde as a Traceless Directing Group for Regioselective C–H Alkylation Catalyzed by Rhodium(III) in Air 2020-02-03 |
|
0.83 |
|
Covalent Organic Framework as a Heterogeneous Ligand for the Regioselective Oxidative Heck Reaction 2020-02-03 |
|
1 |
|
Enantioselective Synthesis of 4-Allyl Tetrahydroquinolines via Copper(I) Hydride-Catalyzed Hydroallylation of 1,2-Dihydroquinolines 2020-02-03 |
|
1 |
|
Late-Stage Modification of Tertiary Phosphines via Ruthenium(II)-Catalyzed C–H Alkylation 2020-02-03 |
|
0.90 |
|
Layered Chirality Relay Model in Rh(I)-Mediated Enantioselective C–Si Bond Activation: A Theoretical Study 2020-02-03 |
|
1 |
|
Rhodium(III)-Catalyzed C–H Alkenylation: Access to Maleimide-Decorated Tryptophan and Tryptophan-Containing Peptides 2020-02-03 |
|
1 |
|
Host–Guest Complexation of Perethylated Pillar[6]arene toward Ferrocene Derivatives Both in Solution and Solid State: Different Binding Modes Induced by Minor Structural Changes of Guests 2020-01-31 |
|
1 |
|
Total Syntheses of (+)-Stemarin and the Proposed Structures of Stemara-13(14)-en-18-ol and Stemara-13(14)-en-17-acetoxy-18-ol 2020-01-31 |
|
1 |
|
Dehydrative Cross-Coupling of Allylic Alcohols with Alkynes 2020-01-30 |
|
0.97 |
|
Enantioselective Cu(I)-Catalyzed Cycloaddition of Prochiral Diazides with Terminal or 1-Iodoalkynes 2020-01-30 |
|
1 |
|
Energetic Derivatives of 8-Nitropyrazolo[1,5-a][1,3,5]triazine-2,4,7-triamine: Achieving Balanced Explosives by Fusing Pyrazole with Triazine 2020-01-30 |
|
0.33 |
|
Intramolecular Aromatic C–H Acyloxylation Enabled by Iron Photocatalysis 2020-01-30 |
|
1 |
|
Melipatulinones A–C, Three Lignan–Phloroglucinol Hybrids from Melicope patulinervia 2020-01-30 |
|
1 |
|
Synthesis of Functionalized Vinylsilanes via Metal-Free Dehydrogenative Silylation of Enamides 2020-01-30 |
|
1 |
|
Synthesis of Multifunctional 2-Aminobenzimidazoles on DNA via Iodine-Promoted Cyclization 2020-01-30 |
|
0.70 |
|
Genome Mining and Biosynthesis of Primary Amine-Acylated Desferrioxamines in a Marine Gliding Bacterium 2020-01-29 |
|
1 |
|
Access to Benzoxazepines and Fully Substituted Indoles via HDDA Coupling 2020-01-28 |
|
1 |
|
Continuous Flow-Enabled Synthesis of Bench-Stable Bicyclo[1.1.1]pentane Trifluoroborate Salts and Their Utilization in Metallaphotoredox Cross-Couplings 2020-01-28 |
|
0.36 |
|
Enantioselective Imino-Ene Reaction of N-Sulfonyl Ketimines with Silyl Enol Ethers: Access to Chiral Benzosultams 2020-01-28 |
|
1 |
|
Enantioselective Synthesis of Spiroindolines via Cascade Isomerization/Spirocyclization/Dearomatization Reaction 2020-01-28 |
|
1 |
|
Synthesis of Monofluoroalkenes through Visible-Light-Promoted Defluorinative Alkylation of gem-Difluoroalkenes with 4-Alkyl-1,4-dihydropyridines 2020-01-28 |
|
1 |
|
Harnessing Thiol as a Benzyl Reagent for Photocatalytic Reductive Benzylation of Imines 2020-01-27 |
|
0.50 |
|
Radical Aza-Cyclization of α-Imino-oxy Acids for Synthesis of Alkene-Containing N-Heterocycles via Dual Cobaloxime and Photoredox Catalysis 2020-01-27 |
|
1 |
|
Copper-Catalyzed Asymmetric Propargylic Alkylation with Oxindoles: Diastereo- and Enantioselective Construction of Vicinal Tertiary and All-Carbon Quaternary Stereocenters 2020-01-24 |
|
1 |
|
Fulleropillar[4]arene: The Synthesis and Complexation Properties 2020-01-24 |
|
1 |
|
Merging Visible Light Photocatalysis and l-/d-Proline Catalysis: Direct Asymmetric Oxidative Dearomatization of 2-Arylindoles To Access C2-Quaternary Indolin-3-ones 2020-01-24 |
|
1 |
|
Morindolestatin, Naturally Occurring Dehydromorpholinocarbazole Alkaloid from Soil-Derived Bacterium of the Genus Streptomyces 2020-01-24 |
|
1 |
|
Remote Directed Isocyanation of Unactivated C(sp3)–H Bonds: Forging Seven-Membered Cyclic Ureas Enabled by Copper Catalysis 2020-01-24 |
|
1 |
|
Ruthenium Carbene-Mediated Construction of Strained Allenes via the Enyne Cross-Metathesis/Cyclopropanation of 1,6-Enynes 2020-01-24 |
|
1 |
|
Synthesis of Stereodefined Trisubstituted Alkenyl Silanes Enabled by Borane Catalysis and Nickel Catalysis 2020-01-24 |
|
1 |
|
Catalytic Diastereoselective [5 + 2] Annulation of N-Acryloyl Indoles with Cyclic Sulfonyl Enamides: Facile Access to Isoeburnamonine 2020-01-23 |
|
1 |
|
Heterologous Expression Leads to Discovery of Diversified Lobophorin Analogues and a Flexible Glycosyltransferase 2020-01-23 |
|
1 |
|
Open-Air Stereoselective Construction of C-Aryl Glycosides 2020-01-23 |
|
0.88 |
|
Regioselective Wacker-Type Oxidation of Internal Olefins in tBuOH Using Oxygen as the Sole Oxidant and tBuONO as the Organic Redox Cocatalyst 2020-01-23 |
|
1 |
|
Selective Dehydrogenative Acylation of Enamides with Aldehydes Leading to Valuable β-Ketoenamides 2020-01-23 |
|
0.93 |
|
Synthesis of 4,7-Difunctionalized Indoles via Imino Exchange and Sulfinyl Migration 2020-01-23 |
|
1 |
|
Visible-Light-Promoted Photocatalyst-Free Hydroacylation and Diacylation of Alkenes Tuned by NiCl2·DME 2020-01-23 |
|
1 |
|
Organocatalytic Cascade β-Functionalization/Aromatization of Pyrrolidines via Double Hydride Transfer 2020-01-22 |
|
1 |
|
Palladium-Catalyzed Carbonylative Synthesis of α-Branched Enones from Aryl Iodides and Arylallenes 2020-01-22 |
|
0.88 |
|
Practical Method for Reductive Deuteration of Ketones with Magnesium and D2O 2020-01-22 |
|
1 |
|
Biomimetic Total Syntheses of Sanctis A–B with Structure Revision 2020-01-21 |
|
1 |
|
Cu(I)-Catalyzed Enantioselective Alkynylation of Thiochromones 2020-01-21 |
|
1 |
|
Iridium-Catalyzed Asymmetric Hydrogenation of γ- and δ-Ketoacids for Enantioselective Synthesis of γ- and δ-Lactones 2020-01-21 |
|
1 |
|
Nickel-Catalyzed Deaminative Acylation of Activated Aliphatic Amines with Aromatic Amides via C–N Bond Activation 2020-01-21 |
|
0.83 |
|
Catalytic Asymmetric Tandem Cycloisomerization/[5+2] Cycloaddition Reaction of N-Aryl Nitrone Alkynes with Methyleneindolinones 2020-01-17 |
|
1 |
|
Photo/N-Heterocyclic Carbene Co-catalyzed Ring Opening and γ-Alkylation of Cyclopropane Enal 2020-01-17 |
|
1 |
|
Regioselective Synthesis of 3-Trifluoromethylpyrazole by Coupling of Aldehydes, Sulfonyl Hydrazides, and 2-Bromo-3,3,3-trifluoropropene 2020-01-17 |
|
1 |
|
Cobalt-Catalyzed Z to E Isomerization of Alkenes: An Approach to (E)-β-Substituted Styrenes 2020-01-16 |
|
1 |
|
Metal-Free sp3 C-SCF3 Coupling Reactions between Cycloketone Oxime Esters and S-trifluoromethyl 4-Methylbenzenesulfonothioate 2020-01-16 |
|
1 |
|
Photoinduced C(sp2)–H/C(sp2)–H Cross-Coupling of Alkenes: Direct Synthesis of 1,3-Dienes 2020-01-16 |
|
1 |
|
Reverse Turn Foldamers: An Expanded β-Turn Motif Reinforced by Double Hydrogen Bonds 2020-01-16 |
|
0.43 |
|
Rhodium-Catalyzed ortho-Selective Carbene C–H Insertion of Unprotected Phenols Directed by a Transient Oxonium Ylide Intermediate 2020-01-16 |
|
1 |
|
Synthesis of Difluoroalkylated Benzofuran, Benzothiophene, and Indole Derivatives via Palladium-Catalyzed Cascade Difluoroalkylation and Arylation of 1,6-Enynes 2020-01-16 |
|
1 |
|
[3,3]-Sigmatropic Rearrangement/Haller–Bauer Reaction of Aryl Sulfoxides and Selenoxides with Difluoroenoxysilanes: Access to CF2H-Containing Chalcogenides 2020-01-16 |
|
1 |
|
Asymmetric Umpolung Hydrogenation and Deuteration of Alkenes Catalyzed by Nickel 2020-01-15 |
|
0.67 |
|
Enantioselective Synthesis of Spirorhodanine-Pyran Derivatives via Organocatalytic [3 + 3] Annulation Reactions between Pyrazolones and Rhodanine-Derived Ketoesters 2020-01-15 |
|
1 |
|
Incarnolides A and B, Two Schinortriterpenoids with a Tricyclo[9.2.1.02,8]tetradecane-Bridged System from Schisandra incarnata 2020-01-15 |
|
1 |
|
Tunable Gold(I)-Catalyzed [4 + 3] Cycloaddition for Divergent Synthesis of Furan-Fused N,O-Heterocycles 2020-01-15 |
|
1 |
|
Electrochemical Oxidative Oxydihalogenation of Alkynes for the Synthesis of α,α-Dihaloketones 2020-01-14 |
|
1 |
|
Palladium-Catalyzed Ligand-Free Double Cyclization Reactions for the Synthesis of 3-(1′-Indolyl)-phthalides 2020-01-14 |
|
1 |
|
Rhodium-Catalyzed Enantioselective Anti-Markovnikov Hydroformylation of α-Substituted Acryl Acid Derivatives 2020-01-14 |
|
1 |
|
Synthesis of Tertiary Benzylic Nitriles via Nickel-Catalyzed Markovnikov Hydrocyanation of α-Substituted Styrenes 2020-01-14 |
|
1 |
|
C- to N-Center Remote Heteroaryl Migration via Electrochemical Initiation of N Radical by Organic Catalyst 2020-01-10 |
|
1 |
|
Nickel-Catalyzed, para-Selective, Radical-Based Alkylation of Aromatic Ketones 2020-01-10 |
|
1 |
|
Chalcone-Based Pyridinium Salts and Their Diastereoselective Dearomatization To Access Bibridged Benzoazepines 2020-01-09 |
|
1 |
|
Cobalt-Catalyzed Migrational Isomerization of Styrenes 2020-01-09 |
|
1 |
|
Copper-Catalyzed Asymmetric Hydrosilylation of β-Nitroethyl Aryl Ketones 2020-01-09 |
|
1 |
|
Crokonoids A–C, A Highly Rearranged and Dual-Bridged Spiro Diterpenoid and Two Other Diterpenoids from Croton kongensis 2020-01-09 |
|
1 |
|
Dimethylformamide-Modulated Kdo Glycosylation for Stereoselective Synthesis of α-Kdo Glycosides 2020-01-09 |
|
1 |
|
Photoredox Oxo-C(sp3)–H Bond Functionalization via in Situ Cu(I)-Acetylide Catalysis 2020-01-09 |
|
1 |
|
Reductase of Mutanobactin Synthetase Triggers Sequential C–C Macrocyclization, C–S Bond Formation, and C–C Bond Cleavage 2020-01-09 |
|
1 |
|
Rh-Catalyzed Asymmetric Hydrogenation of Unsaturated Medium-Ring NH Lactams: Highly Enantioselective Synthesis of N-Unprotected 2,3-Dihydro-1,5-benzothiazepinones 2020-01-09 |
|
1 |
|
CF3SO2Na-Mediated, UV-Light-Induced Friedel–Crafts Alkylation of Indoles with Ketones/Aldehydes and Bioactivities of Products 2020-01-08 |
|
1 |
|
Chiral Discrimination of Varied Ammonium Compounds through 1H NMR Using a Binuclear Ti Complex Sensor 2020-01-08 |
|
1 |
|
DFT Mechanistic Account for the Site Selectivity of Electron-Rich C(sp3)–H Bond in the Manganese-Catalyzed Aminations 2020-01-08 |
|
1 |
|
Enantioselective NHC-Catalyzed [3+3] Annulation of α-Bromoenals with 2-Aminobenzimidazoles 2020-01-08 |
|
1 |
|
Intermolecular Reductive Heck Reaction of Unactivated Aliphatic Alkenes with Organohalides 2020-01-08 |
|
0.95 |
|
Nickel-Catalyzed Asymmetric Hydrocyanation of Allenes 2020-01-08 |
|
1 |
|
Pentafluorophenyl Esters: Highly Chemoselective Ketyl Precursors for the Synthesis of α,α-Dideuterio Alcohols Using SmI2 and D2O as a Deuterium Source 2020-01-08 |
|
0.63 |
|
C–H Insertion by Alkylidene Carbenes To Form 1,2,3-Triazines and Anionic [3 + 2] Dipolar Cycloadditions To Form Tetrazoles: Crucial Roles of Stereoelectronic and Steric Effects 2020-01-07 |
|
0.50 |
|
Heterogeneous Carbon Nitrides Photocatalysis Multicomponent Hydrosulfonylation of Alkynes To Access β-Keto Sulfones with the Insertion of Sulfur Dioxide in Aerobic Aqueous Medium 2020-01-07 |
|
1 |
|
Palladium-Catalyzed Synthesis of 1,2-Diketones from Aryl Halides and Organoaluminum Reagents Using tert-Butyl Isocyanide as the CO Source 2020-01-07 |
|
0.50 |
|
Precise Construction of SCF2H or SeCF2H Groups on Heteroarenes Generated in Situ from CF3-Containing 1,3-Enynes 2020-01-07 |
|
1 |
|
Revision of the Structure of Hypatulone A by NMR, Computations, and Biosynthetic Considerations 2020-01-07 |
|
0.50 |
|
Visible-Light-Driven Dearomatization Reaction toward the Formation of Spiro[4.5]deca-1,6,9-trien-8-ones 2020-01-07 |
|
1 |
|
Visible-Light-Induced Deoxygenation/Defluorination Protocol for Synthesis of γ,γ-Difluoroallylic Ketones 2020-01-07 |
|
1 |
|
Asymmetric Total Synthesis and Biological Evaluation of the Natural PDE4 Inhibitor Toddacoumalone 2020-01-06 |
|
1 |
|
Lewis Acid Catalyzed Electrophilic Aminomethyloxygenative Cyclization of Alkynols with N,O-Aminals 2020-01-06 |
|
1 |
|
NHC-Catalyzed Radical Trifluoromethylation Enabled by Togni Reagent 2020-01-06 |
|
1 |
|
Synthesis of Tribenzo[b,d,f]azepines via Cascade π-Extended Decarboxylative Annulation Involving Cyclic Diaryliodonium Salts 2020-01-06 |
|
1 |
|
Total Synthesis of Galanthamine and Lycoramine Featuring an Early-Stage C–C and a Late-Stage Dehydrogenation via C–H Activation 2020-01-06 |
|
1 |
|
Construction of 2-Arylbenzo[4,5]thieno[2,3-d]thiazole Skeleton via CuCl/S-Mediated Three-Component Reaction 2020-01-02 |
|
0.90 |
|
Pd-Catalyzed Asymmetric Hydroalkylation of 1,3-Dienes: Access to Unnatural α-Amino Acid Derivatives Containing Vicinal Quaternary and Tertiary Stereogenic Centers 2020-01-02 |
|
1 |
|
Rh(III)-Catalyzed Tandem Acylmethylation/Nitroso Migration/Cyclization of N-Nitrosoanilines with Sulfoxonium Ylides in One Pot: Approach to 3-Nitrosoindoles 2020-01-02 |
|
1 |
|
Enantioselective Synthesis of Multifunctionalized 4H-Pyrans via Formal [4 + 2] Annulation Process by Bifunctional Phosphonium Salt Catalysis 2019-12-31 |
|
1 |
|
Genetic Manipulation of an Aminotransferase Family Gene dtlA Activates Youssoufenes in Marine-Derived Streptomyces youssoufiensis 2019-12-31 |
|
1 |
|
Silver-Catalyzed Selective Multicomponent Coupling Reactions of Arynes with Nitriles and Isonitriles 2019-12-31 |
|
0.40 |
|
CuSO4-Catalyzed Tandem C(sp3)–H Insertion Cyclization of Toluenes with Isonitriles to Form Indoles 2019-12-30 |
|
1 |
|
Electrochemical Synthesis of 1-Naphthols by Intermolecular Annulation of Alkynes with 1,3-Dicarbonyl Compounds 2019-12-30 |
|
1 |
|
Practical Synthesis of Benzimidazo[1,2-a]quinolines via Rh(III)-Catalyzed C–H Activation Cascade Reaction from Imidamides and Anthranils 2019-12-30 |
|
1 |
|
Rh(III)-Catalyzed Coupling of Acrylic Acids and Ynenones via Olefinic C–H Activation and Michael Addition 2019-12-30 |
|
1 |
|
Silver-Catalyzed Annulation of Arynes with Nitriles for Synthesis of Structurally Diverse Quinazolines 2019-12-30 |
|
0.40 |
|
Synthesis of 2H-Chromenes via Unexpected [4 + 2] Annulation of Alkynyl Thioethers with o-Hydroxybenzyl Alcohols 2019-12-30 |
|
1 |
|
Botryotins A–H, Tetracyclic Diterpenoids Representing Three Carbon Skeletons from a Deep-Sea-Derived Botryotinia fuckeliana 2019-12-27 |
|
1 |
|
Enantioselective 1,2-Alkylhydroxylmethylation of Alkynes via Chromium/Cobalt Cocatalysis 2019-12-27 |
|
1 |
|
Organocatalytic Double Ugi Reaction with Statistical Amplification of Product Enantiopurity: A Linker Cleavage Approach To Access Highly Enantiopure Ugi Products 2019-12-27 |
|
0.75 |
|
Synthesis of 2-Arylpiperidines via Pd-Catalyzed Arylation of Aza-Achmatowicz Rearrangement Products with Arylboronic Acids 2019-12-27 |
|
0.29 |
|
Highly Enantioselective Nickel-Catalyzed Hydrocyanation of Disubstituted Methylenecyclopropanes Enabled by TADDOL-based Diphosphite Ligands 2019-12-26 |
|
1 |
|
Total Synthesis of Caesalpinnone A 2019-12-26 |
|
1 |
|
Herpotrichones A and B, Two Intermolecular [4 + 2] Adducts with Anti-Neuroinflammatory Activity from a Herpotrichia Species 2019-12-24 |
|
0.78 |
|
Mechanistic Insights into La-Catalyzed Amidation of Aldehyde with Amine 2019-12-24 |
|
1 |
|
Phosphine-Catalyzed (3 + 2)/(3 + 2) Sequential Annulation of γ-Vinyl Allenoates: Access to Fused Carbocycles 2019-12-24 |
|
1 |
|
Phosphine-Mediated MBH-Type/Umpolung Addition Domino Sequence: Divergent Construction of Coumarins 2019-12-24 |
|
1 |
|
Probing the Interconversion of Labdane Lactones from the Chinese Liverwort Pallavicinia ambigua 2019-12-24 |
|
1 |
|
Complementary C–H Functionalization Mode of Benzoylacetonitriles: Computer-Augmented Study of a Regio- and Stereoselective Synthesis of Functionalized Benzofulvenes 2019-12-23 |
|
0.60 |
|
Enantioselective Synthesis of Fused Polycyclic Tropanes via Dearomative [3 + 2] Cycloaddition Reactions of 2-Nitrobenzofurans 2019-12-23 |
|
1 |
|
Palladium-Catalyzed Cascade Reactions of 2-(Cyanomethoxy)chalcones with Arylboronic Acids: Selective Synthesis of Emissive Benzofuro[2,3-c]pyridines 2019-12-23 |
|
1 |
|
Benzene-1,3,5-triyl Triformate (TFBen)-Promoted Palladium-Catalyzed Carbonylative Synthesis of 2-Oxo-2,5-dihydropyrroles from Propargyl Amines 2019-12-20 |
|
0.83 |
|
Direct Use of Unprotected Aliphatic Amines to Generate N-Heterocycles via β-C–H Malonylation with Iodonium Ylide 2019-12-20 |
|
1 |
|
Employing TosMIC as a C1N1 “Two-Atom Synthon” in Imidazole Synthesis by Neighboring Group Assistance Strategy 2019-12-20 |
|
1 |
|
Exploring Aporphine as Anti-inflammatory and Analgesic Lead from Dactylicapnos scandens 2019-12-20 |
|
1 |
|
Selective Insertion of Alkynes into C–C σ Bonds of Indolin-2-ones: Transition-Metal-Free Ring Expansion Reactions to Seven-Membered-Ring Benzolactams or Chromone Derivatives 2019-12-20 |
|
1 |
|
π-Extended C2-Symmetric Double NBN-Heterohelicenes with Exceptional Luminescent Properties 2019-12-20 |
|
1 |
|
Cu-Catalyzed Alkylarylation of Vinylarenes with Masked Alkyl Electrophiles 2019-12-19 |
|
1 |
|
On-Resin Passerini Reaction toward C-Terminal Photocaged Peptides 2019-12-19 |
|
1 |
|
Visible-Light-Induced para-Selective C(sp2)–H Difluoroalkylation of Diverse (Hetero)aromatic Carbonyls 2019-12-19 |
|
1 |
|
Decarboxylative Borylation of mCPBA-Activated Aliphatic Acids 2019-12-18 |
|
1 |
|
Highly Enantioselective Construction of Dihydrooxazines via Pd-Catalyzed Asymmetric Carboetherification 2019-12-18 |
|
1 |
|
Palladium and Brønsted Acid Co-Catalyzed Biginelli-like Multicomponent Reactions via in Situ-Generated Cyclic Enol Ether: Access to Spirofuran-hydropyrimidinones 2019-12-18 |
|
1 |
|
Stable Double and Quadruple [5]Helicene Derivatives: Synthesis, Structural Analysis, and Physical Properties 2019-12-18 |
|
1 |
|
Desymmetrization of Prochiral Cyclopentenes Enabled by Enantioselective Palladium-Catalyzed Oxidative Heck Reaction 2019-12-17 |
|
0.25 |
|
Palladium-Catalyzed Three-Component Tandem Coupling–Carboannulation Reaction Leading to Polysubstituted [60]Fullerene-Fused Cyclopentanes 2019-12-17 |
|
1 |
|
2,3-Dicyano-5,6-dichlorobenzoquinone-Mediated and Selective C–O and C–C Cross-Couplings of Phenols and Porphyrins 2019-12-16 |
|
1 |
|
Alkaline-Earth Metal Catalyzed Dehydrative Allylic Alkylation 2019-12-16 |
|
0.95 |
|
Catalytic Enantioselective Synthesis of 1,4-Benzodioxepines 2019-12-16 |
|
1 |
|
Chiral ScIII–N,N′-Dioxide-Catalyzed 1,3-Dipolar Cycloaddition of Diaziridines with Chalcones 2019-12-13 |
|
1 |
|
Enantio- and Diastereoselective Synthesis of Chromeno[4,3-b]pyrrole Derivatives Bearing Tetrasubstituted Chirality Centers through Carbene Catalyzed Cascade Reactions 2019-12-13 |
|
0.86 |
|
Formation of Terrestric Acid in Penicillium crustosum Requires Redox-Assisted Decarboxylation and Stereoisomerization 2019-12-13 |
|
0.20 |
|
Pd(II)-Catalyzed Regioselective Multiple C–H Arylations of 1-Naphthamides with Cyclic Diaryliodonium Salts: One-Step Access to [4]- and [5]Carbohelicenes 2019-12-13 |
|
1 |
|
RhIII-Catalyzed Synthesis of Cyclopenta[b]carbazoles via Cascade C–H/C–C Bond Cleavage and Cyclization Reactions: Using Amide as a Traceless Directing Group 2019-12-13 |
|
1 |
|
Construction of Bisindolines via Oxidative Coupling Cyclization 2019-12-12 |
|
1 |
|
Copper(II)-Catalyzed C-H Nitrogenation/Annulation Cascade of Ketene N,S-Acetals with Aryldiazonium Salts: A Direct Access to N2-Substituted Triazole and Triazine Derivatives 2019-12-12 |
|
1 |
|
Detoxification of Plant Aromatic Abietanoids via Cleavage of the Benzene Ring into 11,12-Seco-diterpene Polyenes by a Specialist Insect of Leucosceptrum canum 2019-12-12 |
|
1 |
|
Directed Biosynthesis of Iso-aclacinomycins with Improved Anticancer Activity 2019-12-12 |
|
1 |
|
Electrochemically Enabled Double C–H Activation of Amides: Chemoselective Synthesis of Polycyclic Isoquinolinones 2019-12-12 |
|
1 |
|
Jatrofolianes A and B: Two Highly Modified Lathyrane Diterpenoids from Jatropha gossypiifolia 2019-12-12 |
|
1 |
|
Preparation of 4-Diazoisoquinolin-3-ones via Dimroth Rearrangement and Their Extension to 4-Aryltetrahydroisoquinolin-3-ones 2019-12-12 |
|
1 |
|
Structural Revision and Absolute Configuration of Burnettramic Acid A 2019-12-12 |
|
1 |
|
Synthesis and Semiconducting Characteristics of the BF2 Complexes of Bisbenzothiophene-Fused Azadipyrromethenes 2019-12-12 |
|
1 |
|
(3 + 1) Annulation/Rearrangement Cascade of C,N-Cyclic Azomethine Imines and 3-Chlorooxindoles: Construction of Hexahydroindeno[2,1-c]pyrazole Spirooxindole Frameworks 2019-12-11 |
|
1 |
|
Base-Promoted Nitrile–Alkyne Domino-Type Cyclization: A General Method to Trisubstituted Imidazoles 2019-12-10 |
|
1 |
|
Chiral Bis(oxazoline)–Copper Complex Catalyzed Asymmetric Alkenylation of Isatin Imines and 3-Vinylindoles for Construction of Optically Active 3-Alkenyl-3-aminooxindoles 2019-12-10 |
|
1 |
|
Diastereo- and Enantioselective Synthesis of Quaternary α-Amino Acid Precursors by Copper-Catalyzed Propargylation 2019-12-10 |
|
1 |
|
Selectfluor-Mediated Stereoselective [1 + 1 + 4 + 4] Dimerization of Styrylnaphthols 2019-12-10 |
|
1 |
|
A Tetraazapentacene–Pyrene Belt: Toward Synthesis of N-Doped Zigzag Carbon Nanobelts 2019-12-09 |
|
1 |
|
Cp*RhIII-Catalyzed Sulfonamide-Directed Ortho Arene C–H Carbenoid Functionalization with Pyridotriazoles 2019-12-09 |
|
1 |
|
Palladium-Catalyzed Domino Heck/C–H Activation/Decarboxylation: A Rapid Entry to Fused Isoquinolinediones and Isoquinolinones 2019-12-09 |
|
1 |
|
Regiodivergent Vinylogous–Cyclization Reactions of Cyclic α-Amide Enone Acceptors: Synthesis of Highly Enantioenriched Heterobicyclic Structures 2019-12-09 |
|
1 |
|
Catalytic Direct Regioselective Synthesis of Phosphonylated Tetrazoles from Aryl Diazonium Salts and Seyferth-Gilbert Reagent 2019-12-06 |
|
1 |
|
Organic Photoredox-Catalyzed Decarboxylative Trifluoromethylselenolation of Aliphatic Carboxylic Acids with [Me4N][SeCF3] 2019-12-06 |
|
1 |
|
Pd(0)-Catalyzed Intramolecular “Ylide-Ullmann-Type” Cyclization of Carbonyl-Stabilized Phosphonium Ylides and Access to Phosphachromones by Exocyclic P–C Cleavage 2019-12-06 |
|
1 |
|
Visible-Light-Enabled Oxidative Coupling of Alkenes with Dialkylformamides To Access Unsaturated Amides 2019-12-06 |
|
1 |
|
Highly Diastereo- and Enantioselective Ir-Catalyzed Hydrogenation of 2,3-Disubstituted Quinolines with Structurally Fine-Tuned Phosphine–Phosphoramidite Ligands 2019-12-05 |
|
1 |
|
Redox-Neutral [4 + 2] Annulation of N-Methoxybenzamides with Alkynes Enabled by an Osmium(II)/HOAc Catalytic System 2019-12-05 |
|
1 |
|
Copper-Catalyzed Cascade Cyclization Reaction of Enamines and Electron-Deficient Terminal Alkynes: Synthesis of Polysubstituted Pyrido[1,2-a]indoles 2019-12-04 |
|
1 |
|
Copper-Mediated Direct Cyanation of Heteroarene and Arene C–H Bonds by the Combination of Ammonium and DMF 2019-12-04 |
|
1 |
|
Coupling of Trifluoroacetaldehyde N-Triftosylhydrazone with Organoboronic Acids for the Synthesis of gem-Difluoroalkenes 2019-12-04 |
|
1 |
|
Ruthenium-Catalyzed ortho- and meta-H/D Exchange of Arenes 2019-12-04 |
|
1 |
|
Access to 2-Aroylthienothiazoles via C–H/N–O Bond Functionalization of Oximes 2019-12-03 |
|
1 |
|
Access to Functionalized E-Allylsilanes and E-Alkenylsilanes through Visible-Light-Driven Radical Hydrosilylation of Mono- and Disubstituted Allenes 2019-12-03 |
|
1 |
|
Blue Light Induced Difluoroalkylation of Alkynes and Alkenes 2019-12-03 |
|
1 |
|
Excitation Wavelength-Dependent Nearly Pure White Light-Emitting Crystals from a Single Gold(I)-Containing Complex 2019-12-03 |
|
1 |
|
Metal-Free Synthesis of 3-(Iso)quinolinyl 4-Chromenones and 3-(Iso)quinolinyl 4-Quinolones from (Iso)quinoline N-Oxides and Ynones 2019-12-03 |
|
1 |
|
Privilege-Structure-Oriented Three-Component Asymmetric Aminomethylation: Assembly of Chiral 3-Aminomethyl Indolones 2019-12-03 |
|
1 |
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Regioselectivity-Switchable Catalytic Annulations of Alkynyl α-Diketones and α-Cyanoketones 2019-12-03 |
|
1 |
|
A Strategy for the Synthesis of Sulfonamides on DNA 2019-12-02 |
|
0.92 |
|
Gold-Catalyzed Intramolecular Dearomatization Reactions of Indoles for the Synthesis of Spiroindolenines and Spiroindolines 2019-12-02 |
|
0.75 |
|
Regioselective Synthesis and Crystallographic Characterization of Nontethered cis-1 and cis-2 Bis(benzofuro)[60]fullerene Derivatives 2019-12-02 |
|
1 |
|
A Direct Approach to Decoration of Bioactive Compounds via C–H Amination Reaction 2019-11-27 |
|
1 |
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Cascade π-Extended Decarboxylative Annulation Involving Cyclic Diaryliodonium Salts: Site-Selective Synthesis of Phenanthridines and Benzocarbazoles via a Traceless Directing Group Strategy 2019-11-27 |
|
1 |
|
Photocatalytic Annulation–Alkynyl Migration Strategy for Multiple Functionalization of Dual Unactivated Alkenes 2019-11-26 |
|
1 |
|
Rhodium-Catalyzed Pyridine N-Oxide Assisted Suzuki–Miyaura Coupling Reaction via C(O)–C Bond Activation 2019-11-26 |
|
1 |
|
Synthesis of 3-HCF2S-Chromones through Tandem Oxa-Michael Addition and Oxidative Difluoromethylthiolation 2019-11-26 |
|
1 |
|
(−)- and (+)-Asperginulin A, a Pair of Indole Diketopiperazine Alkaloid Dimers with a 6/5/4/5/6 Pentacyclic Skeleton from the Mangrove Endophytic Fungus Aspergillus sp. SK-28 2019-11-25 |
|
1 |
|
Asymmetric Formal Vinylogous Iminium Ion Activation for Vinyl-Substituted Heteroaryl and Aryl Aldehydes 2019-11-25 |
|
0.83 |
|
One-Carbon Incorporation Using Cyclobutanone Oxime Ester Enabled [2 + 2 + 1] Carboannulation of 1,7-Enynes by C–C/N–O Bond Cleavage and C–H Functionalization 2019-11-25 |
|
1 |
|
Pd-Catalyzed Enantioselective Double Heck Reaction 2019-11-25 |
|
1 |
|
Rhodium-Catalyzed Successive C–H Bond Functionalizations To Synthesize Complex Indenols Bearing a Benzofuran Unit 2019-11-25 |
|
1 |
|
Transformation of Alkynes into α- or β-Difluorinated Alkyl Azides by an Efficient One-Pot Two-Step Procedure 2019-11-25 |
|
1 |
|
Asymmetric Allylic Etherification of Vinylethylene Carbonates with Diols via Pd/B Cooperative Catalysis: A Route to Chiral Hemi-Crown Ethers 2019-11-22 |
|
1 |
|
Cleistocaltones A and B, Antiviral Phloroglucinol–Terpenoid Adducts from Cleistocalyx operculatus 2019-11-22 |
|
1 |
|
Copper-Mediated Deacylative Coupling of Ynones via C–C Bond Activation under Mild Conditions 2019-11-22 |
|
1 |
|
Redox-Neutral Borylation of Aryl Sulfonium Salts via C–S Activation Enabled by Light 2019-11-22 |
|
1 |
|
Agelanemoechine, a Dimeric Bromopyrrole Alkaloid with a Pro-Angiogenic Effect from the South China Sea Sponge Agelas nemoechinata 2019-11-20 |
|
0.90 |
|
An Approach to Peri-Fused Heterocycles: A Metal-Mediated Cascade Carbonylative Cyclization/Dearomatic Diels–Alder Reaction 2019-11-20 |
|
1 |
|
Asymmetric Total Synthesis Enables Discovery of Antibacterial Activity of Siladenoserinols A and H 2019-11-20 |
|
1 |
|
Chiral Spiro Phosphoramide-Catalyzed Sulfa-Michael Addition/Enantioselective Protonation of Exocyclic Enones 2019-11-20 |
|
1 |
|
Direct Catalytic Asymmetric Synthesis of Oxindole-Derived δ-Hydroxy-β-ketoesters by Aldol Reactions 2019-11-20 |
|
0.78 |
|
Divergent Reactivity in CuII-Catalyzed Oxidative Coupling between Indole/Tryptamine Derivatives and β-Arylacrylic Acids 2019-11-20 |
|
1 |
|
Electrochemical Synthesis of trans-2,3-Disubstituted Aziridines via Oxidative Dehydrogenative Intramolecular C(sp3)–H Amination 2019-11-20 |
|
1 |
|
Enantioselective Radical Ring-Opening Cyanation of Oxime Esters by Dual Photoredox and Copper Catalysis 2019-11-20 |
|
1 |
|
Gold(I)-Catalyzed Glycosylation with Glycosyl Ynenoates as Donors 2019-11-20 |
|
1 |
|
Morusalones A–D, Diels–Alder Adducts with 6/7/6/6/6/6 Hexacyclic Ring Systems as Potential PTP1B Inhibitors from Cell Cultures of Morus alba 2019-11-20 |
|
1 |
|
One-Pot Enantioselective Synthesis of 2-Pyrrolidinone Derivatives Bearing a Trifluoromethylated All-Carbon Quaternary Stereocenter 2019-11-20 |
|
1 |
|
Oxalic Acid Monothioester for Palladium-Catalyzed Decarboxylative Thiocarbonylation and Hydrothiocarbonylation 2019-11-20 |
|
0.83 |
|
Synthesis of Heterocyclic Core-Expanded Bis-Naphthalene Tetracarboxylic Diimides 2019-11-20 |
|
1 |
|
Carbene-Catalyzed Enantioselective Addition of Thioamides to Bromoenals for Access to Thiazinone Heterocycles 2019-11-19 |
|
0.83 |
|
Lewis-Acid-Mediated Thiocyano Semipinacol Rearrangement of Allylic Alcohols for Construction of α-Quaternary Center β-Thiocyano Carbonyls 2019-11-19 |
|
1 |
|
Ligand-Controlled Regiodivergent Silylation of Allylic Alcohols by Ni/Cu Catalysis for the Synthesis of Functionalized Allylsilanes 2019-11-19 |
|
1 |
|
Visible Light-Induced Amide Bond Formation 2019-11-19 |
|
1 |
|
Divergent Synthesis of Isoquinolone and Isocoumarin Derivatives by the Annulation of Benzoic Acid with N-Vinyl Amide 2019-11-18 |
|
1 |
|
Oxidative Hydro-, Bromo-, and Chloroheptafluoroisopropylation of Unactivated Alkenes with Heptafluoroisopropyl Silver 2019-11-18 |
|
1 |
|
Site-Selective Modification of α-Amino Acids and Oligopeptides via Native Amine-Directed γ-C(sp3)-H Arylation 2019-11-18 |
|
1 |
|
Asymmetric Conjugate Addition of Ethylene Sulfonyl Fluorides to 3-Amido-2-oxindoles: Synthesis of Chiral Spirocyclic Oxindole Sultams 2019-11-14 |
|
1 |
|
Construction of Multiple-Substituted Chiral Cyclohexanes through Hydrogenative Desymmetrization of 2,2,5-Trisubstituted 1,3-Cyclohexanediones 2019-11-14 |
|
1 |
|
LiHMDS-Promoted Palladium-Catalyzed Sonogashira Cross-Coupling of Aryl Fluorides with Terminal Alkynes 2019-11-14 |
|
1 |
|
N-Methoxyamide: An Alternative Amidation Reagent in the Rhodium(III)-Catalyzed C–H Activation 2019-11-14 |
|
1 |
|
Nickel-Catalyzed Transformation of Diazoacetates to Alkyl Radicals Using Alcohol as a Hydrogen Source 2019-11-14 |
|
1 |
|
Palladium-Catalyzed Controllable Reductive/Oxidative Heck Coupling between Cyclic Enones and Thiophenes via C–H Activation 2019-11-14 |
|
1 |
|
Synthesis of Oxadiazolones with Hydrazides: The Mechanism and the Sensing Application as Sensitive, Rapid, and Visual Fluorescent Sensors for Phosgene 2019-11-13 |
|
1 |
|
Access to Stereodefined (E)-2-Silylallylboronates via Regioselective Chloroboration of Allenylsilanes 2019-11-12 |
|
1 |
|
Ni-Catalyzed Intermolecular Allylic Dearomatization Reaction of Tryptophols and Tryptamines 2019-11-12 |
|
1 |
|
Spiroalanfurantones A–D, Four Eudesmanolide–Furan Sesquiterpene Adducts with a Pentacyclic 6/6/5/5/5 Skeleton from Inula helenium 2019-11-12 |
|
1 |
|
Synthesis of Isoxazolines and Oxazines by Electrochemical Intermolecular [2 + 1 + n] Annulation: Diazo Compounds Act as Radical Acceptors 2019-11-12 |
|
1 |
|
Copper-Catalyzed Cascade Cyclization of Arylsulfonylhydrazones Derived from ortho-Alkynyl Arylketones: Regioselective Synthesis of Functionalized Cinnolines 2019-11-11 |
|
1 |
|
Copper-Catalyzed Tandem Cross-Coupling/[2 + 2] Cycloaddition of 1,6-Allenynes with Diazo Compounds to 3-Azabicyclo[5.2.0] Ring Systems 2019-11-11 |
|
1 |
|
Cucurbit[8]uril-Mediated Polypseudorotaxane for Enhanced Lanthanide Luminescence Behavior in Water 2019-11-11 |
|
1 |
|
Direct Access to Allenylphosphine Oxides via a Metal Free Coupling of Propargylic Substrates with P(O)H Compounds 2019-11-11 |
|
1 |
|
Triarylborane-based [5]Helicenes with Full-Color Circularly Polarized Luminescence 2019-11-11 |
|
1 |
|
Pd(0)-Catalyzed Cyclizative Carboboration of n-Iodo-1,6-diene (n = 1 or 2): Access to Structurally Complex Allylboronates and Alkylboronates 2019-11-08 |
|
1 |
|
Pd-Catalyzed Asymmetric Allylic Cycloaddition of N-Containing Allylic Carbonates with Isocyanates 2019-11-08 |
|
1 |
|
Enantioselective Synthesis of Isoxazoline N-Oxides via Pd-Catalyzed Asymmetric Allylic Cycloaddition of Nitro-Containing Allylic Carbonates 2019-11-07 |
|
1 |
|
N-Alkylation-Initiated Redox-Neutral [5 + 2] Annulation of 3-Alkylindoles with o-Aminobenzaldehydes: Access to Indole-1,2-Fused 1,4-Benzodiazepines 2019-11-07 |
|
1 |
|
Total Synthesis of (+)-Jatrophalactam 2019-11-07 |
|
1 |
|
Gold-Catalyzed Highly Diastereoselective Oxy-Propargylamination of Allenamides with C-Alkynyl N-Boc N,O-Acetals 2019-11-06 |
|
1 |
|
Construction of Eight-Membered Cyclic Diaryl Sulfides via Domino Reaction of Arynes with Thioaurone Analogues and DFT Study on the Reaction Mechanism 2019-11-05 |
|
1 |
|
Hydrosulfonylation of Unactivated Alkenes by Visible Light Photoredox Catalysis 2019-11-05 |
|
1 |
|
Iridium-Catalyzed B–H Bond Insertion Reactions Using Sulfoxonium Ylides as Carbene Precursors toward α-Boryl Carbonyls 2019-11-05 |
|
1 |
|
Nickel-Catalyzed Reductive 1,2-Dialkynylation of Alkenes Bearing an 8-Aminoquinoline Directing Group 2019-11-05 |
|
1 |
|
Old Key Opens the Lock in Carborane: The in Situ NHC-Palladium Catalytic System for Selective Arylation of B(3,6)–H Bonds of o-Carboranes via B–H Activation 2019-11-05 |
|
1 |
|
Rhodium(III)-Catalyzed Annulative Coupling of Sulfoxonium Ylides and Allenoates: An Arene C–H Activation/Cyclopropanation Cascade 2019-11-05 |
|
1 |
|
Silver-Assisted Oxidative Isocyanide Insertion of Ethers: A Direct Approach to β-Carbonyl α-Iminonitriles 2019-11-05 |
|
1 |
|
Syntheses of Benzofuranoquinolines and Analogues via Photoinduced Acceptorless Dehydrogenative Annulation of o-Phenylfuranylpyridines 2019-11-05 |
|
1 |
|
Decarbonylative Phosphorylation of Carboxylic Acids via Redox-Neutral Palladium Catalysis 2019-11-04 |
|
0.40 |
|
Photoredox-Catalyzed Remote Difunctionalizations of Alkenes To Synthesize Fluoroalkyl Ketones with Dimethyl Sulfoxide as the Oxidant 2019-11-04 |
|
1 |
|
Pd(OAc)2-Catalyzed Asymmetric Hydrogenation of α-Iminoesters 2019-11-01 |
|
1 |
|
Switchable Synthesis of Aryl Sulfones and Sulfoxides through Solvent-Promoted Oxidation of Sulfides with O2/Air 2019-11-01 |
|
1 |
|
The Efficient Synthesis of Benzannulated Seven-Membered O-Heterocycles via the Intramolecular Ring-Opening Cyclization of Cyclopropanes 2019-11-01 |
|
1 |
|
Transition-Metal-Catalyzed Transformation of Sulfonates via S–O Bond Cleavage: Synthesis of Alkyl Aryl Ether and Diaryl Ether 2019-11-01 |
|
1 |
