Outputs for China

1 November 2019 - 31 October 2020

Subject/journal group: All

Count Share
19252 14369.63

The research outputs below are grouped by journal. Click on the journal to view the list of articles.

Journal Count Share
ACS Nano 605 451.22
Advanced Functional Materials 896 731.44
Advanced Materials 680 515.23
American Journal of Human Genetics 17 8.49
Analytical Chemistry 845 784.73
Angewandte Chemie International Edition 1407 1146.95
Applied Physics Letters 705 602.24
Cancer Cell 17 9.36
Cancer Research 74 41.55
Cell 72 38.12
Cell Host & Microbe 20 15.58
Cell Metabolism 20 9.55
Cell Stem Cell 24 10.98
Chemical Communications 1612 1502.99
Chemical Science 415 334.78
Current Biology 51 22.10
Developmental Cell 26 13.87
Earth and Planetary Science Letters 119 66.65
Ecology Letters 9 4.47
Environmental Science and Technology 665 519.17
European Physical Journal C 299 205.49
Genes & Development 5 1.07
Genome Research 25 14.75
Geochimica et Cosmochimica Acta 127 79.09
Geology 46 24.49
Geophysical Research Letters 427 279.33
Immunity 23 12.57
Inorganic Chemistry 588 526.54
Journal of Biological Chemistry 189 144.19
Journal of Cell Biology 13 9.29
Journal of Clinical Investigation 83 32.70
Journal of Experimental Medicine 28 17.04
Journal of Geophysical Research: Atmospheres 272 205.63
Journal of Geophysical Research: Solid Earth 213 147.68
Journal of High Energy Physics 302 137.15
Journal of Neuroscience 49 28.97
Journal of the American Chemical Society 781 552.80
Macromolecules 268 226.12
Molecular Cell 42 25.47
Molecular Psychiatry 47 24.20
Monthly Notices of the Royal Astronomical Society: Letters 23 14.10
Nano Letters 431 309.76
Nature 197 83.14
Nature Biotechnology 20 9.32
Nature Cell Biology 30 17.12
Nature Chemical Biology 22 12.13
Nature Chemistry 16 8.01
Nature Climate Change 22 10.68
Nature Communications 1552 979.33
Nature Genetics 32 12.08
Nature Geoscience 17 5.04
Nature Immunology 14 5.93
Nature Materials 48 18.18
Nature Medicine 23 11.48
Nature Methods 14 5.79
Nature Nanotechnology 36 19.10
Nature Neuroscience 13 7.56
Nature Photonics 24 10.34
Nature Physics 32 15.35
Nature Structural & Molecular Biology 17 9.03
Neuron 34 17.63
Organic Letters 876 828.90
Asymmetric Synthesis of Quinoline-Naphthalene Atropisomers by Central-to-Axial Chirality Conversion
2020-10-30
1
Palladium-Catalyzed Chemoselective Aminomethylative Cyclization and Aromatizing Allylic Amination: Access to Functionalized Naphthalenes
2020-10-30
1
Chiral Electron-Rich PNP Ligand with a Phospholane Motif: Structural Features and Application in Asymmetric Hydrogenation
2020-10-29
0.95
Nickel-Catalyzed Three-Component Reductive Alkylacylation of Electron-Deficient Activated Alkenes
2020-10-29
1
Total Synthesis and Immunological Evaluation of the Tri-d-glycero-d-manno-heptose Antigen of the Lipopolysaccharide as a Vaccine Candidate against Helicobacter pylori
2020-10-29
1
A CTV Analogue: Arene-Persubstituted Cyclotrixylohydroquinoylene and Its Derivatives
2020-10-28
1
Aaptodines A–D, Spiro Naphthyridine–Furooxazoloquinoline Hybrid Alkaloids from the Sponge Aaptos suberitoides
2020-10-28
0.71
Visible-Light-Promoted Regioselective 1,3-Fluoroallylation of gem-Difluorocyclopropanes
2020-10-28
1
Chemoselective Perfluoromethylation of Thio- and Selenoamides
2020-10-27
1
Cu(II)/Iodine(III) Oxide Dimerization of Heterocyclic Ketene Aminals: Tandem TEMPO Oxidation for the Highly Selective Synthesis of Functionalized 2H-Pyrrolo[1,2-a]imidazol-7(3H)-ones
2020-10-27
1
Dual Nickel- and Photoredox-Catalyzed Reductive Cross-Coupling of Aryl Halides with Dichloromethane via a Radical Process
2020-10-27
1
Modular Synthesis of Drimane Meroterpenoids Leveraging Decarboxylative Borylation and Suzuki Coupling
2020-10-27
1
Asymmetric Total Synthesis and Assignment of Absolute Configuration of Arbornamine
2020-10-26
1
Deciphering the Biosynthetic Mechanism of Pelletierine in Lycopodium Alkaloid Biosynthesis
2020-10-26
0.77
Synthesis and Biological Evaluation of N-Aminoimidazolidin-2-one-Containing Angiotensin-(1–7) Peptidomimetics
2020-10-26
1
Generation of Carbocations under Photoredox Catalysis: Electrophilic Aromatic Substitution with 1-Fluoroalkylbenzyl Bromides
2020-10-23
0.83
Nickel-Catalyzed Highly Selective Hydroalkenylation of Alkenyl Boronic Esters to Access Allyl Boron
2020-10-22
1
Triphenylphosphine-Catalyzed Alkylative Iododecarboxylation with Lithium Iodide under Visible Light
2020-10-22
0.83
Biomimetic Total Synthesis of (±)-Carbocyclinone-534 Reveals Its Biosynthetic Pathway
2020-10-21
1
Cyanide-Free Synthesis of Glycosyl Carboxylic Acids and Application for the Synthesis of Scleropentaside A
2020-10-21
1
Enantioselective Synthesis of 4-Cyanotetrahydroquinolines via Ni-Catalyzed Hydrocyanation of 1,2-Dihydroquinolines
2020-10-21
1
Palladium-Catalyzed Hydroxylation of Aryl Halides with Boric Acid
2020-10-21
1
Diastereodivergent Synthesis of α-Chiral Tertiary Azides through Catalytic Asymmetric Michael Addition
2020-10-20
1
A Bispidine-Based Chiral Amine Catalyst for Asymmetric Mannich Reaction of Ketones with Isatin Ketimines
2020-10-19
1
Cu-Catalyzed Regioselective C–H Alkylation of Benzimidazoles with Aromatic Alkenes
2020-10-19
1
Peptide Modification via N-Terminal-Residue-Directed γ-C(sp3)–H Arylation
2020-10-19
1
Relay Palladium/Copper Catalysis Enabled Silylative [5 + 1] Benzannulation Using Terminal Alkynes as One-Carbon Units
2020-10-19
1
Synthetic Investigation toward QS-21 Analogues
2020-10-19
1
Switching of C–C and C–N Coupling/Cleavage for Hypersensitive Detection of Cu2+ by a Catalytically Mediated 2-Aminoimidazolyl-Tailored Six-Membered Rhodamine Probe
2020-10-16
1
Dichloroacetophenone Derivatives: A Class of Bioconjugation Reagents for Disulfide Bridging
2020-10-14
0.75
Nickel(II)-Catalyzed Oxygen Transfer Reaction of N-Vinyl Nitrones to Prepare 2-(Pyridin-2-yl)ethanols
2020-10-14
1
Pd-Catalyzed Domino Imidoylation/Heck/C(sp2)–H Cyclization: Isocyanide Relay Strategy toward Tricyclic-Fused Heterocycles Containing an All-Carbon Quaternary Center
2020-10-14
1
Rh-Catalyzed Annulation of Benzoic Acids, Formaldehyde, and Malonates via ortho-Hydroarylation to Indanones
2020-10-14
1
A Series of Deoxyfluorination Reagents Featuring OCF2 Functional Groups
2020-10-13
1
Construction of β-Quaternary α,α-Difluoroketones via Catalytic Nucleophilic Substitution of Tertiary Alcohols with Difluoroenoxysilanes
2020-10-13
1
Iodine-Promoted Multicomponent Synthesis of 2,4-Diamino-1,3,5-triazines
2020-10-13
1
Light-Mediated Difluoromethylthiolation of Aldehydes with a Hydrogen Atom Transfer Photocatalyst
2020-10-13
1
NHC/Copper-Cocatalyzed [4 + 3] Annulations of Salicylaldehydes with Aziridines for the Synthesis of 1,4-Benzoxazepinones
2020-10-13
1
Synthesis of C4-Substituted Indoles via a Catellani and C–N Bond Activation Strategy
2020-10-13
1
Visible-Light-Mediated Hydroacylation of Azobenzenes with α-Keto Acids
2020-10-13
1
A Construction of α-Alkenyl Lactones via Reduction Radical Cascade Reaction of Allyl Alcohols and Acetylenic Acids
2020-10-12
1
Asymmetric Transfer Hydrogenation of Densely Functionalized Diheteroaryl and Diaryl Ketones by a Ru-Catalyst of Minimal Stereogenicity
2020-10-12
1
Chemical Synthesis of Homogeneous Human E-Cadherin N-Linked Glycopeptides: Stereoselective Convergent Glycosylation and Chemoselective Solid-Phase Aspartylation
2020-10-12
0.21
Direct Electrochemical Defluorinative Carboxylation of gem-Difluoroalkenes with Carbon Dioxide
2020-10-12
1
Highly Enantioselective Synthesis of Monofluoroalkenes by Rhodium-Catalyzed Asymmetric Arylation/Defluorination of Allyl Difluorides
2020-10-12
0.80
Nickel-Catalyzed Asymmetric Transfer Hydrogenation and α-Selective Deuteration of N-Sulfonyl Imines with Alcohols: Access to α-Deuterated Chiral Amines
2020-10-12
1
P(NMe2)3-Mediated Umpolung Spirocyclopropanation Reaction of p-Quinone Methides: Diastereoselective Synthesis of Spirocyclopropane-Cyclohexadienones
2020-10-12
1
Radical Tandem Bicyclization Triggered by the α-Position of α,β-Unsaturated Ketones Bearing Nonterminal 1,6-Enynes: Synthesis of the 5H-Benzo[a]fluoren-5-one Skeleton
2020-10-12
1
Reductive CO2 Fixation via the Selective Formation of C–C Bonds: Bridging Enaminones and Synthesis of 1,4-Dihydropyridines
2020-10-12
1
Unconventional Transformation of the Two Carbonyl Groups in 4,4′,5,5′-Tetrachloro-10H,10′H-[9,9′-bianthracenylidene]-10,10′-dione into Diallenes
2020-10-12
1
Vinylogous Elimination/C–H Functionalization/Allylation Cascade Reaction of Allenoate Adducts: Synthesis of Ring-Fused Dihydropyridinones
2020-10-12
1
General Synthesis of α-Alkyl Ynones from Morpholine Amides and 1-Copper(I) Alkynes Promoted by Triflic Anhydride
2020-10-09
1
In(OTf)3-Catalyzed Synthesis of 2,3-Dihydro-1H-benzo[e]indoles and 2,3-Dihydrobenzofurans via [3 + 2] Annulation
2020-10-09
1
Combined KOH/BEt3 Catalyst for Selective Deaminative Hydroboration of Aromatic Carboxamides for Construction of Luminophores
2020-10-07
1
Copper-Catalyzed Oxidative Fragmentation of Alkynes with NFSI Provides Aryl Ketones
2020-10-07
1
Stereodivergent Synthesis of Alkenylpyridines via Pd/Cu Catalyzed C–H Alkenylation of Pyridinium Salts with Alkynes
2020-10-07
1
Transition-Metal Free Chemoselective Hydroxylation and Hydroxylation–Deuteration of Heterobenzylic Methylenes
2020-10-07
1
6,12-Dihydro-6,12-diboradibenzo[def,mno]chrysene: A Doubly Boron-Doped Polycyclic Aromatic Hydrocarbon for Organic Light Emitting Diodes by a One-Pot Synthesis
2020-10-06
1
Aminothiolation of α-Bromocinnamaldehydes to Access Imidazo[2,1-b]thiazoles by Incorporation of Two Distinct Photoinduced Processes
2020-10-06
1
Copper-Catalyzed Aerobic Cyclization of β,γ-Unsaturated Hydrazones with Concomitant C═C Bond Cleavage
2020-10-06
1
Scocycamides, a Pair of Macrocyclic Dicaffeoylspermidines with Butyrylcholinesterase Inhibition and Antioxidation Activity from the Roots of Scopolia tangutica
2020-10-06
1
Synthesis of Heterobiaryl 4-Aryl Furans through a Base-Promoted Decarboxylative Propargylation/Cycloisomerization Annulation
2020-10-06
1
γ-Difluoroalkylation: Synthesis of γ-Difluoroalkyl-α,β-Unsaturated Esters via Photoredox NHC-Catalyzed Radical Reaction
2020-10-06
1
The Biomimetic Total Syntheses of the Antiplasmodial Tomentosones A and B
2020-10-05
1
Annulation of Diaryl(aryl)phosphenes and Cyclic Imines to Access Benzo-δ-phospholactams
2020-10-02
1
Nickel-Catalyzed Cyanation of Unactivated Alkyl Sulfonates with Zn(CN)2
2020-10-02
1
Ustethylin Biosynthesis Implies Phenethyl Derivative Formation in Aspergillus ustus
2020-10-02
0.33
Access to Dibenzofurans through Dimerization/Trimerization of Cyclohexanones Followed by Dehydroaromatization
2020-10-01
1
Bisaspochalasins A–C: Three Cytochalasan Homodimers with Highly Fused Ring System from an Endophytic Aspergillus flavipes
2020-10-01
1
Longisglucinols A–C, Structurally Intriguing Polycyclic Polyprenylated Acylphloroglucinols with Anti-inflammatory Activity from Hypericum longistylum
2020-10-01
1
Photochemical Decarboxylative C(sp3)–X Coupling Facilitated by Weak Interaction of N-Heterocyclic Carbene
2020-10-01
1
Polysulfuration via a Bilateral Thiamine Disulfurating Reagent
2020-10-01
1
Cleavage of Aromatic C–O Bonds via Intramolecular SNAr Reaction and Preparation of P,C,Axial-Stereogenic Menthyl Phosphine Derivatives
2020-09-30
1
Copper-Catalyzed Selective 1,2-Difunctionalization of N-Heteroaromatics through Cascade C–N/C═C/C═O Bond Formation
2020-09-30
1
Palladium-Catalyzed Addition/Cyclization of (2-Hydroxyaryl)boronic Acids with Alkynylphosphonates: Access to Phosphacoumarins
2020-09-30
1
Access to Cycloalkeno[c]-Fused Pyridines via Pd-Catalyzed C(sp2)–H Activation and Cyclization of N-Acetyl Hydrazones of Acylcycloalkenes with Vinyl Azides
2020-09-29
1
B(C6F5)3-Catalyzed β-Functionalization of Pyrrolidines Using Isatins via Borrowing Hydrogen: Divergent Access to Substituted Pyrrolidines and Pyrroles
2020-09-29
1
Carboxyl-Assisted meta-Selective C–H Functionalizations of Benzylsulfonamides
2020-09-29
1
Chiral Hydroxytetraphenylene–Boron Complex Catalyzed Asymmetric Diels–Alder Cycloaddition of 2′-Hydroxychalcones
2020-09-29
1
Cu-Catalyzed o-Amino Benzofuranthioether Formation from N-Tosylhydrazone-Bearing Thiocarbamates and Arylative Electrophiles
2020-09-29
1
Difluoroisoxazolacetophenone: A Difluoroalkylation Reagent for Organocatalytic Vinylogous Nitroaldol Reactions of 1,2-Diketones
2020-09-29
1
Euphopias A–C: Three Rearranged Jatrophane Diterpenoids with Tricyclo[8.3.0.02,7]tridecane and Tetracyclo[11.3.0.02,10.03,7]hexadecane Cores from Euphorbia helioscopia
2020-09-29
1
Organocatalytic Regio- and Enantioselective 1,8-Additions of Nitrogen and Sulfur Nucleophiles to 6-Methylene-6H-indoles
2020-09-29
1
Silver-Catalyzed para-Selective Amination and Aminative Dearomatization of Phenols with Azodicarboxylates in Water
2020-09-29
1
Synthesis of l-glycero- and d-glycero-d-manno-Heptose Building Blocks for Stereoselective Assembly of the Lipopolysaccharide Core Trisaccharide of Vibrio parahemolyticus O2
2020-09-29
1
Unconventional [2 + 3] Cyclization Involving [1,4]-Sulfonyl Transfer to Construct Polysubstituted Fluorazones as Inhibitors of Indoleamine 2,3-Dioxygenase 1
2020-09-29
1
Synthesis of Substituted Naphtho[1,8-bc]thiopyrans by Sulfhydryl-Directed Rhodium-Catalyzed peri-Selective C–H Bond Activation and Cyclization of Naphthalene-1-thiols
2020-09-28
1
Chiral Calcium Phosphate Catalyzed Enantioselective Amination of 3-Aryl-2-benzofuranones
2020-09-24
1
Metal-Free Radical-Mediated C(sp3)–H Heteroarylation of Alkanes
2020-09-24
1
Strategic Construction of Ethene-Bridged BODIPY Arrays with Absorption Bands Reaching the Near-Infrared II Region
2020-09-24
1
Thianthrenation-Enabled α-Arylation of Carbonyl Compounds with Arenes
2020-09-24
1
Catalytic Asymmetric Synthesis of Atropisomeric Nitrones: Versatile Intermediate for Axially Chiral Biaryls
2020-09-23
1
Catalytic Direct Construction of Cyano-tetrazoles
2020-09-23
1
Chalcogenide-Catalyzed Intermolecular Electrophilic Thio- and Halofunctionalization of gem-Difluoroalkenes: Construction of Diverse Difluoroalkyl Sulfides and Halides
2020-09-23
1
Copper-Catalyzed Anti-Markovnikov Hydrosilylation of Terminal Alkynes
2020-09-23
1
NHC-Catalyzed Enantioselective [3 + 3] Annulation to Construct 5,6-Dihydropyrimidin-4-ones
2020-09-23
1
Organocatalytic Enantioselective Conjugate Alkynylation of β-Aminoenones: Access to Chiral β-Alkynyl-β-Amino Carbonyl Derivatives
2020-09-23
1
Rh(III)-Catalyzed [3 + 2] Spirocyclization of 2H-Imidazoles with 1,3-Diynes for the Synthesis of Spiro-[imidazole-indene] Derivatives
2020-09-23
1
Synergistic N-Heterocyclic Carbene/Palladium-Catalyzed [3 + 2] Annulation of Vinyl Enolates with 1-Tosyl-2-vinylaziridine
2020-09-23
1
Vinyl Sulfonium Salts as the Radical Acceptor for Metal-Free Decarboxylative Alkenylation
2020-09-23
1
Divergent Synthesis of Trifluoromethyl Sulfoxides and β-SCF3 Carbonyl Compounds by Tandem Trifluoromethylthiolation/Rearrangement of Allylic and Propargylic Alcohols
2020-09-22
1
Oligo(5-amino-N-acylanthranilic acids): Amide Bond Formation without Coupling Reagent and Folding upon Binding Anions
2020-09-22
0.25
Cage-Monoterpenoid Quinoline Alkaloids with Neurite Growth Promoting Effects from the Fruits of Melodinus yunnanensis
2020-09-21
0.83
A Photochemical Dehydrogenative Strategy for Direct and Regioselective Dimerization of BODIPY Dyes
2020-09-18
1
Decarboxylative and Deaminative Alkylation of Difluoroenoxysilanes via Photoredox Catalysis: A General Method for Site-Selective Synthesis of Difluoroalkylated Alkanes
2020-09-18
1
Pd-Catalyzed C(sp3)–H Biarylation via Transient Directing Group Strategy
2020-09-18
1
Ruthenium-Catalyzed Enantioselective Hydrogenation of Hydrazones
2020-09-18
0.20
Synthesis of Enantioenriched α,α-Difluoro-β-arylbutanoic Esters by Pd-Catalyzed Asymmetric Hydrogenation
2020-09-18
1
Tandem [5 + 2]/[4 + 2] Cycloadditions To Construct the [6–7–6] Tricyclic Skeleton of Icetexane Diterpenes: Total Synthesis of Euolutchuol E, Przewalskine E and Brussonol
2020-09-18
1
Asymmetric Dearomative Cascade Multiple Functionalizations of Activated N-Alkylpyridinium and N-Alkylquinolinium Salts
2020-09-17
1
Cross-Dehydrogenative Coupling of Strong C(sp3)–H with N-Heteroarenes through Visible-Light-Induced Energy Transfer
2020-09-17
1
Photoredox-Catalyzed α-C(sp3)–H Activation of Unprotected Secondary Amines: Facile Access to 1,4-Dicarbonyl Compounds
2020-09-17
1
Enantioselective Total Syntheses of Pentacyclic Homoproaporphine Alkaloids
2020-09-16
1
Palladium-Catalyzed Oxidative Annulation of Sulfoximines and Arynes by C–H Functionalization as an Approach to Dibenzothiazines
2020-09-16
1
Pegaharmols A–B, Axially Chiral β-Carboline-quinazoline Dimers from the Roots of Peganum harmala
2020-09-16
0.89
Visible-Light-Mediated Trifluoromethylation/Benzylation of Styrenes Catalyzed by 4-CzIPN
2020-09-16
1
Silver-Catalyzed Cascade Cyclization Reaction of Isocyanides with Sulfoxonium Ylides: Synthesis of 3-Aminofurans and 4-Aminoquinolines
2020-09-15
1
Mono/Dual Amination of Phenols with Amines in Water
2020-09-11
1
Synthesis of Polysubstituted Pyrroles via Silver-Catalyzed Oxidative Radical Addition of Cyclopropanols to Imines
2020-09-11
1
CuI/2-Aminopyridine 1-Oxide Catalyzed Amination of Aryl Chlorides with Aliphatic Amines
2020-09-10
1
Divergent Synthesis of Bicyclo[3.2.1]octenes and Cyclohexenes via Catalytic Annulations of Nazarov Reagent and Vinyl 1,2-Diketones
2020-09-10
1
Nickel-Catalyzed Mizoroki–Heck/Amination Cascade Reactions of o-Dihaloarenes with Allylamines: Synthesis of Indoles
2020-09-10
1
Asymmetric Construction of Cyclobutanes via Direct Vinylogous Michael Addition/Cyclization of β,γ-Unsaturated Amides
2020-09-09
1
Copper(I)/DDQ-Mediated Double-Dehydrogenative Diels–Alder Reaction of Aryl Butenes with 1,4-Diketones and Indolones
2020-09-09
1
Iodonium Ylides as Carbene Precursors in Rh(III)-Catalyzed C–H Activation
2020-09-09
1
Silver-Catalyzed Activation of Pyridotriazoles for Formal Intramolecular Carbene Insertion into Vinylic C(sp2)–H Bonds
2020-09-09
1
Synthesis and Catalytic Properties of Metal–N-Heterocyclic-Carbene-Decorated Covalent Organic Framework
2020-09-09
1
Tuning the Properties of Corannulene-Based Polycyclic Aromatic Hydrocarbons by Varying the Fusing Positions of Corannulene
2020-09-09
1
Visible Light-Driven α-Alkylation of N-Aryl tetrahydroisoquinolines Initiated by Electron Donor–Acceptor Complexes
2020-09-09
1
Visible-Light-Promoted Site-Selective N1-Alkylation of Benzotriazoles with α-Diazoacetates
2020-09-09
0.86
Asymmetric Synthesis of γ-Secondary Amino Alcohols via a Borrowing-Hydrogen Cascade
2020-09-08
1
Chlorotrifluoromethylthiolation of Sulfur Ylides for the Formation of Tetrasubstituted Trifluoromethylthiolated Alkenes
2020-09-08
1
Controlling Keto–Enol Tautomerism of Ureidopyrimidinone to Generate a Single-Quadruple AADD-DDAA Dimeric Array
2020-09-08
1
Iron-Catalyzed Redox-Neutral Radical Cascade Reaction of [60]Fullerene with γ,δ-Unsaturated Oxime Esters: Preparation of Free (N–H) Pyrrolidino[2′,3′:1,2]fullerenes
2020-09-08
1
β-Carboline Alkaloids from the Seeds of Peganum harmala and Their Anti-HSV-2 Virus Activities
2020-09-08
1
Au(I)-Catalyzed Cyclization/Semipinacol Rearrangement Reaction of Allenes to Construct Quaternary Carbon-Containing Scaffolds
2020-09-04
1
Baicalensines A and B, Two Isoquinoline Alkaloids from the Roots of Thalictrum baicalense
2020-09-04
1
Visible-Light-Promoted Intramolecular α-Allylation of Aldehydes in the Absence of Sacrificial Hydrogen Acceptors
2020-09-04
1
Palladium-Catalyzed [5 + 2] Annulation of Vinylethylene Carbonates with Barbiturate-Derived Alkenes
2020-09-03
1
A Role for Isatin Azomethine Imines as a Dipolarophile in Cycloaddition Reactions
2020-09-02
1
A Strategy for Amide to β-Oxo Ester Transformation via N-Alkenoxypyridinium Salts as the Activator and H2O as the Nucleophile
2020-09-02
1
Splitting Methyl Ketones into Two Parts: Synthesis of 4(3H)-Quinazolinones via Consecutive Cyclization/Ring-Opening Reaction
2020-09-02
1
Synthesis of γ-Lactams via Pd(II)-Catalyzed C(sp3)–H Olefination Using a Self-Cleaving Polyfluoroethylsulfinyl Directing Group
2020-09-02
1
Solvation-Free Li+ Lewis Acid Enhancing Reaction: Kinetic Study of [5,6]-Li+@PCBM to [6,6]-Li+@PCBM
2020-09-01
0.33
Visible-Light-Promoted Photoredox Dehydrogenative Coupling of Phosphines and Thiophenols
2020-09-01
1
Zwitterion-Catalyzed Deacylative Dihalogenation of β-Oxo Amides
2020-09-01
1
Access to Cyanoimines Enabled by Dual Photoredox/Copper-Catalyzed Cyanation of O-Acyl Oximes
2020-08-31
1
Iridium-Catalyzed Asymmetric Hydrogenation of α-Fluoro Ketones via a Dynamic Kinetic Resolution Strategy
2020-08-31
1
Visible-Light-Triggered Iodinations Facilitated by Weak Electrostatic Interaction of N-Heterocyclic Carbenes
2020-08-31
1
Catalytic Enantioselective Dearomatization/Rearomatization of 2-Nitroindoles to Access 3-Indolyl-3′-Aryl-/Alkyloxindoles: Application in the Formal Synthesis of Cyclotryptamine Alkaloids
2020-08-28
1
Directing-Group-Assisted C(sp2)–H Arylsulfonylation from Sulfur Dioxide
2020-08-28
1
Palladium-Catalyzed Decarbonylative Heck Coupling of Aromatic Carboxylic Acids with Terminal Alkenes
2020-08-28
1
Rapid Access of Alkynyl and Alkenyl Coumarins via a Dipyridinium Methylide and Propargylamine Cascade Reaction
2020-08-28
1
Regioselective Direct C–H Trifluoromethylation of Pyridine
2020-08-28
1
Synthesis of Indenopyrazole Frameworks via Cascade C–H Functionalization/[3 + 2] Dipolar Cycloaddition/Aromatization Rearrangement Reactions
2020-08-28
1
Copper-Mediated Decarboxylative Sulfonylation of Arylacetic Acids with Sodium Sulfinates
2020-08-27
1
Electrochemical Alkoxyhalogenation of Alkenes with Organohalides as the Halide Sources via Dehalogenation
2020-08-27
1
1,1-Addition of α-C2-Bridged Biphospholes with Alkynes
2020-08-26
1
Arylaminomethyl Radical-Initiated Cascade Annulation Reaction of Quinoxalin-2(1H)-ones Catalyzed by Recyclable Photocatalyst Perovskite
2020-08-26
1
Chiral Naphthyl-C2-Indole as Scaffold for Phosphine Organocatalysis: Application in Asymmetric Formal [4 + 2] Cycloaddition Reactions
2020-08-26
1
Cu(I)-Catalyzed Oxidative Cyclization of Enynamides: Regioselective Access to Cyclopentadiene Frameworks and 2-Aminofurans
2020-08-26
1
Ni-Catalyzed Reductive Antiarylative Cyclization of Alkynones
2020-08-26
1
Lewis-Acid-Mediated Intramolecular Trifluoromethylthiolation of Alkenes with Phenols: Access to SCF3-Containing Chromane and Dihydrobenzofuran Compounds
2020-08-25
1
Terreuspyridine: An Unexpected Pyridine-Fused Meroterpenoid Alkaloid with a Tetracyclic 6/6/6/6 Skeleton from Aspergillus terreus
2020-08-25
1
Hemin-Catalyzed Oxidative Phenol-Hydrazone [3+3] Cycloaddition Enables Rapid Construction of 1,3,4-Oxadiazines
2020-08-24
1
Total Synthesis of Gastrodinol via Photocatalytic 6π Electrocyclization
2020-08-24
1
2-(Dimesitylboryl)phenyl-Substituted [2.2]Paracyclophanes Featuring Intense and Sign-Invertible Circularly Polarized Luminescence
2020-08-21
1
C–H Borylation of Diphenylamines through Adamantane-1-carbonyl Auxiliary by BBr3
2020-08-21
1
Elucidation of the Tailoring Steps in Julichrome Biosynthesis by Marine Gastropod Mollusk-Associated Streptomyces sampsonii SCSIO 054
2020-08-21
1
Hyperfols A and B: Two Highly Modified Polycyclic Polyprenylated Acylphloroglucinols from Hypericum perforatum
2020-08-21
1
Lewis-Acid-Catalyzed Asymmetric Alkynylation of Alkynyl 1,2-Diketones: Controllable Formation of 3(2H)-Furanones and α-Hydroxy Ketones
2020-08-21
1
Palladium-Catalyzed Tandem C–C Activation/Cyclization Induced by Carbopalladation of Functionalized Nitriles: Synthesis of Benzo Dipyrromethenes
2020-08-21
1
Radical-Dual-Difunctionalization and Trifluoromethylative Decarboxylation of Two Different Alkenes
2020-08-21
1
Remote C–H Activation Strategy Enables Total Syntheses of Nortriterpenoids (±)-Walsucochin B and (±)-Walsucochinoids M and N
2020-08-21
1
Asymmetric Catalytic Synthesis of Epoxides via Three-Component Reaction of Diazoacetates, 2-Oxo-3-ynoates, and Nitrosoarenes
2020-08-20
1
Difluorocarbene-Triggered Cyclization: Synthesis of (Hetero)arene-Fused 2,2-Difluoro-2,3-dihydrothiophenes
2020-08-20
1
Ligand-Controlled Palladium-Catalyzed Chemoselective Multicomponent Reaction of Olefin-Tethered Aryl Halides, Isocyanides, and Carboxylic Acids: Diversified Synthesis of Imides
2020-08-20
1
Phosphine-Catalyzed Stereoselective Tandem Annulation Reaction for the Synthesis of Chromeno[4,3-b]pyrroles
2020-08-20
1
Construction of Cyclophane-Braced Peptide Macrocycles via Palladium-Catalyzed Picolinamide-Directed Intramolecular C(sp2)–H Arylation
2020-08-19
1
Electrochemically Enabled Sulfonylation of Alkynes with Sodium Sulfinates
2020-08-19
1
Ni-Catalyzed Direct Carboxylation of an Unactivated C–H Bond with CO2
2020-08-19
1
Acyl Radicals from α-Keto Acids Using a Carbonyl Photocatalyst: Photoredox-Catalyzed Synthesis of Ketones
2020-08-18
0.83
Catalytic Asymmetric Three-Component Reaction of 2-Alkynylbenzaldehydes, Amines, and Dimethylphosphonate
2020-08-18
1
Chemo- and Diastereoselective Synthesis of Pyrrolidines from Aroylformates and δ-Tosylamino Enones via P(NMe2)3-Mediated Reductive Amination/Base-Catalyzed Michael Addition Cascade
2020-08-18
1
Enantioselective Dehydrative γ-Arylation of α-Indolyl Propargylic Alcohols with Phenols: Access to Chiral Tetrasubstituted Allenes and Naphthopyrans
2020-08-18
1
Palladium-Catalyzed Secondary Benzylic Imidoylative Reactions
2020-08-18
1
Photoinduced Copper-Catalyzed Site-Selective C(sp2)–C(sp) Cross-Coupling via Aryl Sulfonium Salts
2020-08-18
1
Ruthenium(II)-Catalyzed C–H Arylation of N,N-Dialkyl Thiobenzamides with Boronic Acids by Sulfur Coordination in 2-MeTHF
2020-08-18
0.92
Synthesis of Spiroisoxazolines via TEMPO/NaNO2-Catalyzed Aerobic Oxidative Dearomatization
2020-08-18
1
Catalytic Claisen Rearrangement by Intercepting Ketenimines with Propargylic Alcohols: A Strategy to Generate and Transform Ketenimines from Radicals
2020-08-14
1
Construction of CF3-Containing Tetrahydropyrano[3,2-b]indoles through DMAP-Catalyzed [4+1]/[3+3] Domino Sequential Annulation
2020-08-14
1
Multiturn Hollow Helices: Synthesis and Folding of Long Aromatic Oligoamides
2020-08-14
0.22
Selective Synthesis of 2-Indolyl-3-oxoindolines or 2-(2-Aminophenyl)quinolines through Cu(II)- or Bi(III)-Catalyzed Tunable Dimerizations of 2-Alkynylanilines
2020-08-14
1
Cu/Ag-Catalyzed Reaction of Azirines with Anthranils: Synthesis of (Quinazolin-2-yl)methanone Derivatives
2020-08-13
1
NHC-Catalyzed Asymmetric α-Regioselective [4 + 2] Annulation to Construct α-Alkylidene-δ-lactones
2020-08-13
1
Nickel-Catalyzed Reductive Aryl Thiocarbonylation of Alkene via Thioester Group Transfer Strategy
2020-08-13
1
Cobalt-Catalyzed Radical Hydrotrifluoroethylation of Styrenes with Trifluoroethyl Iodide
2020-08-12
1
Dehydroxylative Fluorination of Tertiary Alcohols
2020-08-12
0.75
Phthalaldehyde-Amine Capture Reactions for Bioconjugation and Immobilization of Phthalocyanines
2020-08-12
1
Rh(III)-Catalyzed [4 + 2] Annulation of 3-Aryl-5-isoxazolone with Maleimides or Maleic Ester
2020-08-12
1
Ruthenium(II)-Catalyzed Regioselective [3 + 2] Spiroannulation of 2H-Imidazoles with 2-Alkynoates
2020-08-12
1
Asymmetric Reductive Amination/Ring-Closing Cascade: Direct Synthesis of Enantioenriched Biaryl-Bridged NH Lactams
2020-08-11
1
Cu-Catalyzed Direct Amination of Cyclic Amides via C–OH Bond Activation Using DMF
2020-08-11
1
Isothiourea-Catalyzed Atroposelective N-Acylation of Sulfonamides
2020-08-11
0.21
Ynamide-Mediated Thionoester and Dithioester Syntheses
2020-08-11
1
Decarbonylative Suzuki–Miyaura Cross-Coupling of Aroyl Chlorides
2020-08-10
0.60
Engineered Biosynthesis of Fungal 4-Quinolone Natural Products
2020-08-10
0.11
Metal-Free Chemoselective Reaction of Sulfoxonium Ylides and Thiosulfonates: Diverse Synthesis of 1,4-Diketones, Aryl Sulfursulfoxonium Ylides, and β-Keto Thiosulfones Derivatives
2020-08-10
1
Site-Selective Silylation of Arenes Mediated by Thianthrene S-Oxide
2020-08-10
1
Synthesis of Bridged Bicyclic Amines by Intramolecular Amination of Remote C–H Bonds: Synergistic Activation by Light and Heat
2020-08-10
0.09
Cu-Catalyzed Site-Selective and Enantioselective Ring Opening of Cyclic Diaryliodoniums with 1,2,3-Triazoles
2020-08-07
1
Dual Nickel-/Palladium-Catalyzed Reductive Cross-Coupling Reactions between Two Phenol Derivatives
2020-08-07
0.80
Nickel-Catalyzed Thiocarbonylation of Arylboronic Acids with Sulfonyl Chlorides for the Synthesis of Thioesters
2020-08-07
0.88
Synthesis of Aza-Eight-Membered Ring-Fused Indolines Initiated by Zn-Catalyzed C2 Alkylation of Indoles and Subsequent Base-Promoted Ring Expansion
2020-08-06
1
Synthesis of O-Sulfated Human Syndecan-1-like Glyco-polypeptides by Incorporating Peptide Ligation and O-Sulfated Glycopeptide Cassette Strategies
2020-08-06
0.08
Bio- and Medicinally Compatible α-Amino-Acid Modification via Merging Photoredox and N-Heterocyclic Carbene Catalysis
2020-08-05
1
Organocatalytic Atroposelective Construction of Axially Chiral N-Aryl Benzimidazoles Involving Carbon–Carbon Bond Cleavage
2020-08-05
1
Pd/Cu-Catalyzed Domino Cyclization/Deborylation of Alkene-Tethered Carbamoyl Chloride and 1,1-Diborylmethane
2020-08-05
1
Asymmetric Transfer Hydrogenation of Unhindered and Non-Electron-Rich 1-Aryl Dihydroisoquinolines with High Enantioselectivity
2020-08-04
0.33
Novel Meroterpenoids from Hypericum patulum: Highly Potent Late Nav1.5 Sodium Current Inhibitors
2020-08-04
0.96
PIDA-Mediated Rearrangement for the Synthesis of Enantiopure Triazolopyridinones
2020-08-04
1
Penicimeroterpenoids A–C, Meroterpenoids with Rearrangement Skeletons from the Marine-Derived Fungus Penicillium sp. SCSIO 41512
2020-08-04
1
Rapid Access to Tetracyclic Core of Wortmannin via an Intramolecular Reductive Olefin Coupling Strategy
2020-08-04
1
Rationally Designed Self-Immolative Rotaxane Sensor Based on Pillar[5]arene for Fluoride Sensing
2020-08-04
1
Silver-Promoted Direct Phosphorylation of Bulky C(sp2)–H Bond to Build Fully Substituted β-Phosphonodehydroamino Acids
2020-08-04
1
Tris(4-bromophenyl)aminium Hexachloroantimonate-Initiated Oxidative Povarov-Type Reaction between Glycine Esters and (Cyclopropylidenemethyl)benzenes Using the Counterion as a Chlorine Donor
2020-08-04
1
Visible-Light-Induced Pd-Catalyzed Radical Strategy for Constructing C-Vinyl Glycosides
2020-08-04
1
Asymmetric Ruthenium-Catalyzed Hydrogenation of Terpyridine-Type N-Heteroarenes: Direct Access to Chiral Tridentate Nitrogen Ligands
2020-08-03
1
Selective C-5 Oxidative Radical Silylation of Imidazopyridines Promoted by Lewis Acid
2020-08-03
1
Synthesis of Vitamin B12-Antibiotic Conjugates with Greatly Improved Activity against Gram-Negative Bacteria
2020-08-03
1
A B2(OH)4-Mediated Synthesis of 2-Substituted Indazolone and Its Application in a DNA-Encoded Library
2020-08-01
1
Slicing and Splicing of Bromodifluoro-N-arylacetamides: Dearomatization and Difunctionalization of Pyridines
2020-08-01
1
Copper-Catalyzed Asymmetric Cyanation of Alkenes via Carbonyl-Assisted Coupling of Alkyl-Substituted Carbon-Centered Radicals
2020-07-31
1
Ligand-Accelerated Palladium(II)-Catalyzed Enantioselective Amination of C(sp2)–H Bonds
2020-07-31
1
Nickel(II)-Catalyzed Borylation of Alkenyl Methyl Ethers via C–O Bond Cleavage
2020-07-31
1
Asymmetric Synthesis of 3,3′-Tetrahydrofuryl Spirooxindoles via Palladium-Catalyzed [3+2] Cycloadditions of Methyleneindolinones with Vinylethylene Carbonates
2020-07-29
1
Brønsted Acid Catalyzed Cyclization of Aminodiazoesters with Aldehydes to 3-Carboxylate-N-Heterocycles
2020-07-29
1
Divergent Domino Reactions of Prop-2-ynylsulfonium Salts: Access to Sulfur-Containing Benzo-Fused Dioxabicyclo[3.3.1]nonanes and Dihydrofuro[2,3-c]chromenes
2020-07-29
1
Indoline Catalyzed Acylhydrazone/Oxime Condensation under Neutral Aqueous Conditions
2020-07-29
0.38
Synthesis of N–H-Free 1,4-Dihydroisoquinoline-3(2H)-ones via Pd-Catalyzed C–H Olefination Using Polyfluorosulfinyl as the Auxiliary Group
2020-07-29
1
Visible-Light-Induced Beckmann Rearrangement by Organic Photoredox Catalysis
2020-07-29
1
Construction of a Highly Diastereoselective Aldol Reaction System with l-Threonine Aldolase by Computer-Assisted Rational Molecular Modification and Medium Engineering
2020-07-27
1
Rhodium-Catalyzed Carbonylative Synthesis of Aryl Salicylates from Unactivated Phenols
2020-07-27
0.13
BI-OAc-Accelerated C3–H Alkylation of Quinoxalin-2(1H)-ones under Visible-Light Irradiation
2020-07-24
1
Synthesis of Cyclophane-Braced Peptide Macrocycles via Palladium-Catalyzed Intramolecular C(sp3)–H Arylation of N-Methyl Alanine at C-Termini
2020-07-24
1
Phakefustatins A–C: Kynurenine-Bearing Cycloheptapeptides as RXRα Modulators from the Marine Sponge Phakellia fusca
2020-07-23
1
Radical-Mediated Distal Ipso-Migration of O/S-Containing Heteroaryls and DFT Studies for Migratory Aptitude
2020-07-23
1
Cobalt-Catalyzed Reductive C–O Bond Cleavage of Lignin β-O-4 Ketone Models via In Situ Generation of the Cobalt–Boryl Species
2020-07-22
1
Enantioselective Remote C(sp3)–H Cyanation via Dual Photoredox and Copper Catalysis
2020-07-22
1
Regio- and Stereoselective Photoredox-Catalyzed Atom Transfer Radical Addition of Thiosulfonates to Aryl Alkynes
2020-07-22
0.75
Catalytic Asymmetric Transfer Hydrogenation of trans-Chalcone Derivatives Using BINOL-derived Boro-phosphates
2020-07-21
0.50
Direct Synthesis of Mono-α-arylated Ketones from Alcohols and Olefins via Ni-Catalyzed Oxidative Cross-Coupling
2020-07-21
1
Simultaneous Implementation of N-Heterocycle-Fused Bridge and Modified Pyrrole Unit on Ni(II) Porphyrin Dimers
2020-07-21
1
Copper(0)/PPh3-Mediated Bisheteroannulations of o-Nitroalkynes with Methylketoximes Accessing Pyrazo-Fused Pseudoindoxyls
2020-07-20
1
Tetrahydroxydiboron-Promoted Radical Addition of Alkynols
2020-07-19
1
Co(III)-Catalyzed Annulative Vinylene Transfer via C–H Activation: Three-Step Total Synthesis of 8-Oxopseudopalmatine and Oxopalmatine
2020-07-17
1
Copper-Catalyzed Selective Arylation of Nitriles with Cyclic Diaryl Iodonium Salts: Direct Access to Structurally Diversified Diarylmethane Amides with Potential Neuroprotective and Anticancer Activities
2020-07-17
1
Gold-Catalyzed Intermolecular Formal [4 + 2 + 2]-Cycloaddition of Anthranils with Allenamides
2020-07-17
1
Synthesis of 2-Formylpyrroles from Pyridinium Iodide Salts
2020-07-17
1
[4 + 2]-Annulation of Prop-2-ynylsulfonium Salts and Isatoic Anhydrides: Access to 3-Methylthio-4-quinolones
2020-07-17
1
A One-Step Approach to N-(Hetero)aryl-3,5-dinitropyrazoles from (Hetero)aryl Amines
2020-07-16
1
Silver(I)-Mediated Cascade Reaction of 2-(1-Alkynyl)-2-alken-1-ones with 2-Naphthols
2020-07-16
1
Stereoselective Synthesis of Vinylcyclopropa[b]indolines via a Rh-Migration Strategy
2020-07-16
0.67
Ag(I)-Catalyzed Addition of Cyclopropenones and Nitrones to Access Imides
2020-07-14
1
Asymmetric Transfer Hydrogenation of N-Unprotected Indoles with Ammonia Borane
2020-07-14
1
Copper-Catalyzed Direct C(sp3)–H Alkoxylation to Access Quaternary α-Alkoxylated Amino Acid Derivatives
2020-07-14
1
Enantioselective [4 + 2] Cycloaddition Reaction of Vinylquinolines with Dienals Enabled by Synergistic Organocatalysis
2020-07-14
0.93
Imine Amidation Catalyzed by a Chiral VAPOL Calcium Phosphate
2020-07-14
1
Iodine-Mediated Electrochemical C(sp2)–H Amination: Switchable Synthesis of Indolines and Indoles
2020-07-14
1
Palladium-Catalyzed Imidoylation-Triggered [2 + 2 + 1] Cyclization of Internal Alkyne with Isocyanides
2020-07-14
1
Perfluoroalkylation of Thiosulfonates: Synthesis of Perfluoroalkyl Sulfides
2020-07-10
1
Redox-Neutral P(O)–N Coupling between P(O)–H Compounds and Azides via Dual Copper and Photoredox Catalysis
2020-07-10
0.95
Two Reaction Modes of Pyridinium 1,4-Zwitterionic Thiolates with Sulfenes: Synthesis of 3H-1,2-Dithiole 2,2-Dioxides, 1,9a-Dihydropyrido[2,1-c][1,4]thiazines, and Indolizines
2020-07-10
1
A Bifunctional Ligand Enables Gold-Catalyzed Hydroarylation of Terminal Alkynes under Soft Reaction Conditions
2020-07-09
0.72
CaCl2-Promoted Dehydroxytrifluoromethylselenolation of Alcohols with [Me4N][SeCF3]
2020-07-09
1
Construction of Spironaphthalenones via Gold-Catalyzed Intramolecular Dearomatization Reaction of β-Naphthol Derivatives
2020-07-09
0.75
On-DNA Cross-Dehydrogenative Coupling Reaction toward the Synthesis of Focused DNA-Encoded Tetrahydroisoquinoline Libraries
2020-07-09
1
Selective [3 + 2] Cycloaddition of Cyclopropenone Derivatives and Elemental Chalcogens
2020-07-09
1
Silver-Catalyzed C–H Aryloxydifluoromethylation and Arylthiodifluoromethylation of Heteroarenes
2020-07-09
1
Substituent Effect Induces Emission Modulation of Stilbene Photoswitches by Spatial Tuning of the N/B Electronic Constraints
2020-07-09
1
Twisted Bodipy Derivative as a Heavy-Atom-Free Triplet Photosensitizer Showing Strong Absorption of Yellow Light, Intersystem Crossing, and a High-Energy Long-Lived Triplet State
2020-07-09
0.67
Zwitterion-Catalyzed Intermolecular Bromoesterifications
2020-07-08
1
Double Enzyme-Catalyzed One-Pot Synthesis of Enantiocomplementary Vicinal Fluoro Alcohols
2020-07-07
1
I2-Catalyzed Aerobic α,β-Dehydrogenation and Deamination of Tertiary Alkylamines: Highly Selective Synthesis of Polysubstituted Pyrimidines via Hidden Acyclic Enamines
2020-07-07
1
Ruthenium-Catalyzed Brook Rearrangement Involved Domino Sequence Enabled by Acylsilane–Aldehyde Corporation
2020-07-07
1
Site-Selective Pyridyl Alkyl Ketone Synthesis from N-Alkenoxypyridiniums through Boekelheide-Type Rearrangements
2020-07-07
0.67
Regioselective Hydroboration and Hydrosilylation of N-Heteroarenes Catalyzed by a Zinc Alkyl Complex
2020-07-06
1
Rh(III)-Catalyzed C(sp3)–H Acetoxylation of 8-Methylquinolines
2020-07-06
1
Rhodium-Catalyzed Sequential Cycloisomerization/Aldol Addition of Cyclopropene Carboxylic Acids with Isatins
2020-07-06
1
Visible-Light-Mediated Intermolecular Radical Conjugate Addition for the Construction of Vicinal Quaternary Carbon Centers
2020-07-06
1
Oxidant-Induced Azolation of Electron-Rich Phenol Derivatives
2020-07-02
1
Sulfoxide Reduction/C(sp3)–S Metathesis Cascade in Ionic Liquid
2020-07-02
1
Experimental and Computational Studies on Cp*CyRh(III)/KOPiv-Catalyzed Intramolecular Dehydrogenative Cross-Couplings for Building Eight-Membered Sultam/Lactam Frameworks
2020-07-01
1
FeCl3-Mediated Synthesis of 2-(Trifluoromethyl)quinazolin-4(3H)-ones from Isatins and Trifluoroacetimidoyl Chlorides
2020-07-01
0.88
Asymmetric Aza-Diels–Alder Reactions of in Situ Generated β,β-Disubstituted α,β-Unsaturated N–H Ketimines Catalyzed by Chiral Phosphoric Acids
2020-06-30
1
Asymmetric Synthesis of Axially Chiral Anilides via Organocatalytic Atroposelective N-Acylation
2020-06-30
1
Convergent Synthesis of Dihydropyrans from Catalytic Three-Component Reactions of Vinylcyclopropanes, Diazoesters, and Diphenyl Sulfoxide
2020-06-30
1
Copper(II)-Mediated Ring Opening/Alkynylation of Tertiary Cyclopropanols by Using Nonmodified Terminal Alkynes
2020-06-30
1
Palladium-Catalyzed N-Acylation of Tertiary Amines by Carboxylic Acids: A Method for the Synthesis of Amides
2020-06-30
1
Regio- and Enantioselective Palladium-Catalyzed Asymmetric Allylation of N-Fluorenyl Trifluoromethyl Imine
2020-06-30
1
Rh(III)-Catalyzed Oxidative C–H Activation/Domino Annulation of Anilines with 1,3-Diynes: A Rapid Access to Blue-Emitting Tricyclic N,O-Heteroaromatics
2020-06-30
1
Synthesis of Thiazoles and Isothiazoles via Three-Component Reaction of Enaminoesters, Sulfur, and Bromodifluoroacetamides/Esters
2020-06-30
1
Organocatalytic Formal (3 + 2) Cycloaddition toward Chiral Pyrrolo[1,2-a]indoles via Dynamic Kinetic Resolution of Allene Intermediates
2020-06-29
0.71
Ring-Strain-Enabled Catalytic Asymmetric Umpolung C–O Bond-Forming Reactions of 1,2-Oxazetidines for the Synthesis of Functionalized Chiral Ethers
2020-06-28
1
Copper-Catalyzed Intramolecular C–H Alkoxylation of Diaryltriazoles: Synthesis of Tricyclic Triazole Benzoxazines
2020-06-26
0.79
Copper-Catalyzed N,N-Diarylation of Amides for the Construction of 9,10-Dihydroacridine Structure and Applications in the Synthesis of Diverse Nitrogen-Embedded Polyacenes
2020-06-26
1
Hexafluoroisopropanol-Promoted Disulfidation and Diselenation of Alkyne, Alkene, and Allene
2020-06-26
0.17
Merger of C–F and C–N Bond Cleavage in Cross-Electrophile Coupling for the Synthesis of gem-Difluoroalkenes
2020-06-26
1
Palladium(II)-Catalyzed Oxidative Decarboxylative [2 + 2 + 1] Annulation of Cinnamic Acids with Alkynes: Access to Polysubstituted Pentafulvenes
2020-06-26
1
Palladium-Catalyzed Asymmetric Decarboxylative [4+2] Dipolar Cycloaddition of 4-Vinyl-1,3-dioxan-2-ones with α,β-Disubstituted Nitroalkenes Enabled by a Benzylic Substituted P,N-Ligand
2020-06-26
1
Transition-Metal-Free Site-Selective γ-C(sp2)–H Monoiodination of Arenes Directed by an Aliphatic Keto Group
2020-06-26
1
Cobaloxime Catalysis for Enamine Phosphorylation with Hydrogen Evolution
2020-06-25
1
Cu(II)-Catalyzed 6π-Photocyclization of Non-6π Substrates
2020-06-25
1
Development and Mechanistic Studies of Iron-Catalyzed Construction of Csp2–B Bonds via C–O Bond Activation
2020-06-25
1
Divergent Construction of Fully Substituted Pyrroles and Cyclopentadiene Derivatives by Ynamide Annulations: 1,2-Cyclopropyl Migration versus Proton Transfer
2020-06-25
1
Nickel-Catalyzed Asymmetric Addition of Aromatic Halides to Ketones: Highly Enantioselective Synthesis of Chiral 2,3-Dihydrobenzofurans Containing a Tertiary Alcohol
2020-06-23
1
Regio- and Diastereoselective Spirocyclopropanation of Benzofuran-Derived Azadienes through 1,4-Addition-Induced Dearomatization Reaction under Mild Conditions
2020-06-23
1
Ytterbium-Catalyzed Intramolecular [3 + 2] Cycloaddition based on Furan Dearomatization to Construct Fused Triazoles
2020-06-23
1
Catalytic Asymmetric Synthesis of Vicinal Tetrasubstituted Diamines via Umpolung Cross-Mannich Reaction of Cyclic Ketimines
2020-06-22
1
Characterization of SepE and SepF for the N6-Glycosylated Adenine Structure Formation in Septacidin Biosynthesis
2020-06-21
1
Allylboronates from Vinyl Triflates and α-Chloroboronates by Reductive Nickel Catalysis
2020-06-19
1
Direct Intramolecular Aminoboration of Allenes
2020-06-19
1
Palladium-Catalyzed Fluoroarylation of gem-Difluoroenynes to Access Trisubstituted Trifluoromethyl Allenes
2020-06-19
1
Photoinduced, Copper-Catalyzed Three-Component Annulation of gem-Dialkylthio Enynes
2020-06-19
1
Ruthenium(II)-Catalyzed Ortho-C–H Alkylation of Naphthylamines with Diazo Compounds for Synthesis of 2,2-Disubstituted π-Extended 3-Oxindoles in Water
2020-06-19
0.94
An Indirect Strategy for Trifluoromethylation via an Iridium Catalyst: Approach to Generate Isocoumarin Skeletons in Bioactive Molecules
2020-06-18
1
Cobalt-Catalyzed Cycloamination: Synthesis and Photophysical Properties of Polycyclic N-Heterocycles
2020-06-18
1
Synthesis of Cyclopropanes via 1,3-Migration of Acyloxy Groups Triggered by Formation of α-Imino Rhodium Carbenes
2020-06-18
1
Tandem Oxidative Ring Expansion for Synthesis of Dibenzocyclooctaphenanthrenes
2020-06-18
0.10
1,4-Fluoroamination of 1,3-Enynes en Route to Fluorinated Allenes
2020-06-17
1
Atroposelective Synthesis of Axially Chiral 3-Arylindoles by Copper-Catalyzed Asymmetric Cross-Coupling of Indoles with Quinones and Naphthoquinones
2020-06-17
1
Catalytic Asymmetric Acyloin Rearrangements of α-Ketols, α-Hydroxy Aldehydes, and α-Iminols by N,N′-Dioxide–Metal Complexes
2020-06-17
1
Direct Synthesis of Propen-2-yl Sulfones through Cascade Reactions Using Calcium Carbide as an Alkyne Source
2020-06-17
1
General Synthesis of Chiral α,α-Diaryl Carboxamides by Enantioselective Palladium-Catalyzed Cross-Coupling
2020-06-17
1
One-Pot Synthesis of Furo[3,4-c]indolo[2,1-a]isoquinolines through Rh(III)-Catalyzed Cascade Reactions of 2-Phenylindoles with 4-Hydroxy-2-alkynoates
2020-06-17
0.97
Palladium-Catalyzed Stereoselective Hydrodefluorination of Tetrasubstituted gem-Difluoroalkenes
2020-06-17
1
Rhodium-Catalyzed Ring-Opening Hydroacylation of Alkylidenecyclopropanes with Chelating Aldehydes for the Synthesis of γ,δ-Unsaturated Ketones
2020-06-17
1
Silver-Catalyzed Trifluoromethoxylation of Alkyl Trifluoroborates
2020-06-17
1
Synthesis of 3,4-Fused Tricyclic Indoles through Cascade Carbopalladation and C–H Amination: Development and Total Synthesis of Rucaparib
2020-06-17
1
Tuning Vinylethylene Carbonates into [4 + 2] Cycloaddition via Silylation and Vinylogous Peterson Elimination
2020-06-17
1
Unnatural α-Amino Acid Synthesized through α-Alkylation of Glycine Derivatives by Diacyl Peroxides
2020-06-17
1
Visible-Light-Mediated Decarboxylative Tandem Carbocyclization of Acrylamide-Attached Alkylidenecyclopropanes: Access to Polycyclic Benzazepine Derivatives
2020-06-17
1
Asymmetric Total Syntheses of (+)-Penostatins A and C
2020-06-16
1
Copper-Catalyzed Oxalamide-Directed ortho-C–H Amination of Anilines with Alkylamines
2020-06-16
1
Acid-Promoted [3 + 1 + 1] Cyclization of N-Tosylhydrazones and Isocyanides: A Method for the Preparation of 4,5-Diaminopyrazoles
2020-06-15
1
Palladium-Catalyzed Intermolecular Heck-Type Dearomative [4 + 2] Annulation of 2H-Isoindole Derivatives with Internal Alkynes
2020-06-15
1
1,2-Hydroboration of Pyridines by Organomagnesium
2020-06-11
1
Catalytic Asymmetric Addition Reactions of Formaldehyde N,N-Dialkylhydrazone to Synthesize Chiral Nitrile Derivatives
2020-06-11
1
Isolation, Total Synthesis, and Absolute Configuration Determination of Renoprotective Dimeric N-Acetyldopamine–Adenine Hybrids from the Insect Aspongopus chinensis
2020-06-11
0.75
Ni-Catalyzed Denitrogenative Cross-Coupling of Benzotriazinones and Cyclopropanols: An Easy Access to Functionalized β-Aryl Ketones
2020-06-11
1
Highly Chemo- and Enantioselective Hydrogenation of 2-Substituted-4-oxo-2-alkenoic Acids
2020-06-10
1
Palladium-Catalyzed Site-Selective Benzocylization of Aromatic Acids with o-Fluoro-Substituted Diaryliodonium Salts toward 3,4-Benzocoumarins
2020-06-10
1
Visible-Light-Promoted Cross-Coupling Reactions of 4-Alkyl-1,4-dihydropyridines with Thiosulfonate or Selenium Sulfonate: A Unified Approach to Sulfides, Selenides, and Sulfoxides
2020-06-10
1
Palladium-Catalyzed Regioselective Coupling Cyclohexenone into Indoles: Atom-Economic Synthesis of β-Indolyl Cyclohexenones and Derivatization Applications
2020-06-09
1
gem-Dinitromethyl-Functionalized 5-Amino-1,3,4-oxadiazolate Derivatives: Alternate Route, Characterization, and Property Analysis
2020-06-09
0.30
Characterization of Tailoring Methyltransferases Involved in K-41A Biosynthesis: Modulating Methylation to Improve K-41A Anti-infective Activity
2020-06-08
0.89
Cu-Catalyzed C–H Alkenylation of Benzoic Acid and Acrylic Acid Derivatives with Vinyl Boronates
2020-06-08
0.80
Stereodivergent Synthesis of α-Quaternary Serine and Cysteine Derivatives Containing Two Contiguous Stereogenic Centers via Synergistic Cu/Ir Catalysis
2020-06-06
1
Free-Radical-Promoted Dehydrogenative Coupling of Polyfluorinated Alcohol with Quinone, Chromone, and Coumarin
2020-06-05
1
Cu(I)-Catalyzed Asymmetric α-Allenylation of Activated Ketimines with 3-Butynoates
2020-06-04
1
Fe-Catalyzed Sequential C(sp3)–H/N–H Annulation of 2-Methylindoles with Ethyl Trifluoropyruvate at Room Temperature: Construction of Pyrrolo[1,2-α]indoles
2020-06-04
1
Rapid Synthesis of Alkenylated BINOL Derivatives via Rh(III)-Catalyzed C–H Bond Activation
2020-06-04
1
Reciprocal-Activation Strategy for Allylic Sulfination with Unactivated Allylic Alcohols
2020-06-04
0.97
Selective Recognition of Chloride Anion in Water
2020-06-04
1
Remarkable Ligand Effect on Rh-Catalyzed C–H-Active [3 + 2] Annulation of Ketimines and Alkynes
2020-06-03
1
Ruthenium-Catalyzed Hydrogen Evolution o-Aminoalkylation of Phenols with Cyclic Amines
2020-06-03
1
Stereoselective Construction of the Highly Congested Tricyclic Core Structure in Leucosceptroid H
2020-06-03
1
Convergent Synthesis of Calcium-Dependent Antibiotic CDA3a and Analogues with Improved Antibacterial Activity via Late-Stage Serine Ligation
2020-06-02
1
Curved Carbon Skeleton in Oriented External Electric Fields: Modulated Curvature, Directional Bowl Inversion, and Face-Selective Cycloadditions of Corannulene
2020-06-02
1
Discovery, Biosynthesis, and Heterologous Production of Loonamycin, a Potent Anticancer Indolocarbazole Alkaloid
2020-06-02
1
Enantioselective Construction of Spiro Quaternary Carbon Stereocenters via Pd-Catalyzed Intramolecular α-Arylation
2020-06-02
1
O-Phosphination of Aldehydes/Ketones toward Phosphoric Esters: Experimental and Mechanistic Studies
2020-06-02
1
Pd-Catalyzed Asymmetric Allylic Substitution Cascade of But-2-ene-1,4-diyl Dimethyl Dicarbonate for the Synthesis of Chiral 2,3-Dihydrofurans
2020-06-02
1
Geometrically Selective Denitrative Trifluoromethylthiolation of β-Nitrostyrenes with AgSCF3 for (E)-Vinyl Trifluoromethyl Thioethers
2020-06-01
1
Activation and Characterization of Bohemamine Biosynthetic Gene Cluster from Streptomyces sp. CB02009
2020-05-28
1
Azetidine-Containing Heterospirocycles Enhance the Performance of Fluorophores
2020-05-28
1
Cobalt/Bisoxazolinephosphine-Catalyzed Asymmetric Alkynylation of Isatins
2020-05-28
1
Diazo Activation with Diazonium Salts: Synthesis of Indazole and 1,2,4-Triazole
2020-05-28
0.14
Peptide-Catalyzed Highly Asymmetric Cross-Aldol Reaction of Aldehydes to Biomimetically Synthesize 1,4-Dicarbonyls
2020-05-28
1
Radical Pentafluoroethylation of Unactivated Alkenes Using CuCF2CF3
2020-05-28
1
Selective Synthesis of Pyrazolo[1,2-a]pyrazolones and 2-Acylindoles via Rh(III)-Catalyzed Tunable Redox-Neutral Coupling of 1-Phenylpyrazolidinones with Alkynyl Cyclobutanols
2020-05-28
1
Biosynthesis and Chemical Diversification of Verucopeptin Leads to Structural and Functional Versatility
2020-05-27
1
Cobalt-Catalyzed Switchable Intramolecular Thioenolization/C–H Thiolation and C(sp2)–H/C(sp3)–H Dehydrogenative Coupling
2020-05-27
1
Palladium-Catalyzed C-2 and C-3 Dual C–H Functionalization of Indoles: Synthesis of Fluorinated Isocryptolepine Analogues
2020-05-27
1
Regioselective and Diastereoselective Dearomative Multifunctionalization of In-Situ-Activated Azaarenes: An Access to Bridged Azaheterocycles
2020-05-27
1
Remote and Selective C(sp2)–H Olefination for Sequential Regioselective Linkage of Phenanthrenes
2020-05-27
0.90
A Versatile Synthesis of Vinyl-Substituted Heterocycles via Regio- and Enantioselective Pd-Catalyzed Tandem Allylic Substitution
2020-05-26
1
Catalytic Asymmetric [3 + 2] Annulation via Indolyl Copper–Allenylidene Intermediates: Diastereo- and Enantioselective Assembly of Pyrrolo[1,2-a]indoles
2020-05-26
1
Crotonpenoids A and B, Two Highly Modified Clerodane Diterpenoids with a Tricyclo[7.2.1.02,7]dodecane Core from Croton yanhuii: Isolation, Structural Elucidation, and Biomimetic Semisynthesis
2020-05-26
1
One-Pot Preparation of 9,10-Dihydrophenanthrenes Initiated by Rhodium(III)-Catalyzed C–H Activation and Relay Diels–Alder Reaction
2020-05-26
1
Organocatalytic Approach for Assembling Flavanones via a Cascade 1,4-Conjugate Addition/oxa-Michael Addition between Propargylamines with Water
2020-05-22
1
Asymmetric Total Syntheses of (−)-Fennebricin A, (−)-Renieramycin J, (−)-Renieramycin G, (−)-Renieramycin M, and (−)- Jorunnamycin A via C–H Activation
2020-05-21
1
Thermo/Anion Dual-Responsive Supramolecular Organoplatinum–Crown Ether Complex
2020-05-21
0.83
tBuOK-Promoted Cyclization of Imines with Aryl Halides
2020-05-21
1
Cobalt-Bisoxazoline-Catalyzed Enantioselective Cross-Coupling of α-Bromo Esters with Alkenyl Grignard Reagents
2020-05-20
1
Cobalt-Catalyzed Asymmetric Cross-Coupling Reaction of Fluorinated Secondary Benzyl Bromides with Lithium Aryl Boronates/ZnBr2
2020-05-20
1
Palladium-Catalyzed Asymmetric (2+3) Annulation of p-Quinone Methides with Trimethylenemethanes: Enantioselective Synthesis of Functionalized Chiral Spirocyclopentyl p-Dienones
2020-05-20
1
Visible-Light-Induced Dehydrohalogenative Coupling for Intramolecular α-Alkenylation: A Way to Build Seven- and Eight-Membered Rings
2020-05-20
0.31
Waikikiamides A–C: Complex Diketopiperazine Dimer and Diketopiperazine–Polyketide Hybrids from a Hawaiian Marine Fungal Strain Aspergillus sp. FM242
2020-05-20
0.06
[2 + 2 + 1] Heteroannulation of Alkenes with Enynyl Benziodoxolones and Silver Nitrite Involving C≡C bond Oxidative Cleavage: Entry to 3-Aryl-Δ2-isoxazolines
2020-05-20
1
AIBN-Induced Remote Trifluoromethyl-Alkynylation of Thioalkynes
2020-05-19
1
Nickel-Catalyzed Homo- and Cross-Coupling of Allyl Alcohols via Allyl Boronates
2020-05-19
1
The C–H Activation/Bidirecting Group Strategy for Selective Direct Synthesis of Diverse 1,1′-Biisoquinolines
2020-05-19
1
pH-Controlled Chirality Inversion in Enantiodifferentiating Photocyclodimerization of 2-Antharacenecarboxylic Acid Mediated by γ-Cyclodextrin Derivatives
2020-05-17
1
Asymmetric (4 + 3) and (4 + 1) Annulations of Isatin-derived Morita–Baylis–Hillman Carbonates to Construct Diverse Chiral Heterocyclic Frameworks
2020-05-15
1
A Simple Protocol for the Stereoselective Construction of Enaminyl Sulfonyl Fluorides
2020-05-14
1
Blue Light Promoted Difluoroalkylation of Aryl Ketones: Synthesis of Quaternary Alkyl Difluorides and Tetrasubstituted Monofluoroalkenes
2020-05-14
1
Copper-Catalyzed Chemodivergent Cyclization of N-(ortho-alkynyl)aryl-Pyrrole and Indoles
2020-05-14
1
Ruthenium-Catalyzed Highly Enantioselective Synthesis of cis-3-Quinuclidinols via DKR Asymmetric Transfer Hydrogenation
2020-05-14
1
Selective Inclusion of Fluoride within the Cavity of a Two-Wall Bis-calix[4]pyrrole
2020-05-14
0.64
Base-Promoted Radical Azofluoromethylation of Unactivated Alkenes
2020-05-13
0.20
Directed Cobalt-Catalyzed anti-Markovnikov Hydroalkylation of Unactivated Alkenes Enabled by “Co–H” Catalysis
2020-05-13
1
Electrochemical Annulation–Iodosulfonylation of 1,5-Enyne-containing para-Quinone Methides (p-QMs) to Access (E)-Spiroindenes
2020-05-13
1
Rhodium(III)-Catalyzed [4+3] Annulation of N-Aryl-pyrazolidinones and Propargylic Acetates: Access to Benzo[c][1,2]diazepines
2020-05-13
0.96
Structural Diversification of Andiconin-Derived Natural Products by α-Ketoglutarate-Dependent Dioxygenases
2020-05-13
0.33
Asymmetric Linear-Selective Hydroformylation of 1,1-Dialkyl Olefins Assisted by a Steric-Auxiliary Strategy
2020-05-12
1
Quantum Mechanical–NMR-Aided Configuration and Conformation of Two Unreported Macrocycles Isolated from the Soft Coral Lobophytum sp.: Energy Calculations versus Coupling Constants
2020-05-12
0.60
When Anthracene and Quinone Avoid Cycloaddition: Acid-Catalyzed Redox Neutral Functionalization of Anthracene to Aryl Ethers
2020-05-12
1
N-Iodosuccinimide-Mediated Dimerization of 2-Alkynylnaphthols: A Highly Diastereoselective Construction of Bridged Polycyclic Compounds via Vinylidene ortho-Quinone Methide Intermediate
2020-05-11
1
Synthesis of 2-Imino-1,3,4-thiadiazoles from Hydrazides and Isothiocyanates via Sequential Oxidation and P(NMe2)3-Mediated Annulation Reactions
2020-05-10
1
A General One-Pot Protocol for Hindered N-Alkyl Azaheterocycles from Tertiary Carboxylic Acids
2020-05-08
0.57
Copper-Mediated DNA-Compatible One-Pot Click Reactions of Alkynes with Aryl Borates and TMS-N3
2020-05-08
1
Nickel-Catalyzed Formal Aminocarbonylation of Secondary Benzyl Chlorides with Isocyanides
2020-05-08
1
Palladium-Catalyzed Regio- and Stereoselective Cross-Coupling of Vinylethylene Carbonates with Ketimine Esters to Generate (Z)-Tri- and Tetra-substituted Allylic Amino Acid Derivatives
2020-05-08
1
Rh(I)-Catalyzed C6-Selective Decarbonylative Alkylation of 2-Pyridones with Alkyl Carboxylic Acids and Anhydrides
2020-05-08
0.83
Synthesis of Spiroisoxazolines via an Oximation/Dearomatization Cascade under Air
2020-05-08
1
Iron-Catalyzed Oxidative Coupling of Indoline-2-ones with Aminobenzamides via Dual C–H Functionalization
2020-05-07
1
Nickel(II)-Catalyzed Addition of Aryl-, Alkenyl-, and Alkylboronic Acids to Alkenylazaarenes
2020-05-07
1
Sequential Visible-Light and N-Heterocyclic Carbene Catalysis: Stereoselective Synthesis of Tetrahydropyrano[2,3-b]indoles
2020-05-07
1
Enantioselective Copper-Catalyzed Remote C(sp3)–H Alkynylation of Linear Primary Sulfonamides
2020-05-05
1
DNA Compatible Intermolecular Wittig Olefination for the Construction of α, β-Unsaturated Carbonyl Compounds
2020-05-04
1
Organocatalytic Regiodivergent Ring Expansion of Cyclobutanones for the Enantioselective Synthesis of Azepino[1,2-a]indoles and Cyclohepta[b]indoles
2020-05-04
1
Palladium-Catalyzed Cascade Decarboxylative Amination/6-endo-dig Benzannulation of o-Alkynylarylketones with N-Hydroxyamides To Access Diverse 1-Naphthylamine Derivatives
2020-05-04
1
K2S as Sulfur Source and DMSO as Carbon Source for the Synthesis of 2-Unsubstituted Benzothiazoles
2020-05-03
1
Acylation of Aryl Halides and α-Bromo Acetates with Aldehydes Enabled by Nickel/TBADT Cocatalysis
2020-05-01
1
Carbocation versus Carbene Controlled Chemoselectivity: DFT Study on Gold- and Silver-Catalyzed Alkylation/Cyclopropanation of Indoles with Vinyl Diazoesters
2020-05-01
0.80
Chiral Binaphthyl Box-Copper-Catalyzed Enantioselective Tandem Michael–Ketalization Annulations for Optically Active Aryl and Heteroaryl Fused Bicyclicnonanes
2020-05-01
1
Pd-Catalyzed Regiodivergent Synthesis of Diverse Oxindoles Enabled by the Versatile Heck Reaction of Carbamoyl Chlorides
2020-05-01
1
Visible-Light-Induced Palladium-Catalyzed Intermolecular Narasaka–Heck Reaction at Room Temperature
2020-05-01
1
Catalytic C–C Cleavage/Alkyne–Carbonyl Metathesis Sequence of Cyclobutanones
2020-04-30
1
Pd-Catalyzed Cross-Coupling of Highly Sterically Congested Enol Carbamates with Grignard Reagents via C–O Bond Activation
2020-04-30
1
Electrochemical Oxidative Phosphorylation of Aldehyde Hydrazones
2020-04-28
1
Thiol Activation toward Selective Thiolation of Aromatic C–H Bond
2020-04-28
1
A Dual-Protein Cascade Reaction for the Regioselective Synthesis of Quinoxalines
2020-04-27
1
Synthesis of ortho-Phenolic Sulfilimines via an Intermolecular Sulfur Atom Transfer Cascade Reaction
2020-04-27
1
Postulated Biogenesis-Guided Total Synthesis and Structural Revision of 2,18-seco-Lankacidinol A
2020-04-24
1
Total Synthesis of Fawcettimine-Type Alkaloid, Lycojaponicumin A
2020-04-24
1
Visible-Light-Induced Regioselective Dicarbonylation of Indolizines with Oxoaldehydes via Direct C–H Functionalization
2020-04-23
1
Absolute Configurations and Stereochemical Inversion Mechanism of Epimeric Securinega Alkaloids from Flueggea suffruticosa
2020-04-22
1
Structure-Guided Directed Evolution of a Carbonyl Reductase Enables the Stereoselective Synthesis of (2S,3S)-2,2-Disubstituted-3-hydroxycyclopentanones via Desymmetric Reduction
2020-04-22
1
Copper-Catalyzed Radical N-Demethylation of Amides Using N-Fluorobenzenesulfonimide as an Oxidant
2020-04-21
0.83
Redox Neutral Radical-Relay Cobalt Catalysis toward C–H Fluorination and Amination
2020-04-20
1
Cobalt-Catalyzed Regio- and Enantioselective Allylic Alkylation of Malononitriles
2020-04-17
1
Directing-Group-Controlled Ring-Opening Addition and Hydroarylation of Oxa/azabenzonorbornadienes with Arenes via C–H Activation
2020-04-17
1
Terpenoids from Resina Commiphora Regulating Lipid Metabolism via Activating PPARα and CPT1 Expression
2020-04-17
1
Transamidation for the Synthesis of Primary Amides at Room Temperature
2020-04-16
0.50
Directing-Group-Based Strategy Enabling Intermolecular Heck-Type Reaction of Cycloketone Oxime Esters and Unactivated Alkenes
2020-04-15
1
Eleucanainones A and B: Two Dimeric Structures from the Bulbs of Eleutherine americana with Anti-MRSA Activity
2020-04-15
1
Access to Optically Enriched α-Aryloxycarboxylic Esters via Carbene-Catalyzed Dynamic Kinetic Resolution and Transesterification
2020-04-14
0.48
Bimetallic Catalytic Tandem Reaction of Acyclic Enynones: Enantioselective Access to Tetrahydrobenzofuran Derivatives
2020-04-14
1
Spiroinonotsuoxotriols A and B, Two Highly Rearranged Triterpenoids from Inonotus obliquus
2020-04-14
1
Switchable Copper-Catalyzed Approach to Benzodithiole, Benzothiaselenole, and Dibenzodithiocine Skeletons
2020-04-14
0.58
A Family of BODIPY-like Highly Fluorescent and Unsymmetrical Bis(BF2) Pyrrolyl–Acylhydrazone Chromophores: BOAPY
2020-04-13
1
Copper-Catalyzed Annulation of Oxime Acetates with α-Amino Acid Ester Derivatives: Synthesis of 3-Sulfonamido/Imino 4-Pyrrolin-2-ones
2020-04-13
1
Organocatalytic Aza-Michael/Michael Cyclization Cascade Reaction: Enantioselective Synthesis of Spiro-oxindole Piperidin-2-one Derivatives
2020-04-13
1
Photo-on-Demand Synthesis of Chloroformates with a Chloroform Solution Containing an Alcohol and Its One-Pot Conversion to Carbonates and Carbamates
2020-04-13
0.25
Stereocomplementary Synthesis of Pharmaceutically Relevant Chiral 2-Aryl-Substituted Pyrrolidines Using Imine Reductases
2020-04-13
1
Decarboxylative Thiolation of Redox-Active Esters to Thioesters by Merging Photoredox and Copper Catalysis
2020-04-12
1
Cobalt-Catalyzed Regioselective Carboamidation of Alkynes with Imides Enabled by Cleavage of C–N and C–C Bonds
2020-04-10
1
Cyanide Boosting Copper Catalysis: A Mild Approach to Fluorescent Benzazole Derivatives from Nonemissive Schiff Bases in Biological Media
2020-04-10
1
Liquid-Phase Total Synthesis of Plecanatide Aided by Diphenylphosphinyloxyl Diphenyl Ketone (DDK) Derivatives
2020-04-10
1
Photocatalytic Remote Oxyfluoroalkylation of Heteroalkynes: Regio-, Stereo-, and Site-Selective Access to Complex Fluoroalkylated (Z)-Alkenes
2020-04-10
1
Rhodium(III)-Catalyzed Asymmetric Addition of Inert Arene C–H Bond to Aldehydes To Afford Enantioenriched Phthalides
2020-04-10
1
Rhodium(III)-Catalyzed Kinetic Resolution of Racemic 1,6-Dienes via Asymmetric Borylative Cyclization
2020-04-10
1
Titanocene-Catalyzed Reductive Domino Epoxide Ring Opening/Defluorinative Cross-Coupling Reaction
2020-04-10
1
Deacetylative Aryl Migration of Diaryliodonium Salts with C(sp2)–N Bond Formation toward ortho-Iodo N-Aryl Sulfonamides
2020-04-09
1
Copper-Catalyzed Functionalization of Aza-Aromatic Rings with Fluoroalcohols via Direct C(sp2)–H/C(sp3)–H Coupling Reactions
2020-04-08
1
Pd-Catalyzed Oxidative Annulation of Aryl Ethers with Alkynes: Synthesis of Functionalized Spirocycles and Naphthalenes
2020-04-08
1
Computation-Guided Development of the “Click” ortho-Quinone Methide Cycloaddition with Improved Kinetics
2020-04-07
1
Diastereoselective Construction of Cyclopropane-Fused Tetrahydroquinolines via a Sequential [4 + 2]/[2 + 1] Annulation Reaction
2020-04-07
1
Electrochemical Oxidative Dehydrogenative Phosphorylation of N-Heterocycles with P(O)–H Compounds in Imidazolium-Based Ionic Liquid
2020-04-07
1
Electroreductive 4-Pyridylation of Electron-deficient Alkenes with Assistance of Ni(acac)2
2020-04-07
0.71
Time-Economical Radical Cascade Cyclization/Haloazidation of 1,6-Enynes: Construction of Highly Functional Succinimide Derivatives
2020-04-07
1
A Hg(OTf)2-Catalyzed Enolate Umpolung Reaction Enables the Synthesis of Coumaran-3-ones and Indolin-3-ones
2020-04-06
1
Multistep Photoisomerization of Dimesitylboron-Functionalized Stilbene Analogues
2020-04-06
0.13
Three-Component Borylallenylation of Alkynes: Access to Densely Boryl-Substituted Ene-allenes
2020-04-06
1
Cascade Claisen and Meinwald Rearrangement for One-Pot Divergent Synthesis of Benzofurans and 2H-Chromenes
2020-04-03
1
Construction of Thiazole-Fused Dihydropyrans via Formal [4 + 2] Cycloaddition Reaction on DNA
2020-04-03
1
Gold-Catalyzed Oxidative Cascade Cyclization of 1,3-Diynamides: Polycyclic N-Heterocycle Synthesis via Construction of a Furopyridinyl Core
2020-04-03
1
Ni-Catalyzed Allylic Dearomatization Reaction of β-Naphthols with Allylic Alcohols
2020-04-03
1
Nickel-Catalyzed Formal Aminocarbonylation of Unactivated Alkyl Iodides with Isocyanides
2020-04-03
1
Alternarin A, a Drimane Meroterpenoid, Suppresses Neuronal Excitability from the Coral-Associated Fungi Alternaria sp. ZH-15
2020-04-02
0.78
Photocatalytic [2 + 2] Cycloaddition in DNA-Encoded Chemistry
2020-04-02
0.50
Rhodium(III)-Catalyzed Asymmetric C–H Activation of N-Methoxybenzamide with Quinone and Its Application in the Asymmetric Synthesis of a Dihydrolycoricidine Analogue
2020-04-02
1
Brønsted Acid Catalyzed Enantioselective Assembly of Spirochroman-3,3-oxindoles
2020-04-01
1
Copper(I)-Catalyzed Ketenimine Formation/Aza-Claisen Rearrangement Cascade for Stereoselective Synthesis of α-Allylic Amidines
2020-04-01
1
Iron-Catalyzed Borylation of Aryl Ethers via Cleavage of C–O Bonds
2020-04-01
1
Ruthenium-Catalyzed Diastereoselective Synthesis of Fully Substituted Pyrrolidines from Anilines and Diazo Pyruvates
2020-04-01
1
Copper-Catalyzed Trifluoromethylation of Ynones Coupled with Dearomatizing Spirocyclization of Indoles: Access to CF3-Containing Spiro[cyclopentane-1,3′-indole]
2020-03-31
1
Copper-free Sandmeyer-type Reaction for the Synthesis of Sulfonyl Fluorides
2020-03-31
1
CuBr-Catalyzed α-Arylation and Aerobic Oxidative Dehydrogenative C–N Coupling for the Synthesis of Spiro[cyclohexane-1,12′-isoindolo[1,2-b]quinazolin]-10′-one Derivatives
2020-03-31
1
Iron-Catalyzed Alkylazidation of 1,1-Disubstituted Alkenes with Diacylperoxides and TMSN3
2020-03-31
1
Synthesis of Tetramic Acid Derivatives via a Tandem Umpolung Alkylation/Reduction/Cyclization Reaction of γ-Hydrazono β-Ketoester
2020-03-31
0.13
Understanding the Chemoselectivity in Palladium-Catalyzed Three-Component Reaction of o-Bromobenzaldehyde, N-Tosylhydrazone, and Methanol
2020-03-31
1
Visible-Light-Induced, Base-Promoted Transition-Metal-Free Dehalogenation of Aryl Fluorides, Chlorides, Bromides, and Iodides
2020-03-31
1
Gold(I)-Catalyzed [8+4] Cycloaddition of 1,4-All-Carbon Dipoles with Tropone
2020-03-30
1
Hydrogen-Bond-Mediated Aglycone Delivery: Synthesis of β-d-Fructofuranosides
2020-03-30
1
3,3′-Disubstituted Oxindoles Formation via Copper-Catalyzed Arylboration and Arylsilylation of Alkenes
2020-03-27
1
Development of a C2-Symmetric Chiral aza Spirocyclic Diol
2020-03-27
1
Highly Regio- and Enantioselective Hydrogenation of Conjugated α-Substituted Dienoic Acids
2020-03-27
1
Palladium-Catalyzed Tandem Dehydrogenative [4 + 2] Annulation of Terminal Olefins with N-Sulfonyl Amides via C–H Activations
2020-03-27
1
Stereoselective Phenylselenoglycosylation of Glycals Bearing a Fused Carbonate Moiety toward the Synthesis of 2-Deoxy-β-galactosides and β-Mannosides
2020-03-27
1
Gold and Brønsted Acid Catalyzed Spirocyclization of 2- and 3-Indolyl-Tethered 1,4-Enyne Acetates to Spiro[4,n]alkyl[b]indoles
2020-03-26
0.20
Asymmetric Catalytic Diverse Ring Opening/Cycloadditions of Cyclobutenones with (E)-Alkenyloxindoles and (E)-Dioxopyrrolidines
2020-03-25
1
Rh-Catalyzed C–H Amination/Annulation of Acrylic Acids and Anthranils by Using −COOH as a Deciduous Directing Group: An Access to Diverse Quinolines
2020-03-25
1
Copper-Catalyzed Remote C(sp3)–H Amination of Carboxamides
2020-03-24
1
Selective Oxidative Cleavage of 3-Methylindoles with Primary Amines Affording Quinazolinones
2020-03-24
1
Brønsted Base and Lewis Acid Cooperatively Catalyzed Asymmetric exo′-Selective [3 + 2] Cycloaddition of Trifluoromethylated Azomethine Ylides and Methyleneindolinones
2020-03-23
1
Highly Enantioselective Cobalt-Catalyzed Hydroboration of Diaryl Ketones
2020-03-23
1
Iridium-Catalyzed γ-Selective Hydroboration of γ-Substituted Allylic Amides
2020-03-23
1
Nickel-Catalyzed Asymmetric Reductive Arylbenzylation of Unactivated Alkenes
2020-03-23
1
Stereoselective Synthesis of (−)-Verazine and Congeners via a Cascade Ring-Switching Process of Furostan-26-acid
2020-03-23
1
Rhodium-Catalyzed Enantioselective Hydroselenation of Heterobicyclic Alkenes
2020-03-20
1
Carbene-Catalyzed Reaction of Indolyl Methylenemalononitriles and Enals for Access to Complex Tetrahydrocarbazoles
2020-03-19
0.33
Direct Synthesis of Chiral NH Lactams via Ru-Catalyzed Asymmetric Reductive Amination/Cyclization Cascade of Keto Acids/Esters
2020-03-19
1
NHC-Catalyzed Cascade Reaction between β-Methyl Enals and Dienones for Quick Construction of Complex Multicyclic Lactones
2020-03-19
0.77
Total Synthesis of (±)-11-O-Debenzoyltashironin via Palladium-Catalyzed 5-endo Ene-yne Cyclization Enabled trans-5–6 Ring Fusion
2020-03-19
1
Bismuth(III)-Catalyzed Sequential Enamine–Imine Tautomerism/2-Aza-Cope Rearrangement of Stable β-Enaminophosphonates: One-Pot Synthesis of β-Aminophosphonates
2020-03-18
1
Chartspiroton, a Tetracyclic Spiro-naphthoquinone Derivative from a Medicinal Plant Endophytic Streptomyces
2020-03-18
1
Hydride Transfer Initiated Redox-Neutral Cascade Cyclizations of Aurones: Facile Access to [6,5] Spirocycles
2020-03-18
1
Hyperprins A and B, Two Complex Meroterpenoids from Hypericum przewalskii
2020-03-18
1
Iron-Catalyzed Silylation of (Hetero)aryl Chlorides with Et3SiBpin
2020-03-18
1
Phosphine-Catalyzed Cascade Michael Addition/[4+2] Cycloaddition Reaction of Allenoates and 2-Arylidene-1,3-indanediones
2020-03-18
1
Rhodium(III)-Catalyzed Oxidative Annulation of 4-Aminoquinolines and Acrylate through Two Consecutive C(sp2)–H Activations
2020-03-18
0.92
Visible-Light-Driven Radical Multicomponent Reaction of 2-Vinylanilines, Sulfonyl Chlorides, and Sulfur Ylides for Synthesis of Indolines
2020-03-18
1
Direct Hiyama Cross-Coupling of (Hetero)arylsilanes with C(sp2)–H Bonds Enabled by Cobalt Catalysis
2020-03-17
0.89
Fast and Low-Cost Purification Strategy for Oligosaccharide Synthesis Based on a Hop-On/Off Carrier
2020-03-17
1
Stereospecific Electrophilic Fluorocyclization of α,β-Unsaturated Amides with Selectfluor
2020-03-16
0.75
C–O Bond Silylation Catalyzed by Iron: A General Method for the Construction of Csp2–Si Bonds
2020-03-13
1
Ganoderma cochlear Metabolites as Probes to Identify a COX-2 Active Site and as in Vitro and in Vivo Anti-Inflammatory Agents
2020-03-13
1
Kinetic Resolution of Propargylic Ethers via [2,3]-Wittig Rearrangement to Synthesize Chiral α-Hydroxyallenes
2020-03-13
1
Tuning Biradical Character to Enable High and Balanced Ambipolar Charge Transport in a Quinoidal π-System
2020-03-13
1
Highly Chemoselective and Enantioselective Synthesis of 3,4-2H-Pyrindin-2-ones by an NHC-Catalyzed [3 + 3] Cyclization
2020-03-11
1
Visible-Light-Driven Copper-Catalyzed C(sp3)–O Cross-Coupling of Benzylic Radicals with Phenols
2020-03-11
1
Highly Enantioselective [3 + 2] Annulation of 3-Butynoates with β-Trifluoromethyl Enones Promoted by an Amine−Phosphine Binary Catalytic System
2020-03-10
0.44
Three-Component Minisci Reaction with 1,3-Dicarbonyl Compounds Induced by Visible Light
2020-03-10
1
Visible Light Induced Cyclization to Spirobi[indene] Skeletons from Functionalized Alkylidienecyclopropanes
2020-03-10
1
Density Functional Theory Mechanistic Study of Ni-Catalyzed Reductive Alkyne–Alkyne Cyclodimerization: Oxidative Cyclization versus Outer-Sphere Proton Transfer
2020-03-09
1
Intermolecular Vicinal Diaminative Assembly of Tetrahydroquinoxalines via Metal-free Oxidative [4 + 2] Cycloaddition Strategy
2020-03-09
1
Yb(OTf)3-Catalyzed Alkyne–Carbonyl Metathesis–Oxa-Michael Addition Relay for Diastereoselective Synthesis of Functionalized Naphtho[2,1-b]furans
2020-03-09
1
Highly Chemo-, Site-, and Enantioseletive para C–H Aminoalkylation of N-Monosubstituted Aniline Derivatives Affording 3-Amino-2-oxindoles
2020-03-06
1
Ligand-Enabled Ni–Al Bimetallic Catalysis for Nonchelated Dual C–H Annulation of Arylformamides and Alkynes
2020-03-06
1
Organocatalytic Enantioselective Construction of Heterocycle-Substituted Styrenes with Chiral Atropisomerism
2020-03-06
1
Biosynthesis of the Prenylated Salicylaldehyde Flavoglaucin Requires Temporary Reduction to Salicyl Alcohol for Decoration before Reoxidation to the Final Product
2020-03-05
0.20
Directing-Group-Enabled Cycloaddition of Azides and Alkynes toward Functionalized Triazoles
2020-03-05
1
Visible-Light-Mediated β-C–H gem-Difluoroallylation of Aldehydes and Cyclic Ketones through C–F Bond Cleavage of 1-Trifluoromethyl Alkenes
2020-03-05
1
Catalytic Annulation of Alkynyl 1,2-Diketone Leading to Hydroxy Spirocyclopenteneindenedione: An Organic Dye with Strong Crystallization-Induced Emission and Data Storage Application
2020-03-04
1
Dimericchalasine A and Amichalasines D and E: Unexpected Cytochalasan Homodimer and Heterotrimers from Aspergillus micronesiensis PG-1
2020-03-04
1
Kinetically Controlled Radical Addition/Elimination Cascade: From Alkynyl Aziridine to Fluorinated Allenes
2020-03-04
1
Nickel-Catalyzed Claisen Condensation Reaction between Two Different Amides
2020-03-04
0.50
Electrochemical Synthesis of α-Ketoamides under Catalyst-, Oxidant-, and Electrolyte-Free Conditions
2020-03-03
1
Mesoionic Carbene–Iridium Complex Catalyzed Ortho-Selective Hydrogen Isotope Exchange of Anilines with High Functional Group Tolerance
2020-03-03
1
Selective Cross-Dehydrogenative C(sp3)–H Arylation with Arenes
2020-03-03
1
Visible-Light-Driven Nitrogen Radical-Catalyzed [3 + 2] Cyclization of Vinylcyclopropanes and N-Tosyl Vinylaziridines with Alkenes
2020-03-03
1
Arenesulfonyl Fluoride Synthesis via Copper-Catalyzed Fluorosulfonylation of Arenediazonium Salts
2020-03-02
1
Isothiourea and Brønsted Acid Cooperative Catalysis: Enantioselective Construction of Dihydropyridinones
2020-03-02
1
Competitive Selection of Conformation Chirality of Water-Soluble Pillar[5]arene Induced by Amino Acid Derivatives
2020-02-28
1
Highly Enantioselective Ruthenium-Catalyzed Cascade Double Reduction Strategy: Construction of Structurally Diverse Julolidines and Their Analogues
2020-02-28
1
Iridium/Acid Cocatalyzed Direct Access to Fused Indoles via Transfer Hydrogenative Annulation of Quinolines and 1,2-Diketones
2020-02-28
1
2H-Azirines as Potential Bifunctional Chemical Linkers of Cysteine Residues in Bioconjugate Technology
2020-02-27
0.94
Activation of Chiral (Salen)TiCl2 Complex by Phosphorane for the Highly Enantioselective Cyanation of Nitroolefins
2020-02-27
1
Electrophilic Hypervalent Trifluoromethylthio-Iodine(III) Reagent
2020-02-27
1
Iron–Phosphine Complex-Catalyzed Intramolecular C(sp3)–H Amination of Azides
2020-02-27
1
Unraveling the Fungal Strategy for Tetrahydroxanthone Biosynthesis and Diversification
2020-02-27
1
Copper-Catalyzed Disulfonation of Terminal Alkynes with Sodium Arylsulfinates
2020-02-26
1
Iridium(III)-Catalyzed C–H Amidation/Cyclization of NH-Sulfoximines with N-Alkoxyamides: Formation of Thiadiazine 1-Oxides
2020-02-26
1
Construction of Polyfunctionalized 6–5–5 Fused Tricyclic Carbocycles via One-Pot Sequential Semipinacol Rearrangement/Michael Addition/Henry Reaction
2020-02-25
1
Iron-Catalyzed Reductive Vinylation of Tertiary Alkyl Oxalates with Activated Vinyl Halides
2020-02-25
1
Protecting-Group-Free Total Syntheses of (±)-Norascyronones A and B
2020-02-25
1
Total Synthesis of (−)-Gardmultimine A
2020-02-25
1
HNTf2-Catalyzed Synthesis of Hydrodibenzofurans by an Epoxidation/Semipinacol Rearrangement Cascade
2020-02-24
1
Leptosperols A and B, Two Cinnamoylphloroglucinol–Sesquiterpenoid Hybrids from Leptospermum scoparium: Structural Elucidation and Biomimetic Synthesis
2020-02-24
1
Organocatalytic Asymmetric Three-Component Povarov Reactions of Anilines and Aldehydes
2020-02-21
1
Rh(III)-Catalyzed Relay Double Carbenoid Insertion and Diannulation of Sulfoximine Benzamides with α-Diazo Carbonyl Compounds: Access to Furo[2,3-c]isochromenes
2020-02-21
1
Water Compatible Hypophosphites-d2 Reagents: Deuteration Reaction via Deutero-deiodination in Aqueous Solution
2020-02-21
1
Palladium-Catalyzed Three-Component Coupling Reaction of o-Bromobenzaldehyde, N-Tosylhydrazone, and Methanol
2020-02-20
1
Redox Cyclization of Amides and Sulfonamides with Nitrous Oxide for Direct Synthesis of Heterocycles
2020-02-20
1
Visible-Light Mediated Hydrosilylative and Hydrophosphorylative Cyclizations of Enynes and Dienes
2020-02-20
1
C(sp2)–H Bond Multiple Functionalization in Air for Construction of Tetrahydrocarbazoles with Continuous Quaternary Carbons and Polycyclic Diversification
2020-02-19
1
Cobalt-Catalyzed C–H Acetoxylation of Phenols with Removable Monodentate Directing Groups: Access to Pyrocatechol Derivatives
2020-02-19
0.89
Cycloaddition of Trifluoroacetaldehyde N-Triftosylhydrazone (TFHZ-Tfs) with Alkynes for Synthesizing 3-Trifluoromethylpyrazoles
2020-02-19
1
Direct Alkoxycarbonylation of Heteroarenes via Cu-Mediated Trichloromethylation and In Situ Alcoholysis
2020-02-19
1
Direct Synthesis of Sulfonylated Spiro[indole-3,3′-pyrrolidines] by Silver-Mediated Sulfonylation of Acrylamides Coupled with Indole Dearomatization
2020-02-19
1
Enantioselective Synthesis of Axially Chiral Biaryls via Copper-Catalyzed Thiolation of Cyclic Diaryliodonium Salts
2020-02-19
1
On-PKS Baeyer–Villiger-Type O-Atom Insertion Catalyzed by Luciferase-Like Monooxygenase OvmO during Olimycin Biosynthesis
2020-02-19
1
Sequential C–S and S–N Coupling Approach to Sulfonamides
2020-02-19
1
Copper Catalyzed Diastereo- and Enantioselective 1,4-Addition Michael Reaction of 2,3-Dioxopyrrolidines with Nitroalkanes in Aqueous Media
2020-02-18
1
Palladium-Catalyzed Four-Component Carbonylative Cyclization Reaction of Trifluoroacetimidoyl Chlorides, Propargyl Amines, and Diaryliodonium Salts: Access to Trifluoromethyl-Containing Trisubstituted Imidazoles
2020-02-18
0.88
Diastereoselective Synthesis of Cycloheptannelated Indoles via Lewis-Acid-Catalyzed (4 + 3)-Cyclization of Donor–Acceptor Cyclopropanes
2020-02-17
1
Rhodium-Catalyzed Branched and Enantioselective Direct α-Allylic Alkylation of Simple Ketones with Alkynes
2020-02-17
1
Flavipesides A–C, PKS-NRPS Hybrids as Pancreatic Lipase Inhibitors from a Marine Sponge Symbiotic Fungus Aspergillus flavipes 164013
2020-02-14
1
Intermolecular Trifluoromethyl-Hydrazination of Alkenes Enabled by Organic Photoredox Catalysis
2020-02-14
1
Organocatalytic Enantioselective γ-Elimination: Applications in the Preparation of Chiral Peroxides and Epoxides
2020-02-14
1
Copper-Catalyzed Remote C(sp3)–H Phosphorothiolation of Sulfonamides and Carboxamides in a Multicomponent Reaction
2020-02-13
1
Engineered Biosynthesis of 5/5/6 Type Polycyclic Tetramate Macrolactams in an Ikarugamycin (5/6/5 Type)-Producing Chassis
2020-02-13
1
Photocatalytic C–F Bond Borylation of Polyfluoroarenes with NHC-boranes
2020-02-13
1
Syntheses of Epoxyguaiane Sesquiterpenes (−)-Englerin A, (−)-Oxyphyllol, (+)-Orientalol E, and (+)-Orientalol F: A Synthetic Biology Approach
2020-02-13
1
Enhanced DNA Sensing and Chiroptical Performance by Restriction of Double-Bond Rotation of AIE cis-Tetraphenylethylene Macrocycle Diammoniums
2020-02-12
1
Total Synthesis of Dysoxylactam A
2020-02-12
1
A Pd-Catalyzed Site-Controlled Isomerization of Terminal Olefins
2020-02-11
0.88
Copper-Catalyzed Annulation or Homocoupling of Sulfoxonium Ylides: Synthesis of 2,3-Diaroylquinolines or α,α,β-Tricarbonyl Sulfoxonium Ylides
2020-02-11
1
Aspermeroterpenes A–C: Three Meroterpenoids from the Marine-Derived Fungus Aspergillus terreus GZU-31-1
2020-02-10
1
Asymmetric Synthesis of Rugulotrosin A
2020-02-10
1
Asymmetric Total Synthesis of (−)-Guignardones A and B
2020-02-10
1
Synthesis of 17-Deacetoxyl Chromodorolide B Based on a Gold-Catalyzed Alkoxycyclization Reaction
2020-02-10
1
Synthesis, Properties, and Reactivity of Bis-BN Phenanthrenes: Stepwise Bromination of the Main Scaffold
2020-02-10
1
Visible-Light-Induced Charge Transfer Enables Csp3–H Functionalization of Glycine Derivatives: Access to 1,3-Oxazolidines
2020-02-10
1
Copper-Catalyzed Oxidative Thioamination of Maleimides with Amines and Bunte Salts
2020-02-07
1
Efficient Strategy for α-Selective Glycosidation of d-Glucosamine and Its Application to the Synthesis of a Bacterial Capsular Polysaccharide Repeating Unit Containing Multiple α-Linked GlcNAc Residues
2020-02-07
0.80
Copper-Catalyzed Photoinduced Enantioselective Dual Carbofunctionalization of Alkenes
2020-02-06
1
Origins of Unconventional γ Site Selectivity in Palladium-Catalyzed C(sp3)–H Activation and Arylation of Aliphatic Alcohols
2020-02-06
1
Rhodium-Catalyzed Remote Isomerization of Alkenyl Alcohols to Ketones
2020-02-06
1
Catalytic Asymmetric Conjugate Protosilylation and Protoborylation of 2-Trifluoromethyl Enynes for Synthesis of Functionalized Allenes
2020-02-04
1
Cu-Mediated Expeditious Annulation of Alkyl 3-Aminoacrylates with Aryldiazonium Salts: Access to Alkyl N2-Aryl 1,2,3-Triazole-carboxylates for Druglike Molecular Synthesis
2020-02-04
1
Homoleptic Bis(trimethylsilyl)amides of Yttrium Complexes Catalyzed Hydroboration Reduction of Amides to Amines
2020-02-04
1
Synergistic Dual Directing Groups-Enabled Diastereoselective C–H Cyclopropylation via Rh(III)-Catalyzed Couplings with Cyclopropenyl Alcohols
2020-02-04
1
Access to Divergent Fluorinated Enynes and Arenes via Palladium-Catalyzed Ring-Opening Alkynylation of gem-Difluorinated Cyclopropanes
2020-02-03
1
Aldehyde as a Traceless Directing Group for Regioselective C–H Alkylation Catalyzed by Rhodium(III) in Air
2020-02-03
0.83
Covalent Organic Framework as a Heterogeneous Ligand for the Regioselective Oxidative Heck Reaction
2020-02-03
1
Enantioselective Synthesis of 4-Allyl Tetrahydroquinolines via Copper(I) Hydride-Catalyzed Hydroallylation of 1,2-Dihydroquinolines
2020-02-03
1
Late-Stage Modification of Tertiary Phosphines via Ruthenium(II)-Catalyzed C–H Alkylation
2020-02-03
0.90
Layered Chirality Relay Model in Rh(I)-Mediated Enantioselective C–Si Bond Activation: A Theoretical Study
2020-02-03
1
Rhodium(III)-Catalyzed C–H Alkenylation: Access to Maleimide-Decorated Tryptophan and Tryptophan-Containing Peptides
2020-02-03
1
Host–Guest Complexation of Perethylated Pillar[6]arene toward Ferrocene Derivatives Both in Solution and Solid State: Different Binding Modes Induced by Minor Structural Changes of Guests
2020-01-31
1
Total Syntheses of (+)-Stemarin and the Proposed Structures of Stemara-13(14)-en-18-ol and Stemara-13(14)-en-17-acetoxy-18-ol
2020-01-31
1
Dehydrative Cross-Coupling of Allylic Alcohols with Alkynes
2020-01-30
0.97
Enantioselective Cu(I)-Catalyzed Cycloaddition of Prochiral Diazides with Terminal or 1-Iodoalkynes
2020-01-30
1
Energetic Derivatives of 8-Nitropyrazolo[1,5-a][1,3,5]triazine-2,4,7-triamine: Achieving Balanced Explosives by Fusing Pyrazole with Triazine
2020-01-30
0.33
Intramolecular Aromatic C–H Acyloxylation Enabled by Iron Photocatalysis
2020-01-30
1
Melipatulinones A–C, Three Lignan–Phloroglucinol Hybrids from Melicope patulinervia
2020-01-30
1
Synthesis of Functionalized Vinylsilanes via Metal-Free Dehydrogenative Silylation of Enamides
2020-01-30
1
Synthesis of Multifunctional 2-Aminobenzimidazoles on DNA via Iodine-Promoted Cyclization
2020-01-30
0.70
Genome Mining and Biosynthesis of Primary Amine-Acylated Desferrioxamines in a Marine Gliding Bacterium
2020-01-29
1
Access to Benzoxazepines and Fully Substituted Indoles via HDDA Coupling
2020-01-28
1
Continuous Flow-Enabled Synthesis of Bench-Stable Bicyclo[1.1.1]pentane Trifluoroborate Salts and Their Utilization in Metallaphotoredox Cross-Couplings
2020-01-28
0.36
Enantioselective Imino-Ene Reaction of N-Sulfonyl Ketimines with Silyl Enol Ethers: Access to Chiral Benzosultams
2020-01-28
1
Enantioselective Synthesis of Spiroindolines via Cascade Isomerization/Spirocyclization/Dearomatization Reaction
2020-01-28
1
Synthesis of Monofluoroalkenes through Visible-Light-Promoted Defluorinative Alkylation of gem-Difluoroalkenes with 4-Alkyl-1,4-dihydropyridines
2020-01-28
1
Harnessing Thiol as a Benzyl Reagent for Photocatalytic Reductive Benzylation of Imines
2020-01-27
0.50
Radical Aza-Cyclization of α-Imino-oxy Acids for Synthesis of Alkene-Containing N-Heterocycles via Dual Cobaloxime and Photoredox Catalysis
2020-01-27
1
Copper-Catalyzed Asymmetric Propargylic Alkylation with Oxindoles: Diastereo- and Enantioselective Construction of Vicinal Tertiary and All-Carbon Quaternary Stereocenters
2020-01-24
1
Fulleropillar[4]arene: The Synthesis and Complexation Properties
2020-01-24
1
Merging Visible Light Photocatalysis and l-/d-Proline Catalysis: Direct Asymmetric Oxidative Dearomatization of 2-Arylindoles To Access C2-Quaternary Indolin-3-ones
2020-01-24
1
Morindolestatin, Naturally Occurring Dehydromorpholinocarbazole Alkaloid from Soil-Derived Bacterium of the Genus Streptomyces
2020-01-24
1
Remote Directed Isocyanation of Unactivated C(sp3)–H Bonds: Forging Seven-Membered Cyclic Ureas Enabled by Copper Catalysis
2020-01-24
1
Ruthenium Carbene-Mediated Construction of Strained Allenes via the Enyne Cross-Metathesis/Cyclopropanation of 1,6-Enynes
2020-01-24
1
Synthesis of Stereodefined Trisubstituted Alkenyl Silanes Enabled by Borane Catalysis and Nickel Catalysis
2020-01-24
1
Catalytic Diastereoselective [5 + 2] Annulation of N-Acryloyl Indoles with Cyclic Sulfonyl Enamides: Facile Access to Isoeburnamonine
2020-01-23
1
Heterologous Expression Leads to Discovery of Diversified Lobophorin Analogues and a Flexible Glycosyltransferase
2020-01-23
1
Open-Air Stereoselective Construction of C-Aryl Glycosides
2020-01-23
0.88
Regioselective Wacker-Type Oxidation of Internal Olefins in tBuOH Using Oxygen as the Sole Oxidant and tBuONO as the Organic Redox Cocatalyst
2020-01-23
1
Selective Dehydrogenative Acylation of Enamides with Aldehydes Leading to Valuable β-Ketoenamides
2020-01-23
0.93
Synthesis of 4,7-Difunctionalized Indoles via Imino Exchange and Sulfinyl Migration
2020-01-23
1
Visible-Light-Promoted Photocatalyst-Free Hydroacylation and Diacylation of Alkenes Tuned by NiCl2·DME
2020-01-23
1
Organocatalytic Cascade β-Functionalization/Aromatization of Pyrrolidines via Double Hydride Transfer
2020-01-22
1
Palladium-Catalyzed Carbonylative Synthesis of α-Branched Enones from Aryl Iodides and Arylallenes
2020-01-22
0.88
Practical Method for Reductive Deuteration of Ketones with Magnesium and D2O
2020-01-22
1
Biomimetic Total Syntheses of Sanctis A–B with Structure Revision
2020-01-21
1
Cu(I)-Catalyzed Enantioselective Alkynylation of Thiochromones
2020-01-21
1
Iridium-Catalyzed Asymmetric Hydrogenation of γ- and δ-Ketoacids for Enantioselective Synthesis of γ- and δ-Lactones
2020-01-21
1
Nickel-Catalyzed Deaminative Acylation of Activated Aliphatic Amines with Aromatic Amides via C–N Bond Activation
2020-01-21
0.83
Catalytic Asymmetric Tandem Cycloisomerization/[5+2] Cycloaddition Reaction of N-Aryl Nitrone Alkynes with Methyleneindolinones
2020-01-17
1
Photo/N-Heterocyclic Carbene Co-catalyzed Ring Opening and γ-Alkylation of Cyclopropane Enal
2020-01-17
1
Regioselective Synthesis of 3-Trifluoromethylpyrazole by Coupling of Aldehydes, Sulfonyl Hydrazides, and 2-Bromo-3,3,3-trifluoropropene
2020-01-17
1
Cobalt-Catalyzed Z to E Isomerization of Alkenes: An Approach to (E)-β-Substituted Styrenes
2020-01-16
1
Metal-Free sp3 C-SCF3 Coupling Reactions between Cycloketone Oxime Esters and S-trifluoromethyl 4-Methylbenzenesulfonothioate
2020-01-16
1
Photoinduced C(sp2)–H/C(sp2)–H Cross-Coupling of Alkenes: Direct Synthesis of 1,3-Dienes
2020-01-16
1
Reverse Turn Foldamers: An Expanded β-Turn Motif Reinforced by Double Hydrogen Bonds
2020-01-16
0.43
Rhodium-Catalyzed ortho-Selective Carbene C–H Insertion of Unprotected Phenols Directed by a Transient Oxonium Ylide Intermediate
2020-01-16
1
Synthesis of Difluoroalkylated Benzofuran, Benzothiophene, and Indole Derivatives via Palladium-Catalyzed Cascade Difluoroalkylation and Arylation of 1,6-Enynes
2020-01-16
1
[3,3]-Sigmatropic Rearrangement/Haller–Bauer Reaction of Aryl Sulfoxides and Selenoxides with Difluoroenoxysilanes: Access to CF2H-Containing Chalcogenides
2020-01-16
1
Asymmetric Umpolung Hydrogenation and Deuteration of Alkenes Catalyzed by Nickel
2020-01-15
0.67
Enantioselective Synthesis of Spirorhodanine-Pyran Derivatives via Organocatalytic [3 + 3] Annulation Reactions between Pyrazolones and Rhodanine-Derived Ketoesters
2020-01-15
1
Incarnolides A and B, Two Schinortriterpenoids with a Tricyclo[9.2.1.02,8]tetradecane-Bridged System from Schisandra incarnata
2020-01-15
1
Tunable Gold(I)-Catalyzed [4 + 3] Cycloaddition for Divergent Synthesis of Furan-Fused N,O-Heterocycles
2020-01-15
1
Electrochemical Oxidative Oxydihalogenation of Alkynes for the Synthesis of α,α-Dihaloketones
2020-01-14
1
Palladium-Catalyzed Ligand-Free Double Cyclization Reactions for the Synthesis of 3-(1′-Indolyl)-phthalides
2020-01-14
1
Rhodium-Catalyzed Enantioselective Anti-Markovnikov Hydroformylation of α-Substituted Acryl Acid Derivatives
2020-01-14
1
Synthesis of Tertiary Benzylic Nitriles via Nickel-Catalyzed Markovnikov Hydrocyanation of α-Substituted Styrenes
2020-01-14
1
C- to N-Center Remote Heteroaryl Migration via Electrochemical Initiation of N Radical by Organic Catalyst
2020-01-10
1
Nickel-Catalyzed, para-Selective, Radical-Based Alkylation of Aromatic Ketones
2020-01-10
1
Chalcone-Based Pyridinium Salts and Their Diastereoselective Dearomatization To Access Bibridged Benzoazepines
2020-01-09
1
Cobalt-Catalyzed Migrational Isomerization of Styrenes
2020-01-09
1
Copper-Catalyzed Asymmetric Hydrosilylation of β-Nitroethyl Aryl Ketones
2020-01-09
1
Crokonoids A–C, A Highly Rearranged and Dual-Bridged Spiro Diterpenoid and Two Other Diterpenoids from Croton kongensis
2020-01-09
1
Dimethylformamide-Modulated Kdo Glycosylation for Stereoselective Synthesis of α-Kdo Glycosides
2020-01-09
1
Photoredox Oxo-C(sp3)–H Bond Functionalization via in Situ Cu(I)-Acetylide Catalysis
2020-01-09
1
Reductase of Mutanobactin Synthetase Triggers Sequential C–C Macrocyclization, C–S Bond Formation, and C–C Bond Cleavage
2020-01-09
1
Rh-Catalyzed Asymmetric Hydrogenation of Unsaturated Medium-Ring NH Lactams: Highly Enantioselective Synthesis of N-Unprotected 2,3-Dihydro-1,5-benzothiazepinones
2020-01-09
1
CF3SO2Na-Mediated, UV-Light-Induced Friedel–Crafts Alkylation of Indoles with Ketones/Aldehydes and Bioactivities of Products
2020-01-08
1
Chiral Discrimination of Varied Ammonium Compounds through 1H NMR Using a Binuclear Ti Complex Sensor
2020-01-08
1
DFT Mechanistic Account for the Site Selectivity of Electron-Rich C(sp3)–H Bond in the Manganese-Catalyzed Aminations
2020-01-08
1
Enantioselective NHC-Catalyzed [3+3] Annulation of α-Bromoenals with 2-Aminobenzimidazoles
2020-01-08
1
Intermolecular Reductive Heck Reaction of Unactivated Aliphatic Alkenes with Organohalides
2020-01-08
0.95
Nickel-Catalyzed Asymmetric Hydrocyanation of Allenes
2020-01-08
1
Pentafluorophenyl Esters: Highly Chemoselective Ketyl Precursors for the Synthesis of α,α-Dideuterio Alcohols Using SmI2 and D2O as a Deuterium Source
2020-01-08
0.63
C–H Insertion by Alkylidene Carbenes To Form 1,2,3-Triazines and Anionic [3 + 2] Dipolar Cycloadditions To Form Tetrazoles: Crucial Roles of Stereoelectronic and Steric Effects
2020-01-07
0.50
Heterogeneous Carbon Nitrides Photocatalysis Multicomponent Hydrosulfonylation of Alkynes To Access β-Keto Sulfones with the Insertion of Sulfur Dioxide in Aerobic Aqueous Medium
2020-01-07
1
Palladium-Catalyzed Synthesis of 1,2-Diketones from Aryl Halides and Organoaluminum Reagents Using tert-Butyl Isocyanide as the CO Source
2020-01-07
0.50
Precise Construction of SCF2H or SeCF2H Groups on Heteroarenes Generated in Situ from CF3-Containing 1,3-Enynes
2020-01-07
1
Revision of the Structure of Hypatulone A by NMR, Computations, and Biosynthetic Considerations
2020-01-07
0.50
Visible-Light-Driven Dearomatization Reaction toward the Formation of Spiro[4.5]deca-1,6,9-trien-8-ones
2020-01-07
1
Visible-Light-Induced Deoxygenation/Defluorination Protocol for Synthesis of γ,γ-Difluoroallylic Ketones
2020-01-07
1
Asymmetric Total Synthesis and Biological Evaluation of the Natural PDE4 Inhibitor Toddacoumalone
2020-01-06
1
Lewis Acid Catalyzed Electrophilic Aminomethyloxygenative Cyclization of Alkynols with N,O-Aminals
2020-01-06
1
NHC-Catalyzed Radical Trifluoromethylation Enabled by Togni Reagent
2020-01-06
1
Synthesis of Tribenzo[b,d,f]azepines via Cascade π-Extended Decarboxylative Annulation Involving Cyclic Diaryliodonium Salts
2020-01-06
1
Total Synthesis of Galanthamine and Lycoramine Featuring an Early-Stage C–C and a Late-Stage Dehydrogenation via C–H Activation
2020-01-06
1
Construction of 2-Arylbenzo[4,5]thieno[2,3-d]thiazole Skeleton via CuCl/S-Mediated Three-Component Reaction
2020-01-02
0.90
Pd-Catalyzed Asymmetric Hydroalkylation of 1,3-Dienes: Access to Unnatural α-Amino Acid Derivatives Containing Vicinal Quaternary and Tertiary Stereogenic Centers
2020-01-02
1
Rh(III)-Catalyzed Tandem Acylmethylation/Nitroso Migration/Cyclization of N-Nitrosoanilines with Sulfoxonium Ylides in One Pot: Approach to 3-Nitrosoindoles
2020-01-02
1
Enantioselective Synthesis of Multifunctionalized 4H-Pyrans via Formal [4 + 2] Annulation Process by Bifunctional Phosphonium Salt Catalysis
2019-12-31
1
Genetic Manipulation of an Aminotransferase Family Gene dtlA Activates Youssoufenes in Marine-Derived Streptomyces youssoufiensis
2019-12-31
1
Silver-Catalyzed Selective Multicomponent Coupling Reactions of Arynes with Nitriles and Isonitriles
2019-12-31
0.40
CuSO4-Catalyzed Tandem C(sp3)–H Insertion Cyclization of Toluenes with Isonitriles to Form Indoles
2019-12-30
1
Electrochemical Synthesis of 1-Naphthols by Intermolecular Annulation of Alkynes with 1,3-Dicarbonyl Compounds
2019-12-30
1
Practical Synthesis of Benzimidazo[1,2-a]quinolines via Rh(III)-Catalyzed C–H Activation Cascade Reaction from Imidamides and Anthranils
2019-12-30
1
Rh(III)-Catalyzed Coupling of Acrylic Acids and Ynenones via Olefinic C–H Activation and Michael Addition
2019-12-30
1
Silver-Catalyzed Annulation of Arynes with Nitriles for Synthesis of Structurally Diverse Quinazolines
2019-12-30
0.40
Synthesis of 2H-Chromenes via Unexpected [4 + 2] Annulation of Alkynyl Thioethers with o-Hydroxybenzyl Alcohols
2019-12-30
1
Botryotins A–H, Tetracyclic Diterpenoids Representing Three Carbon Skeletons from a Deep-Sea-Derived Botryotinia fuckeliana
2019-12-27
1
Enantioselective 1,2-Alkylhydroxylmethylation of Alkynes via Chromium/Cobalt Cocatalysis
2019-12-27
1
Organocatalytic Double Ugi Reaction with Statistical Amplification of Product Enantiopurity: A Linker Cleavage Approach To Access Highly Enantiopure Ugi Products
2019-12-27
0.75
Synthesis of 2-Arylpiperidines via Pd-Catalyzed Arylation of Aza-Achmatowicz Rearrangement Products with Arylboronic Acids
2019-12-27
0.29
Highly Enantioselective Nickel-Catalyzed Hydrocyanation of Disubstituted Methylenecyclopropanes Enabled by TADDOL-based Diphosphite Ligands
2019-12-26
1
Total Synthesis of Caesalpinnone A
2019-12-26
1
Herpotrichones A and B, Two Intermolecular [4 + 2] Adducts with Anti-Neuroinflammatory Activity from a Herpotrichia Species
2019-12-24
0.78
Mechanistic Insights into La-Catalyzed Amidation of Aldehyde with Amine
2019-12-24
1
Phosphine-Catalyzed (3 + 2)/(3 + 2) Sequential Annulation of γ-Vinyl Allenoates: Access to Fused Carbocycles
2019-12-24
1
Phosphine-Mediated MBH-Type/Umpolung Addition Domino Sequence: Divergent Construction of Coumarins
2019-12-24
1
Probing the Interconversion of Labdane Lactones from the Chinese Liverwort Pallavicinia ambigua
2019-12-24
1
Complementary C–H Functionalization Mode of Benzoylacetonitriles: Computer-Augmented Study of a Regio- and Stereoselective Synthesis of Functionalized Benzofulvenes
2019-12-23
0.60
Enantioselective Synthesis of Fused Polycyclic Tropanes via Dearomative [3 + 2] Cycloaddition Reactions of 2-Nitrobenzofurans
2019-12-23
1
Palladium-Catalyzed Cascade Reactions of 2-(Cyanomethoxy)chalcones with Arylboronic Acids: Selective Synthesis of Emissive Benzofuro[2,3-c]pyridines
2019-12-23
1
Benzene-1,3,5-triyl Triformate (TFBen)-Promoted Palladium-Catalyzed Carbonylative Synthesis of 2-Oxo-2,5-dihydropyrroles from Propargyl Amines
2019-12-20
0.83
Direct Use of Unprotected Aliphatic Amines to Generate N-Heterocycles via β-C–H Malonylation with Iodonium Ylide
2019-12-20
1
Employing TosMIC as a C1N1 “Two-Atom Synthon” in Imidazole Synthesis by Neighboring Group Assistance Strategy
2019-12-20
1
Exploring Aporphine as Anti-inflammatory and Analgesic Lead from Dactylicapnos scandens
2019-12-20
1
Selective Insertion of Alkynes into C–C σ Bonds of Indolin-2-ones: Transition-Metal-Free Ring Expansion Reactions to Seven-Membered-Ring Benzolactams or Chromone Derivatives
2019-12-20
1
π-Extended C2-Symmetric Double NBN-Heterohelicenes with Exceptional Luminescent Properties
2019-12-20
1
Cu-Catalyzed Alkylarylation of Vinylarenes with Masked Alkyl Electrophiles
2019-12-19
1
On-Resin Passerini Reaction toward C-Terminal Photocaged Peptides
2019-12-19
1
Visible-Light-Induced para-Selective C(sp2)–H Difluoroalkylation of Diverse (Hetero)aromatic Carbonyls
2019-12-19
1
Decarboxylative Borylation of mCPBA-Activated Aliphatic Acids
2019-12-18
1
Highly Enantioselective Construction of Dihydrooxazines via Pd-Catalyzed Asymmetric Carboetherification
2019-12-18
1
Palladium and Brønsted Acid Co-Catalyzed Biginelli-like Multicomponent Reactions via in Situ-Generated Cyclic Enol Ether: Access to Spirofuran-hydropyrimidinones
2019-12-18
1
Stable Double and Quadruple [5]Helicene Derivatives: Synthesis, Structural Analysis, and Physical Properties
2019-12-18
1
Desymmetrization of Prochiral Cyclopentenes Enabled by Enantioselective Palladium-Catalyzed Oxidative Heck Reaction
2019-12-17
0.25
Palladium-Catalyzed Three-Component Tandem Coupling–Carboannulation Reaction Leading to Polysubstituted [60]Fullerene-Fused Cyclopentanes
2019-12-17
1
2,3-Dicyano-5,6-dichlorobenzoquinone-Mediated and Selective C–O and C–C Cross-Couplings of Phenols and Porphyrins
2019-12-16
1
Alkaline-Earth Metal Catalyzed Dehydrative Allylic Alkylation
2019-12-16
0.95
Catalytic Enantioselective Synthesis of 1,4-Benzodioxepines
2019-12-16
1
Chiral ScIII–N,N′-Dioxide-Catalyzed 1,3-Dipolar Cycloaddition of Diaziridines with Chalcones
2019-12-13
1
Enantio- and Diastereoselective Synthesis of Chromeno[4,3-b]pyrrole Derivatives Bearing Tetrasubstituted Chirality Centers through Carbene Catalyzed Cascade Reactions
2019-12-13
0.86
Formation of Terrestric Acid in Penicillium crustosum Requires Redox-Assisted Decarboxylation and Stereoisomerization
2019-12-13
0.20
Pd(II)-Catalyzed Regioselective Multiple C–H Arylations of 1-Naphthamides with Cyclic Diaryliodonium Salts: One-Step Access to [4]- and [5]Carbohelicenes
2019-12-13
1
RhIII-Catalyzed Synthesis of Cyclopenta[b]carbazoles via Cascade C–H/C–C Bond Cleavage and Cyclization Reactions: Using Amide as a Traceless Directing Group
2019-12-13
1
Construction of Bisindolines via Oxidative Coupling Cyclization
2019-12-12
1
Copper(II)-Catalyzed C-H Nitrogenation/Annulation Cascade of Ketene N,S-Acetals with Aryldiazonium Salts: A Direct Access to N2-Substituted Triazole and Triazine Derivatives
2019-12-12
1
Detoxification of Plant Aromatic Abietanoids via Cleavage of the Benzene Ring into 11,12-Seco-diterpene Polyenes by a Specialist Insect of Leucosceptrum canum
2019-12-12
1
Directed Biosynthesis of Iso-aclacinomycins with Improved Anticancer Activity
2019-12-12
1
Electrochemically Enabled Double C–H Activation of Amides: Chemoselective Synthesis of Polycyclic Isoquinolinones
2019-12-12
1
Jatrofolianes A and B: Two Highly Modified Lathyrane Diterpenoids from Jatropha gossypiifolia
2019-12-12
1
Preparation of 4-Diazoisoquinolin-3-ones via Dimroth Rearrangement and Their Extension to 4-Aryltetrahydroisoquinolin-3-ones
2019-12-12
1
Structural Revision and Absolute Configuration of Burnettramic Acid A
2019-12-12
1
Synthesis and Semiconducting Characteristics of the BF2 Complexes of Bisbenzothiophene-Fused Azadipyrromethenes
2019-12-12
1
(3 + 1) Annulation/Rearrangement Cascade of C,N-Cyclic Azomethine Imines and 3-Chlorooxindoles: Construction of Hexahydroindeno[2,1-c]pyrazole Spirooxindole Frameworks
2019-12-11
1
Base-Promoted Nitrile–Alkyne Domino-Type Cyclization: A General Method to Trisubstituted Imidazoles
2019-12-10
1
Chiral Bis(oxazoline)–Copper Complex Catalyzed Asymmetric Alkenylation of Isatin Imines and 3-Vinylindoles for Construction of Optically Active 3-Alkenyl-3-aminooxindoles
2019-12-10
1
Diastereo- and Enantioselective Synthesis of Quaternary α-Amino Acid Precursors by Copper-Catalyzed Propargylation
2019-12-10
1
Selectfluor-Mediated Stereoselective [1 + 1 + 4 + 4] Dimerization of Styrylnaphthols
2019-12-10
1
A Tetraazapentacene–Pyrene Belt: Toward Synthesis of N-Doped Zigzag Carbon Nanobelts
2019-12-09
1
Cp*RhIII-Catalyzed Sulfonamide-Directed Ortho Arene C–H Carbenoid Functionalization with Pyridotriazoles
2019-12-09
1
Palladium-Catalyzed Domino Heck/C–H Activation/Decarboxylation: A Rapid Entry to Fused Isoquinolinediones and Isoquinolinones
2019-12-09
1
Regiodivergent Vinylogous–Cyclization Reactions of Cyclic α-Amide Enone Acceptors: Synthesis of Highly Enantioenriched Heterobicyclic Structures
2019-12-09
1
Catalytic Direct Regioselective Synthesis of Phosphonylated Tetrazoles from Aryl Diazonium Salts and Seyferth-Gilbert Reagent
2019-12-06
1
Organic Photoredox-Catalyzed Decarboxylative Trifluoromethylselenolation of Aliphatic Carboxylic Acids with [Me4N][SeCF3]
2019-12-06
1
Pd(0)-Catalyzed Intramolecular “Ylide-Ullmann-Type” Cyclization of Carbonyl-Stabilized Phosphonium Ylides and Access to Phosphachromones by Exocyclic P–C Cleavage
2019-12-06
1
Visible-Light-Enabled Oxidative Coupling of Alkenes with Dialkylformamides To Access Unsaturated Amides
2019-12-06
1
Highly Diastereo- and Enantioselective Ir-Catalyzed Hydrogenation of 2,3-Disubstituted Quinolines with Structurally Fine-Tuned Phosphine–Phosphoramidite Ligands
2019-12-05
1
Redox-Neutral [4 + 2] Annulation of N-Methoxybenzamides with Alkynes Enabled by an Osmium(II)/HOAc Catalytic System
2019-12-05
1
Copper-Catalyzed Cascade Cyclization Reaction of Enamines and Electron-Deficient Terminal Alkynes: Synthesis of Polysubstituted Pyrido[1,2-a]indoles
2019-12-04
1
Copper-Mediated Direct Cyanation of Heteroarene and Arene C–H Bonds by the Combination of Ammonium and DMF
2019-12-04
1
Coupling of Trifluoroacetaldehyde N-Triftosylhydrazone with Organoboronic Acids for the Synthesis of gem-Difluoroalkenes
2019-12-04
1
Ruthenium-Catalyzed ortho- and meta-H/D Exchange of Arenes
2019-12-04
1
Access to 2-Aroylthienothiazoles via C–H/N–O Bond Functionalization of Oximes
2019-12-03
1
Access to Functionalized E-Allylsilanes and E-Alkenylsilanes through Visible-Light-Driven Radical Hydrosilylation of Mono- and Disubstituted Allenes
2019-12-03
1
Blue Light Induced Difluoroalkylation of Alkynes and Alkenes
2019-12-03
1
Excitation Wavelength-Dependent Nearly Pure White Light-Emitting Crystals from a Single Gold(I)-Containing Complex
2019-12-03
1
Metal-Free Synthesis of 3-(Iso)quinolinyl 4-Chromenones and 3-(Iso)quinolinyl 4-Quinolones from (Iso)quinoline N-Oxides and Ynones
2019-12-03
1
Privilege-Structure-Oriented Three-Component Asymmetric Aminomethylation: Assembly of Chiral 3-Aminomethyl Indolones
2019-12-03
1
Regioselectivity-Switchable Catalytic Annulations of Alkynyl α-Diketones and α-Cyanoketones
2019-12-03
1
A Strategy for the Synthesis of Sulfonamides on DNA
2019-12-02
0.92
Gold-Catalyzed Intramolecular Dearomatization Reactions of Indoles for the Synthesis of Spiroindolenines and Spiroindolines
2019-12-02
0.75
Regioselective Synthesis and Crystallographic Characterization of Nontethered cis-1 and cis-2 Bis(benzofuro)[60]fullerene Derivatives
2019-12-02
1
A Direct Approach to Decoration of Bioactive Compounds via C–H Amination Reaction
2019-11-27
1
Cascade π-Extended Decarboxylative Annulation Involving Cyclic Diaryliodonium Salts: Site-Selective Synthesis of Phenanthridines and Benzocarbazoles via a Traceless Directing Group Strategy
2019-11-27
1
Photocatalytic Annulation–Alkynyl Migration Strategy for Multiple Functionalization of Dual Unactivated Alkenes
2019-11-26
1
Rhodium-Catalyzed Pyridine N-Oxide Assisted Suzuki–Miyaura Coupling Reaction via C(O)–C Bond Activation
2019-11-26
1
Synthesis of 3-HCF2S-Chromones through Tandem Oxa-Michael Addition and Oxidative Difluoromethylthiolation
2019-11-26
1
(−)- and (+)-Asperginulin A, a Pair of Indole Diketopiperazine Alkaloid Dimers with a 6/5/4/5/6 Pentacyclic Skeleton from the Mangrove Endophytic Fungus Aspergillus sp. SK-28
2019-11-25
1
Asymmetric Formal Vinylogous Iminium Ion Activation for Vinyl-Substituted Heteroaryl and Aryl Aldehydes
2019-11-25
0.83
One-Carbon Incorporation Using Cyclobutanone Oxime Ester Enabled [2 + 2 + 1] Carboannulation of 1,7-Enynes by C–C/N–O Bond Cleavage and C–H Functionalization
2019-11-25
1
Pd-Catalyzed Enantioselective Double Heck Reaction
2019-11-25
1
Rhodium-Catalyzed Successive C–H Bond Functionalizations To Synthesize Complex Indenols Bearing a Benzofuran Unit
2019-11-25
1
Transformation of Alkynes into α- or β-Difluorinated Alkyl Azides by an Efficient One-Pot Two-Step Procedure
2019-11-25
1
Asymmetric Allylic Etherification of Vinylethylene Carbonates with Diols via Pd/B Cooperative Catalysis: A Route to Chiral Hemi-Crown Ethers
2019-11-22
1
Cleistocaltones A and B, Antiviral Phloroglucinol–Terpenoid Adducts from Cleistocalyx operculatus
2019-11-22
1
Copper-Mediated Deacylative Coupling of Ynones via C–C Bond Activation under Mild Conditions
2019-11-22
1
Redox-Neutral Borylation of Aryl Sulfonium Salts via C–S Activation Enabled by Light
2019-11-22
1
Agelanemoechine, a Dimeric Bromopyrrole Alkaloid with a Pro-Angiogenic Effect from the South China Sea Sponge Agelas nemoechinata
2019-11-20
0.90
An Approach to Peri-Fused Heterocycles: A Metal-Mediated Cascade Carbonylative Cyclization/Dearomatic Diels–Alder Reaction
2019-11-20
1
Asymmetric Total Synthesis Enables Discovery of Antibacterial Activity of Siladenoserinols A and H
2019-11-20
1
Chiral Spiro Phosphoramide-Catalyzed Sulfa-Michael Addition/Enantioselective Protonation of Exocyclic Enones
2019-11-20
1
Direct Catalytic Asymmetric Synthesis of Oxindole-Derived δ-Hydroxy-β-ketoesters by Aldol Reactions
2019-11-20
0.78
Divergent Reactivity in CuII-Catalyzed Oxidative Coupling between Indole/Tryptamine Derivatives and β-Arylacrylic Acids
2019-11-20
1
Electrochemical Synthesis of trans-2,3-Disubstituted Aziridines via Oxidative Dehydrogenative Intramolecular C(sp3)–H Amination
2019-11-20
1
Enantioselective Radical Ring-Opening Cyanation of Oxime Esters by Dual Photoredox and Copper Catalysis
2019-11-20
1
Gold(I)-Catalyzed Glycosylation with Glycosyl Ynenoates as Donors
2019-11-20
1
Morusalones A–D, Diels–Alder Adducts with 6/7/6/6/6/6 Hexacyclic Ring Systems as Potential PTP1B Inhibitors from Cell Cultures of Morus alba
2019-11-20
1
One-Pot Enantioselective Synthesis of 2-Pyrrolidinone Derivatives Bearing a Trifluoromethylated All-Carbon Quaternary Stereocenter
2019-11-20
1
Oxalic Acid Monothioester for Palladium-Catalyzed Decarboxylative Thiocarbonylation and Hydrothiocarbonylation
2019-11-20
0.83
Synthesis of Heterocyclic Core-Expanded Bis-Naphthalene Tetracarboxylic Diimides
2019-11-20
1
Carbene-Catalyzed Enantioselective Addition of Thioamides to Bromoenals for Access to Thiazinone Heterocycles
2019-11-19
0.83
Lewis-Acid-Mediated Thiocyano Semipinacol Rearrangement of Allylic Alcohols for Construction of α-Quaternary Center β-Thiocyano Carbonyls
2019-11-19
1
Ligand-Controlled Regiodivergent Silylation of Allylic Alcohols by Ni/Cu Catalysis for the Synthesis of Functionalized Allylsilanes
2019-11-19
1
Visible Light-Induced Amide Bond Formation
2019-11-19
1
Divergent Synthesis of Isoquinolone and Isocoumarin Derivatives by the Annulation of Benzoic Acid with N-Vinyl Amide
2019-11-18
1
Oxidative Hydro-, Bromo-, and Chloroheptafluoroisopropylation of Unactivated Alkenes with Heptafluoroisopropyl Silver
2019-11-18
1
Site-Selective Modification of α-Amino Acids and Oligopeptides via Native Amine-Directed γ-C(sp3)-H Arylation
2019-11-18
1
Asymmetric Conjugate Addition of Ethylene Sulfonyl Fluorides to 3-Amido-2-oxindoles: Synthesis of Chiral Spirocyclic Oxindole Sultams
2019-11-14
1
Construction of Multiple-Substituted Chiral Cyclohexanes through Hydrogenative Desymmetrization of 2,2,5-Trisubstituted 1,3-Cyclohexanediones
2019-11-14
1
LiHMDS-Promoted Palladium-Catalyzed Sonogashira Cross-Coupling of Aryl Fluorides with Terminal Alkynes
2019-11-14
1
N-Methoxyamide: An Alternative Amidation Reagent in the Rhodium(III)-Catalyzed C–H Activation
2019-11-14
1
Nickel-Catalyzed Transformation of Diazoacetates to Alkyl Radicals Using Alcohol as a Hydrogen Source
2019-11-14
1
Palladium-Catalyzed Controllable Reductive/Oxidative Heck Coupling between Cyclic Enones and Thiophenes via C–H Activation
2019-11-14
1
Synthesis of Oxadiazolones with Hydrazides: The Mechanism and the Sensing Application as Sensitive, Rapid, and Visual Fluorescent Sensors for Phosgene
2019-11-13
1
Access to Stereodefined (E)-2-Silylallylboronates via Regioselective Chloroboration of Allenylsilanes
2019-11-12
1
Ni-Catalyzed Intermolecular Allylic Dearomatization Reaction of Tryptophols and Tryptamines
2019-11-12
1
Spiroalanfurantones A–D, Four Eudesmanolide–Furan Sesquiterpene Adducts with a Pentacyclic 6/6/5/5/5 Skeleton from Inula helenium
2019-11-12
1
Synthesis of Isoxazolines and Oxazines by Electrochemical Intermolecular [2 + 1 + n] Annulation: Diazo Compounds Act as Radical Acceptors
2019-11-12
1
Copper-Catalyzed Cascade Cyclization of Arylsulfonylhydrazones Derived from ortho-Alkynyl Arylketones: Regioselective Synthesis of Functionalized Cinnolines
2019-11-11
1
Copper-Catalyzed Tandem Cross-Coupling/[2 + 2] Cycloaddition of 1,6-Allenynes with Diazo Compounds to 3-Azabicyclo[5.2.0] Ring Systems
2019-11-11
1
Cucurbit[8]uril-Mediated Polypseudorotaxane for Enhanced Lanthanide Luminescence Behavior in Water
2019-11-11
1
Direct Access to Allenylphosphine Oxides via a Metal Free Coupling of Propargylic Substrates with P(O)H Compounds
2019-11-11
1
Triarylborane-based [5]Helicenes with Full-Color Circularly Polarized Luminescence
2019-11-11
1
Pd(0)-Catalyzed Cyclizative Carboboration of n-Iodo-1,6-diene (n = 1 or 2): Access to Structurally Complex Allylboronates and Alkylboronates
2019-11-08
1
Pd-Catalyzed Asymmetric Allylic Cycloaddition of N-Containing Allylic Carbonates with Isocyanates
2019-11-08
1
Enantioselective Synthesis of Isoxazoline N-Oxides via Pd-Catalyzed Asymmetric Allylic Cycloaddition of Nitro-Containing Allylic Carbonates
2019-11-07
1
N-Alkylation-Initiated Redox-Neutral [5 + 2] Annulation of 3-Alkylindoles with o-Aminobenzaldehydes: Access to Indole-1,2-Fused 1,4-Benzodiazepines
2019-11-07
1
Total Synthesis of (+)-Jatrophalactam
2019-11-07
1
Gold-Catalyzed Highly Diastereoselective Oxy-Propargylamination of Allenamides with C-Alkynyl N-Boc N,O-Acetals
2019-11-06
1
Construction of Eight-Membered Cyclic Diaryl Sulfides via Domino Reaction of Arynes with Thioaurone Analogues and DFT Study on the Reaction Mechanism
2019-11-05
1
Hydrosulfonylation of Unactivated Alkenes by Visible Light Photoredox Catalysis
2019-11-05
1
Iridium-Catalyzed B–H Bond Insertion Reactions Using Sulfoxonium Ylides as Carbene Precursors toward α-Boryl Carbonyls
2019-11-05
1
Nickel-Catalyzed Reductive 1,2-Dialkynylation of Alkenes Bearing an 8-Aminoquinoline Directing Group
2019-11-05
1
Old Key Opens the Lock in Carborane: The in Situ NHC-Palladium Catalytic System for Selective Arylation of B(3,6)–H Bonds of o-Carboranes via B–H Activation
2019-11-05
1
Rhodium(III)-Catalyzed Annulative Coupling of Sulfoxonium Ylides and Allenoates: An Arene C–H Activation/Cyclopropanation Cascade
2019-11-05
1
Silver-Assisted Oxidative Isocyanide Insertion of Ethers: A Direct Approach to β-Carbonyl α-Iminonitriles
2019-11-05
1
Syntheses of Benzofuranoquinolines and Analogues via Photoinduced Acceptorless Dehydrogenative Annulation of o-Phenylfuranylpyridines
2019-11-05
1
Decarbonylative Phosphorylation of Carboxylic Acids via Redox-Neutral Palladium Catalysis
2019-11-04
0.40
Photoredox-Catalyzed Remote Difunctionalizations of Alkenes To Synthesize Fluoroalkyl Ketones with Dimethyl Sulfoxide as the Oxidant
2019-11-04
1
Pd(OAc)2-Catalyzed Asymmetric Hydrogenation of α-Iminoesters
2019-11-01
1
Switchable Synthesis of Aryl Sulfones and Sulfoxides through Solvent-Promoted Oxidation of Sulfides with O2/Air
2019-11-01
1
The Efficient Synthesis of Benzannulated Seven-Membered O-Heterocycles via the Intramolecular Ring-Opening Cyclization of Cyclopropanes
2019-11-01
1
Transition-Metal-Catalyzed Transformation of Sulfonates via S–O Bond Cleavage: Synthesis of Alkyl Aryl Ether and Diaryl Ether
2019-11-01
1
PLOS Biology 43 28.44
PLOS Genetics 57 39.10
Physical Review A 34 22.80
Physical Review B 147 95.13
Physical Review D 26 12.79
Physical Review Letters 548 326.08
Physical Review X 34 17.99
Proceedings of the National Academy of Sciences of the United States of America 478 258.87
Proceedings of the Royal Society B 39 22.73
Science 140 71.25
Science Advances 544 342.24
Science Translational Medicine 39 19.60
The Astrophysical Journal Letters 162 94.38
The EMBO Journal 49 38.78
The ISME Journal: Multidisciplinary Journal of Microbial Ecology 52 34.66
The Journal of Physical Chemistry Letters 497 400.72
The Plant Cell 88 70.54
Water Research 564 472.06
eLife 112 67.41

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